JP2025512999A5 - - Google Patents

Info

Publication number
JP2025512999A5
JP2025512999A5 JP2024559459A JP2024559459A JP2025512999A5 JP 2025512999 A5 JP2025512999 A5 JP 2025512999A5 JP 2024559459 A JP2024559459 A JP 2024559459A JP 2024559459 A JP2024559459 A JP 2024559459A JP 2025512999 A5 JP2025512999 A5 JP 2025512999A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
cancer
composition according
inhibitor
adenocarcinoma
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024559459A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025512999A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/015097 external-priority patent/WO2023196086A2/en
Publication of JP2025512999A publication Critical patent/JP2025512999A/ja
Publication of JP2025512999A5 publication Critical patent/JP2025512999A5/ja
Pending legal-status Critical Current

Links

JP2024559459A 2022-04-08 2023-03-13 Sos1阻害剤及びegfr阻害剤を含む併用療法 Pending JP2025512999A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263329090P 2022-04-08 2022-04-08
US63/329,090 2022-04-08
PCT/US2023/015097 WO2023196086A2 (en) 2022-04-08 2023-03-13 Combination therapies comprising a sos1 inhibitor and an egfr inhibitor

Publications (2)

Publication Number Publication Date
JP2025512999A JP2025512999A (ja) 2025-04-22
JP2025512999A5 true JP2025512999A5 (https=) 2026-03-25

Family

ID=88243368

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024559459A Pending JP2025512999A (ja) 2022-04-08 2023-03-13 Sos1阻害剤及びegfr阻害剤を含む併用療法

Country Status (10)

Country Link
US (1) US20250177410A1 (https=)
EP (1) EP4504171A4 (https=)
JP (1) JP2025512999A (https=)
KR (1) KR20240170920A (https=)
CN (1) CN119031916A (https=)
AU (1) AU2023250819A1 (https=)
CA (1) CA3245678A1 (https=)
IL (1) IL315645A (https=)
MX (1) MX2024012445A (https=)
WO (1) WO2023196086A2 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022271679A1 (en) * 2021-06-21 2022-12-29 Mirati Therapeutics, Inc. Sos1 inhibitors
WO2025090810A1 (en) * 2023-10-25 2025-05-01 Kumquat Biosciences Inc. Use of sos1 inhibitors and amivantamab to treat cancer
WO2025090808A1 (en) * 2023-10-25 2025-05-01 Kumquat Biosciences Inc. Combinations of sos-1 inhibitors with osimertinib and/or met inhibitors to treat cancer

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1833803A4 (en) * 2005-01-03 2009-08-05 Myriad Genetics Inc PHARMACEUTICAL COMPOUNDS AS ACTIVATORS OF CASPASES AND INDUCTORS OF APOPTOSIS AND THEIR USE
WO2016077793A1 (en) * 2014-11-14 2016-05-19 Children's Hospital Medical Center Sos1 inhibitors for cancer treatment
EP3558979B1 (en) * 2016-12-22 2021-02-17 Boehringer Ingelheim International GmbH Novel benzylamino substituted quinazolines and derivatives as sos1 inhibitors
PH12022551513A1 (en) * 2019-12-20 2023-04-24 Mirati Therapeutics Inc Sos1 inhibitors
WO2022083657A1 (zh) * 2020-10-20 2022-04-28 苏州泽璟生物制药股份有限公司 取代苯并或吡啶并嘧啶胺类抑制剂及其制备方法和应用
CA3221608A1 (en) * 2021-06-14 2022-12-22 Kumquat Biosciences Inc. Fused heteroaryl compounds useful as anticancer agents

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