JP5579432B2 - 新規ヒドロキシフェニル誘導体およびその生物学的適用 - Google Patents

新規ヒドロキシフェニル誘導体およびその生物学的適用 Download PDF

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JP5579432B2
JP5579432B2 JP2009504857A JP2009504857A JP5579432B2 JP 5579432 B2 JP5579432 B2 JP 5579432B2 JP 2009504857 A JP2009504857 A JP 2009504857A JP 2009504857 A JP2009504857 A JP 2009504857A JP 5579432 B2 JP5579432 B2 JP 5579432B2
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アレキシス ドゥニ
ヴァンサン ゲリュス
ヤニック ボンヴァン
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ファブ ファルマ エス アー エス
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    • C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/092—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings with aromatic radicals attached to the chain
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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  • Plural Heterocyclic Compounds (AREA)
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  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
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EP1845087A1 (en) 2006-04-14 2007-10-17 Mutabilis SA Hydroxyphenyl derivatives and biological applications thereof
DE102008053242A1 (de) * 2008-10-25 2010-05-06 Saltigo Gmbh Heteroaryl-Arylether
JP5626737B2 (ja) * 2009-09-01 2014-11-19 ファブ ファーマ エスエーエス 新規抗菌性ヒドロキシフェニル化合物
JP5752138B2 (ja) * 2009-10-20 2015-07-22 ファブ ファーマ エスエーエス 新規なアシルピペラジノン、及び医薬としてのそれらの使用
MX2012005759A (es) 2009-11-18 2012-10-03 Fab Pharma S A S Acrilamidas heterociclicas novedosas y su uso como farmacos.
WO2011106630A2 (en) 2010-02-27 2011-09-01 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Chrysophaentin antimicrobial compounds that inhibit ftsz protein
EP2474313A1 (en) * 2011-01-11 2012-07-11 ABRA Pharmaceuticals sàrl Novel self-assembling polyphenol-quinonoid polymer derivatives and use thereof
GB201522179D0 (en) * 2015-12-16 2016-01-27 Autifony Therapeutics Ltd Novel compounds
US11905286B2 (en) 2018-08-09 2024-02-20 Antabio Sas Diazabicyclooctanones as inhibitors of serine beta-lactamases
EP3833665B1 (en) 2018-08-09 2023-07-19 Antabio SAS Diazabicyclooctanones as inhibitors of serine beta-lactamases

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JP5626737B2 (ja) 2009-09-01 2014-11-19 ファブ ファーマ エスエーエス 新規抗菌性ヒドロキシフェニル化合物

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CA2649196C (en) 2016-06-07
JP2009533417A (ja) 2009-09-17
US20100041658A1 (en) 2010-02-18
WO2007135562A3 (en) 2008-01-24
IL194781A (en) 2013-08-29
CN101500999A (zh) 2009-08-05
EP2010495A2 (en) 2009-01-07
CN101500999B (zh) 2014-01-15
AU2007252917A1 (en) 2007-11-29
US8722746B2 (en) 2014-05-13
EP1845087A1 (en) 2007-10-17
US20160185724A1 (en) 2016-06-30
IL194781A0 (en) 2009-08-03
AU2007252917C1 (en) 2014-05-29
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