JP4975435B2 - 置換されたチアゾールの製造方法 - Google Patents

置換されたチアゾールの製造方法 Download PDF

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Publication number
JP4975435B2
JP4975435B2 JP2006522112A JP2006522112A JP4975435B2 JP 4975435 B2 JP4975435 B2 JP 4975435B2 JP 2006522112 A JP2006522112 A JP 2006522112A JP 2006522112 A JP2006522112 A JP 2006522112A JP 4975435 B2 JP4975435 B2 JP 4975435B2
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JP
Japan
Prior art keywords
solvent
temperature
formula
compound
psi
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
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JP2006522112A
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English (en)
Japanese (ja)
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JP2007500724A (ja
JP2007500724A5 (https=
Inventor
ロビンス，テイモシー・エイ
チユー，ヘレン
シヤオ，チユン
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Abbott Laboratories
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Abbott Laboratories
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Publication of JP2007500724A publication Critical patent/JP2007500724A/ja
Publication of JP2007500724A5 publication Critical patent/JP2007500724A5/ja
Application granted granted Critical
Publication of JP4975435B2 publication Critical patent/JP4975435B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2006522112A 2003-07-30 2004-07-30 置換されたチアゾールの製造方法 Expired - Lifetime JP4975435B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/630,043 2003-07-30
US10/630,043 US20050027128A1 (en) 2003-07-30 2003-07-30 Substituted thiazoles
PCT/US2004/024758 WO2005012273A2 (en) 2003-07-30 2004-07-30 Process for the preparation of substituted thiazoles

Publications (3)

Publication Number Publication Date
JP2007500724A JP2007500724A (ja) 2007-01-18
JP2007500724A5 JP2007500724A5 (https=) 2007-08-16
JP4975435B2 true JP4975435B2 (ja) 2012-07-11

Family

ID=34103748

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2006522112A Expired - Lifetime JP4975435B2 (ja) 2003-07-30 2004-07-30 置換されたチアゾールの製造方法

Country Status (6)

Country Link
US (1) US20050027128A1 (https=)
EP (2) EP2386548A2 (https=)
JP (1) JP4975435B2 (https=)
CA (1) CA2533658C (https=)
MX (1) MXPA06001201A (https=)
WO (1) WO2005012273A2 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2710453C (en) * 2007-12-26 2019-07-02 Biotest Ag Agents targeting cd138 and uses thereof
US8791077B2 (en) * 2008-05-22 2014-07-29 Astrazeneca Ab Method for treating hyperuricemia employing an SGLT2 inhibitor and composition containing same
US20120078013A1 (en) * 2009-06-09 2012-03-29 Teijin Pharma Limited Method for producing 4-substituted benzothioamide derivative
WO2011073617A1 (en) 2009-12-14 2011-06-23 Cipla Limited Processes for the preparation of febuxostat and salts thereof
US8857343B2 (en) * 2012-05-29 2014-10-14 Liberty Ammunition, Llc High volume multiple component projectile assembly
CN102702054A (zh) * 2012-06-29 2012-10-03 晋城海斯制药有限公司 一种对羟基硫代苯甲酰胺的制备方法
CN104610110A (zh) * 2014-03-12 2015-05-13 广东东阳光药业有限公司 一种制备4-取代硫代苯甲酰胺衍生物的方法

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3518279A (en) * 1967-08-29 1970-06-30 American Cyanamid Co Thiazolylphenyl phosphates
US3852287A (en) * 1970-03-26 1974-12-03 Uniroyal Ltd Preparation of thionamides
US4528291A (en) * 1982-06-22 1985-07-09 Schering Corporation 2-(4'-Pyridinyl)-thiazole compounds and their use in increasing cardiac contractility
DE4031804A1 (de) * 1990-10-08 1992-04-09 Basf Ag Indophenolfarbstoffe und ein verfahren zu ihrer thermischen uebertragung
DK0513379T3 (da) * 1990-11-30 1996-09-30 Teijin Ltd 2-Arylthiazolderivater og farmaceutisk præparat indeholdende sådanne
JP2706037B2 (ja) * 1993-04-13 1998-01-28 帝人株式会社 シアノ化合物およびその製造方法
JPH10139770A (ja) * 1996-11-08 1998-05-26 Teijin Ltd ２−（３−シアノフェニル）チアゾール誘導体の製造法
JP3440196B2 (ja) * 1997-08-13 2003-08-25 帝人株式会社 チオベンズアミド誘導体の製造方法
DE19934066A1 (de) * 1999-07-23 2001-01-25 Basf Ag Verfahren zur Herstellung von 4-Cyano-2-aminomethylthiazol
PE20011010A1 (es) * 1999-12-02 2001-10-18 Glaxo Group Ltd Oxazoles y tiazoles sustituidos como agonista del receptor activado por el proliferador de peroxisomas humano
JP4716547B2 (ja) * 2000-08-10 2011-07-06 住友精化株式会社 ２−フェニルチアゾール類の製造方法
WO2002079177A1 (en) * 2001-03-29 2002-10-10 Nippon Soda Co.,Ltd. Process for producing (4-phenylthiazol-2-yl)alkanenitrile
JP2003002863A (ja) * 2001-06-25 2003-01-08 Nippon Soda Co Ltd 安息香酸類の製造方法および新規化合物

Also Published As

Publication number Publication date
EP1651624A2 (en) 2006-05-03
JP2007500724A (ja) 2007-01-18
WO2005012273A3 (en) 2005-05-12
CA2533658A1 (en) 2005-02-10
HK1093725A1 (en) 2007-03-09
MXPA06001201A (es) 2006-05-15
US20050027128A1 (en) 2005-02-03
EP2386548A2 (en) 2011-11-16
WO2005012273A2 (en) 2005-02-10
CA2533658C (en) 2013-10-22
EP1651624B1 (en) 2015-03-11

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