JP2025508932A5 - - Google Patents

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Publication number
JP2025508932A5
JP2025508932A5 JP2024551922A JP2024551922A JP2025508932A5 JP 2025508932 A5 JP2025508932 A5 JP 2025508932A5 JP 2024551922 A JP2024551922 A JP 2024551922A JP 2024551922 A JP2024551922 A JP 2024551922A JP 2025508932 A5 JP2025508932 A5 JP 2025508932A5
Authority
JP
Japan
Prior art keywords
subject
pharmaceutical composition
heart disease
person suffering
grk5
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024551922A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508932A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/063451 external-priority patent/WO2023168246A2/en
Publication of JP2025508932A publication Critical patent/JP2025508932A/ja
Publication of JP2025508932A5 publication Critical patent/JP2025508932A5/ja
Pending legal-status Critical Current

Links

JP2024551922A 2022-03-01 2023-03-01 選択的gタンパク質共役受容体キナーゼ5阻害剤、組成物、及び使用方法 Pending JP2025508932A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263315118P 2022-03-01 2022-03-01
US63/315,118 2022-03-01
PCT/US2023/063451 WO2023168246A2 (en) 2022-03-01 2023-03-01 Selective g protein-coupled receptor kinase 5 inhibitors, compositions, and methods of use

Publications (2)

Publication Number Publication Date
JP2025508932A JP2025508932A (ja) 2025-04-10
JP2025508932A5 true JP2025508932A5 (enExample) 2026-03-05

Family

ID=87884331

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024551922A Pending JP2025508932A (ja) 2022-03-01 2023-03-01 選択的gタンパク質共役受容体キナーゼ5阻害剤、組成物、及び使用方法

Country Status (9)

Country Link
US (1) US20250388567A1 (enExample)
EP (1) EP4486335A4 (enExample)
JP (1) JP2025508932A (enExample)
KR (1) KR20240169624A (enExample)
CN (1) CN118891039A (enExample)
AU (1) AU2023228660A1 (enExample)
CA (1) CA3244988A1 (enExample)
IL (1) IL315279A (enExample)
WO (1) WO2023168246A2 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN119350363A (zh) * 2024-10-22 2025-01-24 中国药科大学 一类protac分子及其应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR035721A1 (es) * 2000-12-20 2004-07-07 Sugen Inc Indolinonas 4-aril sustituidas; sus composiciones farmaceuticas y metodo para modular la actividad catalitica de una proteina quinasa
CN102276584A (zh) * 2010-06-08 2011-12-14 齐鲁制药有限公司 吡咯取代的2-二氢吲哚酮衍生物、其制备方法及用途
CN103012428A (zh) * 2013-01-08 2013-04-03 中国药科大学 4-(五元杂环并嘧啶/吡啶取代)氨基-1H-3-吡唑甲酰胺类CDK/Aurora双重抑制剂及其用途
EP2837626A1 (en) * 2013-08-16 2015-02-18 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Indolinone derivatives as GRK5 modulators
WO2021243040A2 (en) * 2020-05-29 2021-12-02 The Regents Of The University Of Michigan Small molecule inhibitors of grk5 and grk5 subfamily members and uses thereof

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