JP4329290B2 - 脂肪族含窒素五員環化合物 - Google Patents

脂肪族含窒素五員環化合物 Download PDF

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Publication number
JP4329290B2
JP4329290B2 JP2001309558A JP2001309558A JP4329290B2 JP 4329290 B2 JP4329290 B2 JP 4329290B2 JP 2001309558 A JP2001309558 A JP 2001309558A JP 2001309558 A JP2001309558 A JP 2001309558A JP 4329290 B2 JP4329290 B2 JP 4329290B2
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JP
Japan
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group
trans
cyano
cyclohexylamino
acetylpyrrolidine
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Expired - Fee Related
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JP2001309558A
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English (en)
Japanese (ja)
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JP2002356471A (ja
JP2002356471A5 (cg-RX-API-DMAC7.html
Inventor
公助 安田
啓氏 森本
三郎 河南
匡毅 彦田
健 松本
健司 荒川
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Mitsubishi Tanabe Pharma Corp
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Mitsubishi Tanabe Pharma Corp
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Priority to JP2001309558A priority Critical patent/JP4329290B2/ja
Publication of JP2002356471A publication Critical patent/JP2002356471A/ja
Publication of JP2002356471A5 publication Critical patent/JP2002356471A5/ja
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Publication of JP4329290B2 publication Critical patent/JP4329290B2/ja
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Expired - Fee Related legal-status Critical Current

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  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
JP2001309558A 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物 Expired - Fee Related JP4329290B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
JP2000308528 2000-10-06
JP2000-308528 2000-10-06
JP2000312562 2000-10-12
JP2000-312562 2000-10-12
JP2001099251 2001-03-30
JP2001-99251 2001-03-30
JP2001309558A JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2003368572A Division JP2004035574A (ja) 2000-10-06 2003-10-29 脂肪族含窒素五員環化合物

Publications (3)

Publication Number Publication Date
JP2002356471A JP2002356471A (ja) 2002-12-13
JP2002356471A5 JP2002356471A5 (cg-RX-API-DMAC7.html) 2004-10-28
JP4329290B2 true JP4329290B2 (ja) 2009-09-09

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JP2001309558A Expired - Fee Related JP4329290B2 (ja) 2000-10-06 2001-10-05 脂肪族含窒素五員環化合物

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JP (1) JP4329290B2 (cg-RX-API-DMAC7.html)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10213051B4 (de) * 2002-03-23 2013-03-07 Grünenthal GmbH Substituierte 4-Aminocyclohexanole
US20050197350A1 (en) * 2003-03-31 2005-09-08 Taisho Pharmaceutical Co., Ltd. Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof
KR101130433B1 (ko) 2004-02-05 2012-03-27 교린 세이야꾸 가부시키 가이샤 비시클로에스테르 유도체
DE102004023632A1 (de) * 2004-05-10 2005-12-08 Grünenthal GmbH Substituierte Cyclohexylcarbonsäure-Derivate
WO2006040625A1 (en) * 2004-10-12 2006-04-20 Glenmark Pharmaceuticals S.A. Novel dipeptidyl peptidase iv inhibitors, pharmaceutical compositions containing them, and process for their preparation
DOP2006000008A (es) 2005-01-10 2006-08-31 Arena Pharm Inc Terapia combinada para el tratamiento de la diabetes y afecciones relacionadas y para el tratamiento de afecciones que mejoran mediante un incremento de la concentración sanguínea de glp-1
EP1995237A4 (en) 2006-03-08 2011-07-06 Kyorin Seiyaku Kk PROCESS FOR PREPARING AN AMINOACETYLPYRROLIDINCARBONITRILE DERIVATIVE AND PRODUCTION PRODUCT THEREOF
EP2410330A3 (en) 2006-04-11 2012-06-13 Arena Pharmaceuticals, Inc. Methods of using GPR119 receptor to identify compounds useful for increasing bone mass in an individual
PE20071221A1 (es) 2006-04-11 2007-12-14 Arena Pharm Inc Agonistas del receptor gpr119 en metodos para aumentar la masa osea y para tratar la osteoporosis y otras afecciones caracterizadas por masa osea baja, y la terapia combinada relacionada a estos agonistas
WO2008066083A1 (fr) * 2006-11-29 2008-06-05 Mitsubishi Tanabe Pharma Corporation Procédé de production d'un dérivé de n-(n'-glycyle substitué)-2-cyanopyrrolidine
JPWO2008114857A1 (ja) 2007-03-22 2010-07-08 杏林製薬株式会社 アミノアセチルピロリジンカルボニトリル誘導体の製造方法
EA201070839A1 (ru) * 2008-01-10 2010-12-30 Сан Фарма Адвансед Ресьёрч Компани Лимитед Новые производные ацилцианопирролидинов
EP2108960A1 (en) 2008-04-07 2009-10-14 Arena Pharmaceuticals, Inc. Methods of using A G protein-coupled receptor to identify peptide YY (PYY) secretagogues and compounds useful in the treatment of conditons modulated by PYY
CA2732984A1 (en) 2008-08-07 2010-02-11 Kyorin Pharmaceutical Co., Ltd. Process for production of bicyclo[2.2.2]octylamine derivative
AR077642A1 (es) 2009-07-09 2011-09-14 Arena Pharm Inc Moduladores del metabolismo y el tratamiento de trastornos relacionados con el mismo
JP2013523819A (ja) 2010-04-06 2013-06-17 アリーナ ファーマシューティカルズ， インコーポレイテッド Ｇｐｒ１１９レセプターのモジュレーターおよびそれに関連する障害の処置
EP3323818A1 (en) 2010-09-22 2018-05-23 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012135570A1 (en) 2011-04-01 2012-10-04 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145361A1 (en) 2011-04-19 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145604A1 (en) 2011-04-22 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2012145603A1 (en) 2011-04-22 2012-10-26 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
HUE064883T2 (hu) * 2011-04-22 2024-04-28 Signal Pharm Llc Szubsztituált diaminokarboxamid- és diaminokarbonitril-pirimidinek, azok készítményei és azokkal történõ kezelési eljárások
WO2012170702A1 (en) 2011-06-08 2012-12-13 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2013055910A1 (en) 2011-10-12 2013-04-18 Arena Pharmaceuticals, Inc. Modulators of the gpr119 receptor and the treatment of disorders related thereto
WO2014074668A1 (en) 2012-11-08 2014-05-15 Arena Pharmaceuticals, Inc. Modulators of gpr119 and the treatment of disorders related thereto
HK1249847A1 (zh) 2015-03-09 2018-11-16 Intekrin Therapeutics, Inc. 用於治疗非酒精性脂肪肝疾病和/或脂肪营养不良的方法
BR112019020485A2 (pt) 2017-04-03 2020-05-12 Coherus Biosciences, Inc. Agonista ppary para tratamento de paralisia supranuclear progressiva
US11214540B2 (en) 2017-05-15 2022-01-04 Cognition Therapeutics, Inc. Compositions for treating neurodegenerative diseases

Also Published As

Publication number Publication date
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