JP5021155B2 - エピナスチンと１種以上のさらなる抗−ｈ１−ヒスタミン類との組合せを含む皮膚疾患治療用製薬組成物 - Google Patents
エピナスチンと１種以上のさらなる抗−ｈ１−ヒスタミン類との組合せを含む皮膚疾患治療用製薬組成物 Download PDFInfo
- Publication number
- JP5021155B2 JP5021155B2 JP2004223680A JP2004223680A JP5021155B2 JP 5021155 B2 JP5021155 B2 JP 5021155B2 JP 2004223680 A JP2004223680 A JP 2004223680A JP 2004223680 A JP2004223680 A JP 2004223680A JP 5021155 B2 JP5021155 B2 JP 5021155B2
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- JP
- Japan
- Prior art keywords
- epinastine
- pharmaceutical composition
- range
- pharmaceutically acceptable
- oral
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
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- WHWZLSFABNNENI-UHFFFAOYSA-N epinastine Chemical compound C1C2=CC=CC=C2C2CN=C(N)N2C2=CC=CC=C21 WHWZLSFABNNENI-UHFFFAOYSA-N 0.000 title claims abstract description 57
- 229960003449 epinastine Drugs 0.000 title claims abstract description 40
- 208000017520 skin disease Diseases 0.000 title claims abstract description 31
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract description 28
- 150000003839 salts Chemical class 0.000 claims abstract description 28
- 239000002552 dosage form Substances 0.000 claims abstract description 22
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- 239000003826 tablet Substances 0.000 claims description 29
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- 229960002548 epinastine hydrochloride Drugs 0.000 claims description 16
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- ZZVUWRFHKOJYTH-UHFFFAOYSA-N diphenhydramine Chemical compound C=1C=CC=CC=1C(OCCN(C)C)C1=CC=CC=C1 ZZVUWRFHKOJYTH-UHFFFAOYSA-N 0.000 claims description 8
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- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| EP03016681.3 | 2003-08-01 |
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| JP2005053907A JP2005053907A (ja) | 2005-03-03 |
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| RU2472499C2 (ru) * | 2007-06-08 | 2013-01-20 | Байер Конзюмер Кер АГ | Лекарственное средство, включающее комбинацию активных веществ, содержащую пантотеновую кислоту или ее производные, для лечения аллергических симптомов |
| JP2019043853A (ja) * | 2017-08-30 | 2019-03-22 | 旭化成株式会社 | 経皮吸収促進剤、経皮吸収促進助剤、及び経皮製剤 |
| WO2022138826A1 (ja) * | 2020-12-24 | 2022-06-30 | 参天製薬株式会社 | エピナスチン又はその塩を含有する塗布投与用医薬組成物 |
| WO2022138842A1 (ja) * | 2020-12-24 | 2022-06-30 | 参天製薬株式会社 | エピナスチン又はその塩と硫黄系抗酸化剤を含有する経皮投与用医薬組成物 |
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| JP4563522B2 (ja) * | 1999-02-19 | 2010-10-13 | 豊也 加藤 | アレルギー疾患治療剤 |
| PE20020324A1 (es) * | 2000-10-06 | 2002-06-18 | Boehringer Ingelheim Int | Nuevas composiciones farmaceuticas que contienen epinastina y pseudoefedrina |
| US6827946B2 (en) * | 2001-12-05 | 2004-12-07 | Collegium Pharmaceutical, Inc. | Compositions containing both sedative and non-sedative antihistamines |
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