JP4787529B2 - 医薬組成物 - Google Patents

医薬組成物 Download PDF

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Publication number
JP4787529B2
JP4787529B2 JP2005113726A JP2005113726A JP4787529B2 JP 4787529 B2 JP4787529 B2 JP 4787529B2 JP 2005113726 A JP2005113726 A JP 2005113726A JP 2005113726 A JP2005113726 A JP 2005113726A JP 4787529 B2 JP4787529 B2 JP 4787529B2
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Japan
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group
substituted
halogen
unsubstituted
phenyl
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JP2005113726A
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Japanese (ja)
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JP2005330266A5 (enrdf_load_stackoverflow
JP2005330266A (ja
Inventor
英継 壷内
博文 佐々木
英明 黒田
元宏 糸谷
武司 長谷川
佳和 原口
武志 黒田
敬之 松崎
国憲 田井
眞 小松
真 松本
博之 橋詰
辰夫 富重
祐治 清家
昌則 川▲崎▼
卓美 住田
伸 宮村
絹枝 大黒
一穂 田中
勲 竹村
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Otsuka Pharmaceutical Co Ltd
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Otsuka Pharmaceutical Co Ltd
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Priority to JP2005113726A priority Critical patent/JP4787529B2/ja
Publication of JP2005330266A publication Critical patent/JP2005330266A/ja
Publication of JP2005330266A5 publication Critical patent/JP2005330266A5/ja
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  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2005113726A 2004-04-09 2005-04-11 医薬組成物 Expired - Lifetime JP4787529B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2005113726A JP4787529B2 (ja) 2004-04-09 2005-04-11 医薬組成物

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2004114975 2004-04-09
JP2004114975 2004-04-09
JP2004125055 2004-04-21
JP2004125055 2004-04-21
JP2005113726A JP4787529B2 (ja) 2004-04-09 2005-04-11 医薬組成物

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2008103907A Division JP4789966B2 (ja) 2004-04-09 2008-04-11 医薬組成物
JP2011101480A Division JP5345174B2 (ja) 2004-04-09 2011-04-28 医薬組成物

Publications (3)

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JP2005330266A JP2005330266A (ja) 2005-12-02
JP2005330266A5 JP2005330266A5 (enrdf_load_stackoverflow) 2008-05-29
JP4787529B2 true JP4787529B2 (ja) 2011-10-05

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JP2005113726A Expired - Lifetime JP4787529B2 (ja) 2004-04-09 2005-04-11 医薬組成物

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JP (1) JP4787529B2 (enrdf_load_stackoverflow)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016119706A1 (zh) * 2015-01-29 2016-08-04 南京明德新药研发股份有限公司 抗肺结核病的硝基咪唑衍生物
WO2018014863A1 (zh) * 2016-07-22 2018-01-25 南京明德新药研发股份有限公司 一种硝基咪唑类化合物的晶型、盐型及其制备方法

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JP2007297305A (ja) * 2006-04-28 2007-11-15 Daiso Co Ltd Ｎ−（２，３−エポキシ−２−メチルプロピル）フタルイミドの製造法
US7638541B2 (en) 2006-12-28 2009-12-29 Metabolex Inc. 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine
AR070301A1 (es) * 2007-05-08 2010-03-31 Otsuka Pharma Co Ltd Compuesto epoxi y metodo para producir el mismo
EP2152269B1 (en) 2007-06-08 2014-04-23 Janssen Pharmaceutica, N.V. Piperidine/piperazine derivatives
WO2008148840A1 (en) 2007-06-08 2008-12-11 Janssen Pharmaceutica N.V. Piperidine/piperazine derivatives
RU2470017C2 (ru) 2007-06-08 2012-12-20 Янссен Фармацевтика Н.В. Производные пиперидина/пиперазина
JO2972B1 (en) 2007-06-08 2016-03-15 جانسين فارماسوتيكا ان. في Piperidine / piperazine derivatives
CA2719000A1 (en) * 2008-03-20 2009-09-24 Forest Laboratories Holdings Limited Piperidine derivatives as inhibitors of stearoyl-coa desaturase
NZ587096A (en) * 2008-03-26 2011-11-25 Global Alliance For Tb Drug Dev Bicyclic nitroimidazoles covalently linked to substituted phenyl oxazolidinones
EP2296659B1 (en) 2008-06-05 2016-12-21 Janssen Pharmaceutica, N.V. Drug combinations comprising a DGAT inhibitor and a PPAR-agonist
BRPI0914891A2 (pt) * 2008-06-20 2015-11-24 Metabolex Inc agonistas de aril gpr119 e usos dos mesmos
WO2011014776A1 (en) 2009-07-31 2011-02-03 Global Alliance For Tb Drug Development Nitroimidazooxazine and nitroimidazooxazole analogues and their uses
ES2497566T3 (es) 2009-10-01 2014-09-23 Cymabay Therapeutics, Inc. Sales de tetrazol-1-il-fenoximetil-tiazol-2-il-piperidinil-pirimidina sustituida
WO2011052522A1 (ja) 2009-10-26 2011-05-05 富士フイルムＲｉファーマ株式会社 感染症診断薬
WO2014014845A1 (en) 2012-07-18 2014-01-23 Vertex Pharmaceuticals Incorporated Combination therapy comprising|1 -ethyl-3-[5-[2-{1 -hydroxy-1 -methyl-ethyl}pyrimidin-5-yl]-7-(tetra hydrofuran-2-|yl}-1 h-benzimidazol-2-yl]urea and derivatives thereof to treat mycobacterium|diseases
US9845330B2 (en) * 2013-10-04 2017-12-19 Council Of Scientific & Industrial Research 6-nitro-2,3-dihydroimidazo[2,1-b]oxazoles and a process for the preparation thereof
JP6467042B2 (ja) * 2014-10-21 2019-02-06 カウンシル オブ サイエンティフィック アンド インダストリアル リサーチ 抗マイコバクテリア剤としての置換１，２，３−トリアゾール−１−イル−メチル−２，３−ジヒドロ−２−メチル−６−ニトロイミダゾ［２，１−ｂ］オキサゾールとその調製方法
US10252995B2 (en) 2015-03-27 2019-04-09 Otsuka Pharmaceutical Co., Ltd. Method for producing 1-(4-hydroxyphenyl)-4-(4-trifluoromethoxyphenoxy)piperidine or salt thereof
CN106317072B (zh) * 2015-06-17 2020-03-17 盟科医药技术(上海)有限公司 用于分枝杆菌感染治疗的杂环化合物及其应用
US10292983B2 (en) 2016-08-03 2019-05-21 Cymabay Therapeutics, Inc. Oxymethylene aryl compounds for treating inflammatory gastrointestinal diseases or gastrointestinal conditions
GB201617758D0 (en) * 2016-10-20 2016-12-07 Almac Discovery Limited Pharmaceutical compounds
AU2018272359B2 (en) * 2017-05-26 2022-03-03 Cspc Zhongqi Pharmaceutical Technology (Shijiazhuang) Co., Ltd. Lactam compound as FXR receptor agonist
WO2019128963A1 (zh) * 2017-12-26 2019-07-04 南京明德新药研发股份有限公司 抗肺结核病的硝基咪唑衍生物
WO2020202205A1 (en) * 2019-04-01 2020-10-08 Council Of Scientific And Industrial Research Process for the preparation of derivatives of 1,1-dialkylethane-1,2-diols as useful intermediates
CN112300192B (zh) * 2019-08-02 2023-08-11 南京长澳医药科技有限公司 硝基咪唑类化合物及其制备方法和用途
CN115368252B (zh) * 2022-09-19 2024-01-12 西北农林科技大学 一种4-胺基酚类衍生物及应用
CN116570592B (zh) * 2023-04-17 2025-01-14 首都医科大学附属北京胸科医院 Gsk1292263在制备抑制结核分枝杆菌药物中的应用
CN119059990B (zh) * 2024-11-01 2025-02-07 安徽昊帆生物有限公司 1-氨基甲酸叔丁酯哌嗪的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5668127A (en) * 1995-06-26 1997-09-16 Pathogenesis Corporation Nitroimidazole antibacterial compounds and methods of use thereof
TWI347946B (en) * 2002-10-11 2011-09-01 Otsuka Pharma Co Ltd 2,3-dihydro-6-nitroimidazo[2,1-b]oxazole compound
JP4258630B2 (ja) * 2002-10-15 2009-04-30 大塚製薬株式会社 １位置換−４−ニトロイミダゾール化合物及びその製造法

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016119706A1 (zh) * 2015-01-29 2016-08-04 南京明德新药研发股份有限公司 抗肺结核病的硝基咪唑衍生物
EP3252059A4 (en) * 2015-01-29 2018-07-11 Medshine Discovery Inc. Anti-pulmonary tuberculosis nitroimidazole derivative
RU2675622C1 (ru) * 2015-01-29 2018-12-21 Медшайн Дискавери Инк. Производное нитроимидазола против туберкулеза легких
US10227362B2 (en) 2015-01-29 2019-03-12 Medshine Discovery Inc. Anti-pulmonary tuberculosis nitroimidazole derivative
WO2018014863A1 (zh) * 2016-07-22 2018-01-25 南京明德新药研发股份有限公司 一种硝基咪唑类化合物的晶型、盐型及其制备方法

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