JP4329290B2 - 脂肪族含窒素五員環化合物 - Google Patents

脂肪族含窒素五員環化合物 Download PDF

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Publication number
JP4329290B2
JP4329290B2 JP2001309558A JP2001309558A JP4329290B2 JP 4329290 B2 JP4329290 B2 JP 4329290B2 JP 2001309558 A JP2001309558 A JP 2001309558A JP 2001309558 A JP2001309558 A JP 2001309558A JP 4329290 B2 JP4329290 B2 JP 4329290B2
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Japan
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group
trans
cyano
cyclohexylamino
acetylpyrrolidine
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Expired - Fee Related
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JP2001309558A
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English (en)
Japanese (ja)
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JP2002356471A5 (enExample
JP2002356471A (ja
Inventor
公助 安田
啓氏 森本
三郎 河南
匡毅 彦田
健 松本
健司 荒川
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Mitsubishi Tanabe Pharma Corp
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Mitsubishi Tanabe Pharma Corp
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Priority to JP2001309558A priority Critical patent/JP4329290B2/ja
Publication of JP2002356471A publication Critical patent/JP2002356471A/ja
Publication of JP2002356471A5 publication Critical patent/JP2002356471A5/ja
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Publication of JP4329290B2 publication Critical patent/JP4329290B2/ja
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Expired - Fee Related legal-status Critical Current

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
JP2001309558A 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物 Expired - Fee Related JP4329290B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2000308528 2000-10-06
JP2000312562 2000-10-12
JP2001099251 2001-03-30
JP2000-312562 2001-03-30
JP2000-308528 2001-03-30
JP2001-99251 2001-03-30
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2003368572A Division JP2004035574A (ja) 2000-10-06 2003-10-29 脂肪族含窒素五員環化合物

Publications (3)

Publication Number Publication Date
JP2002356471A JP2002356471A (ja) 2002-12-13
JP2002356471A5 JP2002356471A5 (enExample) 2004-10-28
JP4329290B2 true JP4329290B2 (ja) 2009-09-09

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JP2001309558A Expired - Fee Related JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

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JP (1) JP4329290B2 (enExample)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10213051B4 (de) * 2002-03-23 2013-03-07 Grünenthal GmbH Substituierte 4-Aminocyclohexanole
US20050197350A1 (en) * 2003-03-31 2005-09-08 Taisho Pharmaceutical Co., Ltd. Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
CN101684089A (zh) 2004-02-05 2010-03-31 杏林制药株式会社 双环酯类衍生物
DE102004023632A1 (de) * 2004-05-10 2005-12-08 Grünenthal GmbH Substituierte Cyclohexylcarbonsäure-Derivate
NZ554515A (en) * 2004-10-12 2009-12-24 Glenmark Pharmaceuticals Sa Novel dipeptidyl peptidase IV inhibitors, pharmaceutical compositions containing them, and process for their preparation
DOP2006000008A (es) 2005-01-10 2006-08-31 Arena Pharm Inc Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1
WO2007102286A1 (ja) 2006-03-08 2007-09-13 Kyorin Pharmaceutical Co., Ltd. アミノアセチルピロリジンカルボニトリル誘導体の製造方法およびその製造中間体
PE20071221A1 (es) 2006-04-11 2007-12-14 Arena Pharm Inc Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas
DE602007010420D1 (de) 2006-04-11 2010-12-23 Arena Pharm Inc Verfahren zur verwendung des gpr119-rezeptors zur identifizierung von verbindungen zur erhöhung der knochenmasse bei einer person
WO2008066083A1 (fr) * 2006-11-29 2008-06-05 Mitsubishi Tanabe Pharma Corporation Procédé de production d'un dérivé de n-(n'-glycyle substitué)-2-cyanopyrrolidine
EP2123636B1 (en) 2007-03-22 2012-03-21 Kyorin Pharmaceutical Co., Ltd. Method for producing aminoacetylpyrrolidinecarbonitrile derivative
MX2010007593A (es) * 2008-01-10 2010-10-13 Sun Pharma Advanced Res Co Ltd Derivados novedosos de acil cianopirrolidinas.
EP2146210A1 (en) 2008-04-07 2010-01-20 Arena Pharmaceuticals, Inc. Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditions modulated by PYY
WO2010016584A1 (ja) 2008-08-07 2010-02-11 杏林製薬株式会社 ビシクロ[２．２．２]オクチルアミン誘導体の製造方法
AR077642A1 (es) 2009-07-09 2011-09-14 Arena Pharm Inc Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo
WO2011127051A1 (en) 2010-04-06 2011-10-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
MX2013003184A (es) 2010-09-22 2013-06-07 Arena Pharm Inc Moduladores del receptor gpr119 y el tratamiento de transtornos relacionados con el mismo.
WO2012135570A1 (en) 2011-04-01 2012-10-04 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145361A1 (en) 2011-04-19 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145603A1 (en) 2011-04-22 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
US20140051714A1 (en) 2011-04-22 2014-02-20 Arena Pharmaceuticals, Inc. Modulators Of The GPR119 Receptor And The Treatment Of Disorders Related Thereto
PE20140502A1 (es) * 2011-04-22 2014-05-02 Signal Pharm Llc Pirimidinas sustituidas de diaminocarboxamida y diaminocarbonitrilo, composiciones de las mismas y metodos de tratamiento con las mismas
WO2012170702A1 (en) 2011-06-08 2012-12-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2013055910A1 (en) 2011-10-12 2013-04-18 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2014074668A1 (en) 2012-11-08 2014-05-15 Arena Pharmaceuticals, Inc. Modulators of gpr119 and the treatment of disorders related thereto
CA2979033A1 (en) 2015-03-09 2016-09-15 Intekrin Therapeutics, Inc. Methods for the treatment of nonalcoholic fatty liver disease and/or lipodystrophy
CN110996951A (zh) 2017-04-03 2020-04-10 科赫罗斯生物科学股份有限公司 治疗进行性核上性麻痹的PPARγ激动剂
CA3061787A1 (en) * 2017-05-15 2018-11-22 Cognition Therapeutics, Inc. Compositions for treating neurodegenerative diseases

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Publication number Publication date
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