JP5026635B2 - 医薬物質の迅速放出医薬組成物 - Google Patents

医薬物質の迅速放出医薬組成物 Download PDF

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Publication number
JP5026635B2
JP5026635B2 JP2000569779A JP2000569779A JP5026635B2 JP 5026635 B2 JP5026635 B2 JP 5026635B2 JP 2000569779 A JP2000569779 A JP 2000569779A JP 2000569779 A JP2000569779 A JP 2000569779A JP 5026635 B2 JP5026635 B2 JP 5026635B2
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composition
dissolution
substance
particle size
test
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Expired - Lifetime
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Japanese (ja)
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JP2002524492A5 (enExample
JP2002524492A (ja
Inventor
ポウル・ベルテルセン
ニルス・グイェルロヴ・ハンセン
ヘルマン・ルッケノルファー
茂 板井
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Takeda Pharma AS
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Nycomed Danmark AS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1611—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2000569779A 1998-09-10 1999-09-10 医薬物質の迅速放出医薬組成物 Expired - Lifetime JP5026635B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DK199801143 1998-09-10
DKPA199801143 1998-09-10
DKPA199801143 1998-09-10
PCT/DK1999/000480 WO2000015195A1 (en) 1998-09-10 1999-09-10 Quick release pharmaceutical compositions of drug substances

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2011227314A Division JP5622703B2 (ja) 1998-09-10 2011-10-14 医薬物質の迅速放出医薬組成物

Publications (3)

Publication Number Publication Date
JP2002524492A JP2002524492A (ja) 2002-08-06
JP2002524492A5 JP2002524492A5 (enExample) 2006-11-24
JP5026635B2 true JP5026635B2 (ja) 2012-09-12

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JP2000569779A Expired - Lifetime JP5026635B2 (ja) 1998-09-10 1999-09-10 医薬物質の迅速放出医薬組成物
JP2011227314A Expired - Lifetime JP5622703B2 (ja) 1998-09-10 2011-10-14 医薬物質の迅速放出医薬組成物

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JP2011227314A Expired - Lifetime JP5622703B2 (ja) 1998-09-10 2011-10-14 医薬物質の迅速放出医薬組成物

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Country Link
US (1) US6713089B1 (enExample)
EP (1) EP1109534B1 (enExample)
JP (2) JP5026635B2 (enExample)
AT (1) ATE232382T1 (enExample)
AU (1) AU5504599A (enExample)
CA (1) CA2343148C (enExample)
DE (1) DE69905380T2 (enExample)
DK (1) DK1109534T3 (enExample)
EA (1) EA004032B1 (enExample)
ES (1) ES2190241T3 (enExample)
PT (1) PT1109534E (enExample)
TR (1) TR200100708T2 (enExample)
WO (1) WO2000015195A1 (enExample)

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Publication number Publication date
US6713089B1 (en) 2004-03-30
JP5622703B2 (ja) 2014-11-12
EA200100331A1 (ru) 2001-08-27
AU5504599A (en) 2000-04-03
EA004032B1 (ru) 2003-12-25
DK1109534T3 (da) 2003-06-10
PT1109534E (pt) 2003-06-30
ES2190241T3 (es) 2003-07-16
JP2012082197A (ja) 2012-04-26
JP2002524492A (ja) 2002-08-06
EP1109534B1 (en) 2003-02-12
CA2343148C (en) 2005-11-15
CA2343148A1 (en) 2000-03-23
WO2000015195A1 (en) 2000-03-23
DE69905380T2 (de) 2003-11-27
TR200100708T2 (tr) 2001-07-23
ATE232382T1 (de) 2003-02-15
DE69905380D1 (de) 2003-03-20
EP1109534A1 (en) 2001-06-27

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