JP2024537136A5 - - Google Patents

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Publication number
JP2024537136A5
JP2024537136A5 JP2024520700A JP2024520700A JP2024537136A5 JP 2024537136 A5 JP2024537136 A5 JP 2024537136A5 JP 2024520700 A JP2024520700 A JP 2024520700A JP 2024520700 A JP2024520700 A JP 2024520700A JP 2024537136 A5 JP2024537136 A5 JP 2024537136A5
Authority
JP
Japan
Application number
JP2024520700A
Other languages
Japanese (ja)
Other versions
JPWO2023059596A5 (https=
JP2024537136A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/045621 external-priority patent/WO2023059596A1/en
Publication of JP2024537136A publication Critical patent/JP2024537136A/ja
Publication of JPWO2023059596A5 publication Critical patent/JPWO2023059596A5/ja
Publication of JP2024537136A5 publication Critical patent/JP2024537136A5/ja
Pending legal-status Critical Current

Links

JP2024520700A 2021-10-05 2022-10-04 KRAS G12D阻害剤と汎ErbBファミリー阻害剤との併用療法 Pending JP2024537136A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163252534P 2021-10-05 2021-10-05
US63/252,534 2021-10-05
PCT/US2022/045621 WO2023059596A1 (en) 2021-10-05 2022-10-04 COMBINATION THERAPIES OF KRAS G12D INHIBITORS WITH Pan ErbB FAMILY INHIBITORS

Publications (3)

Publication Number Publication Date
JP2024537136A JP2024537136A (ja) 2024-10-10
JPWO2023059596A5 JPWO2023059596A5 (https=) 2025-10-10
JP2024537136A5 true JP2024537136A5 (https=) 2025-10-10

Family

ID=85803674

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024520700A Pending JP2024537136A (ja) 2021-10-05 2022-10-04 KRAS G12D阻害剤と汎ErbBファミリー阻害剤との併用療法

Country Status (10)

Country Link
US (1) US20240408099A1 (https=)
EP (1) EP4412717A4 (https=)
JP (1) JP2024537136A (https=)
KR (1) KR20240089340A (https=)
CN (1) CN118369119A (https=)
AU (1) AU2022359880A1 (https=)
CA (1) CA3233567A1 (https=)
IL (1) IL311835A (https=)
MX (1) MX2024004216A (https=)
WO (1) WO2023059596A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2024543879A (ja) * 2021-11-24 2024-11-26 メルク・シャープ・アンド・ドーム・エルエルシー Kras変異型タンパク質の小分子阻害剤
WO2025034919A1 (en) * 2023-08-08 2025-02-13 Quanta Therapeutics, Inc. Combination therapies with kras modulators
AU2024337913A1 (en) 2023-09-08 2026-03-26 Gilead Sciences, Inc. Pyrimidine-containing polycyclic derivatives as kras g12d modulating compounds
US20250114339A1 (en) 2023-10-09 2025-04-10 Incyte Corporation Combination therapy comprising a kras g12d inhibitor and an egfr inhibitor
AU2024357850A1 (en) 2023-10-09 2026-04-23 Incyte Corporation Combination therapy using a kras g12d inhibitor and pd-1 inhibitor or pd-l1 inhibitor
WO2025145207A1 (en) 2023-12-29 2025-07-03 Bristol-Myers Squibb Company Combination therapy of kras inhibitor and treg-depleting agent
WO2026060400A1 (en) * 2024-09-16 2026-03-19 Quanta Therapeutics, Inc. Combination therapies with kras modulators

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2013234767B2 (en) 2012-03-19 2017-02-23 Merck Patent Gmbh Combination of a 6-oxo-1,6-dihydro-pyridazine derivative having anti-cancer activity with other anti-tumor compounds
CA3112043A1 (en) 2018-09-10 2020-03-19 Mirati Therapeutics, Inc. Combination therapies
WO2020146613A1 (en) 2019-01-10 2020-07-16 Mirati Therapeutics, Inc. Kras g12c inhibitors
WO2021041671A1 (en) 2019-08-29 2021-03-04 Mirati Therapeutics, Inc. Kras g12d inhibitors
WO2021106231A1 (en) * 2019-11-29 2021-06-03 Taiho Pharmaceutical Co., Ltd. A compound having inhibitory activity against kras g12d mutation
WO2023284730A1 (en) * 2021-07-14 2023-01-19 Nikang Therapeutics, Inc. Alkylidene derivatives as kras inhibitors

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