JP5128578B2 - 解離性障害の治療のためのκ−オピオイド受容体アンタゴニスト含有組成物の利用 - Google Patents
解離性障害の治療のためのκ−オピオイド受容体アンタゴニスト含有組成物の利用 Download PDFInfo
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- JP5128578B2 JP5128578B2 JP2009503576A JP2009503576A JP5128578B2 JP 5128578 B2 JP5128578 B2 JP 5128578B2 JP 2009503576 A JP2009503576 A JP 2009503576A JP 2009503576 A JP2009503576 A JP 2009503576A JP 5128578 B2 JP5128578 B2 JP 5128578B2
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- opioid receptor
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- A61K31/4748—Quinolines; Isoquinolines forming part of bridged ring systems
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
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- Neurosurgery (AREA)
- Emergency Medicine (AREA)
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102006015733.8 | 2006-04-04 | ||
| DE102006015733A DE102006015733A1 (de) | 2006-04-04 | 2006-04-04 | Verwendung von Buprenorphin und Buprenorphin-Derivaten zur Herstellung eines Medikaments zur Behandlung von emotional instabiler Persönlichkeitsstörung, Alkoholabhängigkeit und/oder multipler Substanzabhängigkeit |
| DE102006016991A DE102006016991A1 (de) | 2006-04-11 | 2006-04-11 | Verwendung von kappa-Opioidrezeptor-Antagonisten zur Behandlung von dissoziativen Störungen |
| DE102006016991.3 | 2006-04-11 | ||
| PCT/EP2007/053248 WO2007115975A2 (de) | 2006-04-04 | 2007-04-03 | Verwendung von zusammensetzungen enthaltend kappa-opioidrezeptor-antagonisten zur behandlung von dissoziativen störungen |
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| JP2009532434A JP2009532434A (ja) | 2009-09-10 |
| JP2009532434A5 JP2009532434A5 (enExample) | 2010-11-11 |
| JP5128578B2 true JP5128578B2 (ja) | 2013-01-23 |
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| JO2797B1 (en) | 2008-01-22 | 2014-03-15 | ايلي ليلي اند كومباني | Selective opioid receptor antagonist kappa |
| US9192570B2 (en) | 2013-12-20 | 2015-11-24 | AntiOP, Inc. | Intranasal naloxone compositions and methods of making and using same |
| AU2014368548B2 (en) * | 2013-12-20 | 2019-09-19 | H. Lundbeck A/S | Use of an opioid receptor antagonist with kappa-activity and vortioxetine for treatment of depressive disorder with melancholic features |
| CN106470999B (zh) | 2014-04-28 | 2018-11-13 | 奥佛麦德公司 | 叔丁啡二聚体及其在治疗肠胃失调中的应用 |
| US10316021B2 (en) | 2016-11-28 | 2019-06-11 | Pfizer Inc. | Heteroarylphenoxy benzamide kappa opioid ligands |
| US12161622B2 (en) | 2021-05-04 | 2024-12-10 | Janssen Pharmaceuticals, Inc. | Compositions and methods for the treatment of depression |
| CA3254546A1 (en) | 2022-03-07 | 2023-09-14 | Janssen Pharmaceuticals, Inc. | COMPOSITIONS CONTAINING ATICAPRANT |
| WO2023170550A1 (en) | 2022-03-07 | 2023-09-14 | Janssen Pharmaceuticals, Inc. | Polymorph forms of aticaprant for use in treating major depressive disorder |
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| US5028612A (en) * | 1990-03-22 | 1991-07-02 | Hillel Glover | Method for treating emotional numbness |
| US5780479A (en) * | 1997-04-04 | 1998-07-14 | Regents Of The University Of Minnesota | Use of opioid antagonists to treat impulse-control disorders |
| EP1061924A1 (en) * | 1998-03-09 | 2000-12-27 | Trustees Of Tufts College | Treatment of compulsive behaviours in man and animals |
| US20020045572A1 (en) * | 2000-08-15 | 2002-04-18 | Cpd, Llc | Method of treating the syndrome of type 2 diabetes in humans |
| WO2002013759A2 (en) | 2000-08-15 | 2002-02-21 | Cpd Llc | Method of treating the syndrome of type 2 diabetes in humans |
| EP1353665A4 (en) * | 2000-12-21 | 2004-05-06 | Mclean Hospital Corp | Treatment of depression |
| US7666876B2 (en) * | 2002-03-19 | 2010-02-23 | Vernalis (R&D) Limited | Buprenorphine formulations for intranasal delivery |
| US7268151B2 (en) * | 2003-04-04 | 2007-09-11 | Merck & Co., Inc. | Di-aryl substituted triazole modulators of metabotropic glutamate receptor-5 |
| WO2005084654A2 (en) | 2004-03-02 | 2005-09-15 | Pharmacia Corporation | Methods and compositions for treating or preventing psychiatric disorders with cox-2 inhibitors alone and in combination with antidepressant agents |
| ATE462704T1 (de) * | 2004-05-26 | 2010-04-15 | Inotek Pharmaceuticals Corp | Purinderivate als adenosin a 1 rezeptoragonisten und anwendungsverfahren dafür |
| DE602004017514D1 (de) | 2004-06-02 | 2008-12-11 | Galephar M F | Stabile orale pharmazeutische zusammensetzungen von buprenorphin und salz davon |
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Also Published As
| Publication number | Publication date |
|---|---|
| EA014820B1 (ru) | 2011-02-28 |
| EA200802104A1 (ru) | 2009-04-28 |
| EP2001456B1 (de) | 2009-12-02 |
| PT2001456E (pt) | 2010-03-03 |
| SI2001456T1 (sl) | 2010-04-30 |
| DE502007002185D1 (de) | 2010-01-14 |
| PL2001456T3 (pl) | 2010-05-31 |
| US8063059B2 (en) | 2011-11-22 |
| WO2007115975A2 (de) | 2007-10-18 |
| HRP20100113T1 (hr) | 2010-04-30 |
| EP2001456A2 (de) | 2008-12-17 |
| CY1109862T1 (el) | 2014-09-10 |
| WO2007115975A3 (de) | 2008-02-14 |
| JP2009532434A (ja) | 2009-09-10 |
| ATE450256T1 (de) | 2009-12-15 |
| CA2646899A1 (en) | 2007-10-18 |
| RS51211B (sr) | 2010-12-31 |
| CA2646899C (en) | 2014-05-06 |
| AU2007236003A1 (en) | 2007-10-18 |
| DK2001456T3 (da) | 2010-04-12 |
| ES2337622T3 (es) | 2010-04-27 |
| AU2007236003B2 (en) | 2012-10-18 |
| US20090181999A1 (en) | 2009-07-16 |
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