JP5596799B2 - カナグリフロジン含有錠剤 - Google Patents
カナグリフロジン含有錠剤 Download PDFInfo
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- JP5596799B2 JP5596799B2 JP2012551398A JP2012551398A JP5596799B2 JP 5596799 B2 JP5596799 B2 JP 5596799B2 JP 2012551398 A JP2012551398 A JP 2012551398A JP 2012551398 A JP2012551398 A JP 2012551398A JP 5596799 B2 JP5596799 B2 JP 5596799B2
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Landscapes
- Health & Medical Sciences (AREA)
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- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33331210P | 2010-05-11 | 2010-05-11 | |
| US61/333,312 | 2010-05-11 | ||
| PCT/JP2011/061354 WO2011142478A1 (fr) | 2010-05-11 | 2011-05-11 | Comprimés contenant de la canagliflozine |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013526482A JP2013526482A (ja) | 2013-06-24 |
| JP2013526482A5 JP2013526482A5 (fr) | 2013-12-26 |
| JP5596799B2 true JP5596799B2 (ja) | 2014-09-24 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012551398A Active JP5596799B2 (ja) | 2010-05-11 | 2011-05-11 | カナグリフロジン含有錠剤 |
Country Status (8)
| Country | Link |
|---|---|
| US (2) | US20130052266A1 (fr) |
| EP (1) | EP2568971B1 (fr) |
| JP (1) | JP5596799B2 (fr) |
| KR (1) | KR101869110B1 (fr) |
| CN (3) | CN106890147A (fr) |
| ES (1) | ES2836952T3 (fr) |
| TW (1) | TWI564034B (fr) |
| WO (1) | WO2011142478A1 (fr) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110009347A1 (en) | 2009-07-08 | 2011-01-13 | Yin Liang | Combination therapy for the treatment of diabetes |
| WO2014157603A1 (fr) | 2013-03-29 | 2014-10-02 | アステラス製薬株式会社 | Composition pharmaceutique pour administration orale |
| US20160083374A1 (en) * | 2013-05-30 | 2016-03-24 | Cadila Healthcare Limited | Amorphous form of canagliflozin and process for preparing thereof |
| CN103641822B (zh) * | 2013-10-21 | 2016-06-08 | 江苏奥赛康药业股份有限公司 | 一种卡格列净化合物及其药物组合物 |
| EP3068779A4 (fr) * | 2013-11-11 | 2017-06-28 | Crystal Pharmatech Co. Ltd. | Formes b, c et d cristallines de la canagliflozine |
| CN103655539B (zh) * | 2013-12-13 | 2019-09-13 | 重庆医药工业研究院有限责任公司 | 一种卡格列净的口服固体制剂及其制备方法 |
| US10174010B2 (en) | 2014-03-19 | 2019-01-08 | Hangzhou Pushai Pharmaceutical Technology Co., Ltd. | Canagliflozin monohydrate and its crystalline forms, preparation methods and uses thereof |
| CN103980262B (zh) * | 2014-04-01 | 2016-06-22 | 天津大学 | 卡格列净的b晶型及其结晶制备方法 |
| CN103980261B (zh) * | 2014-04-01 | 2016-06-29 | 天津大学 | 卡格列净的a晶型及其结晶制备方法 |
| EP2947077A1 (fr) | 2014-05-19 | 2015-11-25 | LEK Pharmaceuticals d.d. | Synthèse stéréosélective d'intermédiaires dans la préparation de ß-C-arylglucosides |
| KR20170008239A (ko) * | 2014-05-29 | 2017-01-23 | 노파르티스 아게 | 세리티닙 제제 |
| CN105330706B (zh) * | 2014-06-05 | 2019-04-16 | 江苏豪森药业集团有限公司 | 卡格列净中间体的制备方法 |
| US20160002275A1 (en) * | 2014-07-03 | 2016-01-07 | Cadila Healthcare Limited | Process for preparation and purification of canagliflozin |
| EP2990029A1 (fr) | 2014-08-29 | 2016-03-02 | Sandoz Ag | Compositions pharmaceutiques comprenant du canagliflozin |
| CN104402946B (zh) * | 2014-11-17 | 2018-01-02 | 连云港恒运药业有限公司 | 卡格列净中间体及其无定形的制备方法 |
| CN105769803A (zh) * | 2014-12-16 | 2016-07-20 | 康普药业股份有限公司 | 一种用于治疗2型糖尿病的药物组合物及其制备方法 |
| JP6027710B1 (ja) * | 2014-12-25 | 2016-11-16 | 田辺三菱製薬株式会社 | 糖尿病治療用固形製剤 |
| CN104523573A (zh) * | 2014-12-29 | 2015-04-22 | 成都恒瑞制药有限公司 | 一种卡格列净快速释放片剂及其制备方法 |
| WO2016142950A1 (fr) * | 2015-03-11 | 2016-09-15 | Harman Finochem Limited | Nouveau procédé de préparation de (2s,3r,4r,5s,6r)-2-{3-[5-[4-fluoro-phényl)-thiophén-2-ylméthyl]-4-méthyl-phényl}-6-hydroxyméthyl-tétrahydro-pyran-3,4,5-triol et de sa forme semi-hydratée amorphe stable |
| CN106279134A (zh) * | 2015-06-23 | 2017-01-04 | 中美华世通生物医药科技（武汉）有限公司 | 卡格列净单晶及其制备方法和用途 |
| US20170071970A1 (en) * | 2015-09-15 | 2017-03-16 | Janssen Pharmaceutica Nv | Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders |
| CN106749212A (zh) * | 2015-11-24 | 2017-05-31 | 重庆圣华曦药业股份有限公司 | 一种卡格列净中间体的精制方法 |
| CN105503845A (zh) * | 2015-12-01 | 2016-04-20 | 北京普德康利医药科技发展有限公司 | 去氟卡格列净化合物及其制备方法和应用 |
| TWI835735B (zh) * | 2017-06-12 | 2024-03-21 | 比利時商健生藥品公司 | 減少或預防第ii型糖尿病患者中心血管事件之方法 |
| CN109553649B (zh) * | 2017-09-26 | 2020-12-04 | 北大方正集团有限公司 | 一种卡格列净中间体的制备方法 |
| CN109553609B (zh) * | 2017-09-26 | 2020-09-04 | 北大方正集团有限公司 | 一种卡格列净的制备方法 |
| US11857559B2 (en) | 2018-09-10 | 2024-01-02 | Aurobindo Pharma Ltd. | Pharmaceutical composition comprising Canagliflozin, process of preparation and use thereof |
| CN110946840B (zh) * | 2019-12-31 | 2021-11-26 | 常州恒邦药业有限公司 | 一种卡格列净药物组合物及其制备方法 |
| WO2024053680A1 (fr) * | 2022-09-07 | 2024-03-14 | 田辺三菱製薬株式会社 | Comprimé orodispersible |
| CN115531376A (zh) * | 2022-10-26 | 2022-12-30 | 河南省人民医院 | 卡格列净在菌群调节方面的新应用 |
Family Cites Families (8)
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|---|---|---|---|---|
| US6635278B1 (en) * | 1998-12-15 | 2003-10-21 | Gilead Sciences, Inc. | Pharmaceutical formulations |
| US6515117B2 (en) | 1999-10-12 | 2003-02-04 | Bristol-Myers Squibb Company | C-aryl glucoside SGLT2 inhibitors and method |
| CA2424770A1 (fr) * | 2000-10-06 | 2003-04-03 | Takeda Chemical Industries, Ltd. | Preparations solides |
| EP1651658B2 (fr) * | 2003-08-01 | 2020-08-12 | Mitsubishi Tanabe Pharma Corporation | Nouveaux composes possedant une activite inhibitrice dirigee contre le transporteur dependant du sodium |
| UY30730A1 (es) | 2006-12-04 | 2008-07-03 | Mitsubishi Tanabe Pharma Corp | Forma cristalina del hemihidrato de 1-(b (beta)-d-glucopiranosil) -4-metil-3-[5-(4-fluorofenil) -2-tienilmetil]benceno |
| AR065809A1 (es) * | 2007-03-22 | 2009-07-01 | Bristol Myers Squibb Co | Formulaciones farmaceuticas que contienen un inhibidor sglt2 |
| CL2008002425A1 (es) * | 2007-08-16 | 2009-09-11 | Boehringer Ingelheim Int | Composición farmacéutica que comprende un inhibidor de sglt2 y 1-(4-metil-quinazolin-2-il)metil-3metil-7-(-2-butin-1-il)-8-(3-(r)-amino-piperidin-1il)-xantina, un inhibidor de dpp iv y su uso para el tratamiento de la obesidad y de la diabetes tipo 1 y 2 y complicaciones de esta. |
| SG173619A1 (en) * | 2009-02-13 | 2011-09-29 | Boehringer Ingelheim Int | Pharmaceutical composition comprising a sglt2 inhibitor, a dpp-iv inhibitor and optionally a further antidiabetic agent and uses thereof |
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2011
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- 2011-05-11 WO PCT/JP2011/061354 patent/WO2011142478A1/fr active Application Filing
- 2011-05-11 TW TW100116437A patent/TWI564034B/zh active
- 2011-05-11 CN CN201610158907.XA patent/CN105769792A/zh active Pending
- 2011-05-11 KR KR1020127032207A patent/KR101869110B1/ko active IP Right Grant
- 2011-05-11 JP JP2012551398A patent/JP5596799B2/ja active Active
- 2011-05-11 EP EP11725825.1A patent/EP2568971B1/fr active Active
- 2011-05-11 US US13/697,225 patent/US20130052266A1/en not_active Abandoned
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| Publication number | Publication date |
|---|---|
| TWI564034B (zh) | 2017-01-01 |
| KR20130106279A (ko) | 2013-09-27 |
| WO2011142478A1 (fr) | 2011-11-17 |
| JP2013526482A (ja) | 2013-06-24 |
| US9655852B2 (en) | 2017-05-23 |
| US20130052266A1 (en) | 2013-02-28 |
| CN105769792A (zh) | 2016-07-20 |
| US20160228375A1 (en) | 2016-08-11 |
| EP2568971A1 (fr) | 2013-03-20 |
| CN102985075A (zh) | 2013-03-20 |
| ES2836952T3 (es) | 2021-06-28 |
| CN106890147A (zh) | 2017-06-27 |
| KR101869110B1 (ko) | 2018-06-19 |
| TW201200164A (en) | 2012-01-01 |
| EP2568971B1 (fr) | 2020-10-14 |
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