JP2025511974A5 - - Google Patents

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Publication number
JP2025511974A5
JP2025511974A5 JP2024559703A JP2024559703A JP2025511974A5 JP 2025511974 A5 JP2025511974 A5 JP 2025511974A5 JP 2024559703 A JP2024559703 A JP 2024559703A JP 2024559703 A JP2024559703 A JP 2024559703A JP 2025511974 A5 JP2025511974 A5 JP 2025511974A5
Authority
JP
Japan
Prior art keywords
alkyl
cycloalkyl
group
halogen
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024559703A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025511974A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/058978 external-priority patent/WO2023194458A1/en
Publication of JP2025511974A publication Critical patent/JP2025511974A/ja
Publication of JP2025511974A5 publication Critical patent/JP2025511974A5/ja
Pending legal-status Critical Current

Links

JP2024559703A 2022-04-05 2023-04-05 がんの治療のためのラクテート/ATP産生阻害剤としてのN-(3-(ベンゾ[b]チオフェン-2-カルボキシアミド)-フェニル)-2,3-ジヒドロベンゾ[b][1,4]ジオキシン-6-カルボキシアミド誘導体及び関連化合物 Pending JP2025511974A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP22166685 2022-04-05
EP22166685.2 2022-04-05
PCT/EP2023/058978 WO2023194458A1 (en) 2022-04-05 2023-04-05 N-(3-(benzo[b]thiophene-2-carboxamido)-phenyl)-2,3-dihydrobenzo[b][1,4]dioxine-6-carboxamide derivatives and related compounds as lactate/atp production inhibitors for the treatment of cancer

Publications (2)

Publication Number Publication Date
JP2025511974A JP2025511974A (ja) 2025-04-16
JP2025511974A5 true JP2025511974A5 (https=) 2026-04-13

Family

ID=81328159

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024559703A Pending JP2025511974A (ja) 2022-04-05 2023-04-05 がんの治療のためのラクテート/ATP産生阻害剤としてのN-(3-(ベンゾ[b]チオフェン-2-カルボキシアミド)-フェニル)-2,3-ジヒドロベンゾ[b][1,4]ジオキシン-6-カルボキシアミド誘導体及び関連化合物

Country Status (10)

Country Link
US (1) US20260028334A1 (https=)
EP (1) EP4504723A1 (https=)
JP (1) JP2025511974A (https=)
KR (1) KR20240172217A (https=)
CN (1) CN118974040A (https=)
AU (1) AU2023248671A1 (https=)
CA (1) CA3246966A1 (https=)
IL (1) IL316122A (https=)
MX (1) MX2024012179A (https=)
WO (1) WO2023194458A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202523302A (zh) 2023-11-02 2025-06-16 美商阿克思生物科學有限公司 噻唑化合物及其使用方法
WO2025165930A1 (en) * 2024-01-31 2025-08-07 Biogen Ma Inc. Methods for treating spinal muscular atrophy
JP7818251B2 (ja) * 2024-02-29 2026-02-20 株式会社Moresco オートファジー機能活性化化合物
CN118340765B (zh) * 2024-04-30 2024-08-23 广州市朝利良生物科技有限公司 苯甲酰胺类化合物在制备促伤口愈合药物中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2547072T3 (es) * 2009-07-21 2015-10-01 The Board Of Trustees Of The Leland Stanford Junior University Heteroaril benzamidas, composiciones y métodos de utilización
GB201317609D0 (en) 2013-10-04 2013-11-20 Cancer Rec Tech Ltd Inhibitor compounds
GB201505658D0 (en) 2015-04-01 2015-05-13 Cancer Rec Tech Ltd Inhibitor compounds
GB201617103D0 (en) * 2016-10-07 2016-11-23 Cancer Research Technology Limited Compound

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