JP2025511974A5 - - Google Patents
Info
- Publication number
- JP2025511974A5 JP2025511974A5 JP2024559703A JP2024559703A JP2025511974A5 JP 2025511974 A5 JP2025511974 A5 JP 2025511974A5 JP 2024559703 A JP2024559703 A JP 2024559703A JP 2024559703 A JP2024559703 A JP 2024559703A JP 2025511974 A5 JP2025511974 A5 JP 2025511974A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- cycloalkyl
- group
- halogen
- cancer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP22166685 | 2022-04-05 | ||
| EP22166685.2 | 2022-04-05 | ||
| PCT/EP2023/058978 WO2023194458A1 (en) | 2022-04-05 | 2023-04-05 | N-(3-(benzo[b]thiophene-2-carboxamido)-phenyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide derivatives and related compounds as lactate/atp production inhibitors for the treatment of cancer |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025511974A JP2025511974A (ja) | 2025-04-16 |
| JP2025511974A5 true JP2025511974A5 (https=) | 2026-04-13 |
Family
ID=81328159
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024559703A Pending JP2025511974A (ja) | 2022-04-05 | 2023-04-05 | がんの治療のためのラクテート/ATP産生阻害剤としてのN-(3-(ベンゾ[b]チオフェン-2-カルボキシアミド)-フェニル)-2,3-ジヒドロベンゾ[b][1,4]ジオキシン-6-カルボキシアミド誘導体及び関連化合物 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20260028334A1 (https=) |
| EP (1) | EP4504723A1 (https=) |
| JP (1) | JP2025511974A (https=) |
| KR (1) | KR20240172217A (https=) |
| CN (1) | CN118974040A (https=) |
| AU (1) | AU2023248671A1 (https=) |
| CA (1) | CA3246966A1 (https=) |
| IL (1) | IL316122A (https=) |
| MX (1) | MX2024012179A (https=) |
| WO (1) | WO2023194458A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202523302A (zh) | 2023-11-02 | 2025-06-16 | 美商阿克思生物科學有限公司 | 噻唑化合物及其使用方法 |
| WO2025165930A1 (en) * | 2024-01-31 | 2025-08-07 | Biogen Ma Inc. | Methods for treating spinal muscular atrophy |
| JP7818251B2 (ja) * | 2024-02-29 | 2026-02-20 | 株式会社Moresco | オートファジー機能活性化化合物 |
| CN118340765B (zh) * | 2024-04-30 | 2024-08-23 | 广州市朝利良生物科技有限公司 | 苯甲酰胺类化合物在制备促伤口愈合药物中的应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2547072T3 (es) * | 2009-07-21 | 2015-10-01 | The Board Of Trustees Of The Leland Stanford Junior University | Heteroaril benzamidas, composiciones y métodos de utilización |
| GB201317609D0 (en) | 2013-10-04 | 2013-11-20 | Cancer Rec Tech Ltd | Inhibitor compounds |
| GB201505658D0 (en) | 2015-04-01 | 2015-05-13 | Cancer Rec Tech Ltd | Inhibitor compounds |
| GB201617103D0 (en) * | 2016-10-07 | 2016-11-23 | Cancer Research Technology Limited | Compound |
-
2023
- 2023-04-05 EP EP23718214.2A patent/EP4504723A1/en active Pending
- 2023-04-05 JP JP2024559703A patent/JP2025511974A/ja active Pending
- 2023-04-05 AU AU2023248671A patent/AU2023248671A1/en active Pending
- 2023-04-05 CA CA3246966A patent/CA3246966A1/en active Pending
- 2023-04-05 CN CN202380032324.0A patent/CN118974040A/zh active Pending
- 2023-04-05 KR KR1020247036954A patent/KR20240172217A/ko active Pending
- 2023-04-05 WO PCT/EP2023/058978 patent/WO2023194458A1/en not_active Ceased
- 2023-04-05 US US18/854,499 patent/US20260028334A1/en active Pending
- 2023-04-05 IL IL316122A patent/IL316122A/en unknown
-
2024
- 2024-10-02 MX MX2024012179A patent/MX2024012179A/es unknown
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