JP5080263B2 - 勃起不全の治療のためのプロピオニルｌ−カルニチンおよびシルデナフィルと組み合わせてのアセチルｌ−カルニチンの使用 - Google Patents
勃起不全の治療のためのプロピオニルｌ−カルニチンおよびシルデナフィルと組み合わせてのアセチルｌ−カルニチンの使用 Download PDFInfo
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- JP5080263B2 JP5080263B2 JP2007540521A JP2007540521A JP5080263B2 JP 5080263 B2 JP5080263 B2 JP 5080263B2 JP 2007540521 A JP2007540521 A JP 2007540521A JP 2007540521 A JP2007540521 A JP 2007540521A JP 5080263 B2 JP5080263 B2 JP 5080263B2
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- Prior art keywords
- carnitine
- acid
- acetyl
- propionyl
- treatment
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/191—Carboxylic acids, e.g. valproic acid having two or more hydroxy groups, e.g. gluconic acid
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
Landscapes
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- Veterinary Medicine (AREA)
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- General Health & Medical Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT000561A ITRM20040561A1 (it) | 2004-11-11 | 2004-11-11 | Uso della acetil l-carnitina in combinazione con propionil l-carnitina e sildenafil per il trattamento della disfunzione erettile. |
| ITRM2004A000561 | 2004-11-11 | ||
| PCT/EP2005/011238 WO2006050794A1 (en) | 2004-11-11 | 2005-10-19 | Use of acetyl l-carnitine in combination with propionyl l-carnitine and sildenafil for the treatment of erectile dysfunction |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008531466A JP2008531466A (ja) | 2008-08-14 |
| JP2008531466A5 JP2008531466A5 (enExample) | 2008-12-04 |
| JP5080263B2 true JP5080263B2 (ja) | 2012-11-21 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007540521A Expired - Fee Related JP5080263B2 (ja) | 2004-11-11 | 2005-10-19 | 勃起不全の治療のためのプロピオニルｌ−カルニチンおよびシルデナフィルと組み合わせてのアセチルｌ−カルニチンの使用 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US8003652B2 (enExample) |
| EP (1) | EP1811988B1 (enExample) |
| JP (1) | JP5080263B2 (enExample) |
| KR (1) | KR101455275B1 (enExample) |
| AT (1) | ATE456950T1 (enExample) |
| CA (1) | CA2585654C (enExample) |
| CY (1) | CY1110239T1 (enExample) |
| DE (1) | DE602005019251D1 (enExample) |
| DK (1) | DK1811988T3 (enExample) |
| ES (1) | ES2339265T3 (enExample) |
| IT (1) | ITRM20040561A1 (enExample) |
| MX (1) | MX2007005518A (enExample) |
| PL (1) | PL1811988T3 (enExample) |
| PT (1) | PT1811988E (enExample) |
| SI (1) | SI1811988T1 (enExample) |
| WO (1) | WO2006050794A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2010222347A (ja) * | 2009-02-24 | 2010-10-07 | Daiichi Sankyo Healthcare Co Ltd | Ｐｄｅ５阻害剤及びカルニチンを含有する医薬組成物 |
| WO2012000634A1 (de) | 2010-06-29 | 2012-01-05 | Georg Bambach | Pharmazeutische zusammensetzung zur behandlung von erektiler dysfunktion |
| WO2018070971A1 (ru) * | 2016-10-10 | 2018-04-19 | Товарыство З Обмэжэною Видповидальнистю Науково-Выробныча Фирма "Микрохим" | Фармацевтическая композиция в форме оромукозного спрея для лечения эректильной дисфункции и легочной артериальной гипертензии |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1077260B1 (en) | 1999-08-13 | 2010-03-31 | Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts | Parvovirus NS1 variants |
| IT1306722B1 (it) * | 1999-10-08 | 2001-10-02 | Sigma Tau Healthscience Spa | Composizione per la prevenzione e/o il trattamento di disfunzionicircolatorie, comprendente derivati della l-carnitina ed estratti di |
| JP2001233770A (ja) * | 2000-02-23 | 2001-08-28 | Dountsuendorufaa Udo | 勃起機能不全治療用の経口薬の組合わせ |
| ITRM20010621A1 (it) * | 2001-10-18 | 2003-04-18 | Aldo Fassi | Sali metallici non igroscopici e idrosolubili di alcanoil l-carnitine, integratori dietetici che li contengono e kit dietetici, per contrast |
| ITRM20010708A1 (it) * | 2001-12-04 | 2003-06-04 | Sigma Tau Ind Farmaceuti | Uso di una alcanoil l-carnitina per il trattamento della disfunzione erettile. |
| ITRM20020620A1 (it) * | 2002-12-13 | 2004-06-14 | Sigma Tau Ind Farmaceuti | Uso delle carnitine per la prevenzione e/o il trattamento dei disturbi causati dall'andropausa. |
-
2004
- 2004-11-11 IT IT000561A patent/ITRM20040561A1/it unknown
-
2005
- 2005-10-19 AT AT05798477T patent/ATE456950T1/de active
- 2005-10-19 DE DE602005019251T patent/DE602005019251D1/de not_active Expired - Lifetime
- 2005-10-19 ES ES05798477T patent/ES2339265T3/es not_active Expired - Lifetime
- 2005-10-19 CA CA2585654A patent/CA2585654C/en not_active Expired - Fee Related
- 2005-10-19 WO PCT/EP2005/011238 patent/WO2006050794A1/en not_active Ceased
- 2005-10-19 PT PT05798477T patent/PT1811988E/pt unknown
- 2005-10-19 PL PL05798477T patent/PL1811988T3/pl unknown
- 2005-10-19 US US11/719,011 patent/US8003652B2/en not_active Expired - Fee Related
- 2005-10-19 JP JP2007540521A patent/JP5080263B2/ja not_active Expired - Fee Related
- 2005-10-19 KR KR1020077013019A patent/KR101455275B1/ko not_active Expired - Fee Related
- 2005-10-19 DK DK05798477.5T patent/DK1811988T3/da active
- 2005-10-19 EP EP05798477A patent/EP1811988B1/en not_active Expired - Lifetime
- 2005-10-19 SI SI200530953T patent/SI1811988T1/sl unknown
- 2005-10-19 MX MX2007005518A patent/MX2007005518A/es active IP Right Grant
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2010
- 2010-04-23 CY CY20101100362T patent/CY1110239T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US8003652B2 (en) | 2011-08-23 |
| ITRM20040561A1 (it) | 2005-02-11 |
| DE602005019251D1 (de) | 2010-03-25 |
| CA2585654C (en) | 2013-04-02 |
| WO2006050794A1 (en) | 2006-05-18 |
| JP2008531466A (ja) | 2008-08-14 |
| CA2585654A1 (en) | 2006-05-18 |
| ATE456950T1 (de) | 2010-02-15 |
| PL1811988T3 (pl) | 2010-07-30 |
| PT1811988E (pt) | 2010-04-08 |
| EP1811988A1 (en) | 2007-08-01 |
| SI1811988T1 (sl) | 2010-10-29 |
| DK1811988T3 (da) | 2010-05-17 |
| EP1811988B1 (en) | 2010-02-03 |
| CY1110239T1 (el) | 2015-01-14 |
| ES2339265T3 (es) | 2010-05-18 |
| MX2007005518A (es) | 2007-05-18 |
| US20080090906A1 (en) | 2008-04-17 |
| KR101455275B1 (ko) | 2014-10-27 |
| KR20070085961A (ko) | 2007-08-27 |
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