JP2926257B2 - 抗ウイルス性で高い水溶性を持ち且つ安定な結晶性２′，３′‐ジデオキシイノシン・モノ水和物塩、２′，３′‐ジデオキシ‐２′，３′‐ジデヒドロチミジン・モノ水和物塩及び２′，３′‐ジデオキシ‐２′‐フルオロイノシン・ヘミ水和物塩 - Google Patents

抗ウイルス性で高い水溶性を持ち且つ安定な結晶性２′，３′‐ジデオキシイノシン・モノ水和物塩、２′，３′‐ジデオキシ‐２′，３′‐ジデヒドロチミジン・モノ水和物塩及び２′，３′‐ジデオキシ‐２′‐フルオロイノシン・ヘミ水和物塩

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Publication number
JP2926257B2
JP2926257B2 JP12326390A JP12326390A JP2926257B2 JP 2926257 B2 JP2926257 B2 JP 2926257B2 JP 12326390 A JP12326390 A JP 12326390A JP 12326390 A JP12326390 A JP 12326390A JP 2926257 B2 JP2926257 B2 JP 2926257B2
Authority
JP
Japan
Prior art keywords
salt
dideoxy
didehydrothymidine
dideoxyinosine
fluoroinosine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP12326390A
Other languages
English (en)
Japanese (ja)
Other versions
JPH035477A (ja
Inventor
アーサー カプラン マーレイ
ケビン ペロン ロバート
バラード ボーガルダス ジヨセフ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BURISUTORU MAIYAAZU SUKUIBU CO
Original Assignee
BURISUTORU MAIYAAZU SUKUIBU CO
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BURISUTORU MAIYAAZU SUKUIBU CO filed Critical BURISUTORU MAIYAAZU SUKUIBU CO
Publication of JPH035477A publication Critical patent/JPH035477A/ja
Application granted granted Critical
Publication of JP2926257B2 publication Critical patent/JP2926257B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP12326390A 1989-05-15 1990-05-15 抗ウイルス性で高い水溶性を持ち且つ安定な結晶性２′，３′‐ジデオキシイノシン・モノ水和物塩、２′，３′‐ジデオキシ‐２′，３′‐ジデヒドロチミジン・モノ水和物塩及び２′，３′‐ジデオキシ‐２′‐フルオロイノシン・ヘミ水和物塩 Expired - Lifetime JP2926257B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35206589A 1989-05-15 1989-05-15
US352065 1989-05-15

Publications (2)

Publication Number Publication Date
JPH035477A JPH035477A (ja) 1991-01-11
JP2926257B2 true JP2926257B2 (ja) 1999-07-28

Family

ID=23383649

Family Applications (1)

Application Number Title Priority Date Filing Date
JP12326390A Expired - Lifetime JP2926257B2 (ja) 1989-05-15 1990-05-15 抗ウイルス性で高い水溶性を持ち且つ安定な結晶性２′，３′‐ジデオキシイノシン・モノ水和物塩、２′，３′‐ジデオキシ‐２′，３′‐ジデヒドロチミジン・モノ水和物塩及び２′，３′‐ジデオキシ‐２′‐フルオロイノシン・ヘミ水和物塩

Country Status (11)

Country Link
JP (1) JP2926257B2 (cg-RX-API-DMAC7.html)
CA (1) CA2016765C (cg-RX-API-DMAC7.html)
CZ (1) CZ9602347A3 (cg-RX-API-DMAC7.html)
DD (1) DD298406A5 (cg-RX-API-DMAC7.html)
MY (1) MY116824A (cg-RX-API-DMAC7.html)
NZ (1) NZ233646A (cg-RX-API-DMAC7.html)
PL (1) PL163999B1 (cg-RX-API-DMAC7.html)
SK (2) SK279130B6 (cg-RX-API-DMAC7.html)
TW (1) TW233301B (cg-RX-API-DMAC7.html)
YU (1) YU92890A (cg-RX-API-DMAC7.html)
ZA (1) ZA903662B (cg-RX-API-DMAC7.html)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7122207B2 (en) 1998-05-22 2006-10-17 Bristol-Myers Squibb Company High drug load acid labile pharmaceutical composition
JP4731121B2 (ja) * 2004-02-02 2011-07-20 協和発酵キリン株式会社 キサンチン誘導体水和物
WO2009119785A1 (ja) * 2008-03-28 2009-10-01 浜理薬品工業株式会社 エチニルチミジン化合物の精製方法
JP5485140B2 (ja) * 2008-04-10 2014-05-07 浜理薬品工業株式会社 ５−メチルウリジンを出発原料とするエチニルチミジン化合物の製造方法

Also Published As

Publication number Publication date
CA2016765A1 (en) 1990-11-15
CA2016765C (en) 1997-10-21
SK127397A3 (en) 1998-08-05
TW233301B (cg-RX-API-DMAC7.html) 1994-11-01
PL285175A1 (en) 1991-01-14
NZ233646A (en) 1991-10-25
PL163999B1 (pl) 1994-06-30
YU92890A (sh) 1992-09-07
CZ288463B6 (en) 2001-06-13
SK279253B6 (sk) 1998-08-05
JPH035477A (ja) 1991-01-11
DD298406A5 (de) 1992-02-20
CZ9602347A3 (en) 2001-06-13
SK237290A3 (en) 1998-07-08
SK279130B6 (sk) 1998-07-08
MY116824A (en) 2004-04-30
ZA903662B (en) 1991-01-30

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