JP2025508932A5 - - Google Patents
Info
- Publication number
- JP2025508932A5 JP2025508932A5 JP2024551922A JP2024551922A JP2025508932A5 JP 2025508932 A5 JP2025508932 A5 JP 2025508932A5 JP 2024551922 A JP2024551922 A JP 2024551922A JP 2024551922 A JP2024551922 A JP 2024551922A JP 2025508932 A5 JP2025508932 A5 JP 2025508932A5
- Authority
- JP
- Japan
- Prior art keywords
- subject
- pharmaceutical composition
- heart disease
- person suffering
- grk5
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202263315118P | 2022-03-01 | 2022-03-01 | |
| US63/315,118 | 2022-03-01 | ||
| PCT/US2023/063451 WO2023168246A2 (en) | 2022-03-01 | 2023-03-01 | Selective g protein-coupled receptor kinase 5 inhibitors, compositions, and methods of use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025508932A JP2025508932A (ja) | 2025-04-10 |
| JP2025508932A5 true JP2025508932A5 (enExample) | 2026-03-05 |
Family
ID=87884331
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024551922A Pending JP2025508932A (ja) | 2022-03-01 | 2023-03-01 | 選択的gタンパク質共役受容体キナーゼ5阻害剤、組成物、及び使用方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20250388567A1 (enExample) |
| EP (1) | EP4486335A4 (enExample) |
| JP (1) | JP2025508932A (enExample) |
| KR (1) | KR20240169624A (enExample) |
| CN (1) | CN118891039A (enExample) |
| AU (1) | AU2023228660A1 (enExample) |
| CA (1) | CA3244988A1 (enExample) |
| IL (1) | IL315279A (enExample) |
| WO (1) | WO2023168246A2 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN119350363A (zh) * | 2024-10-22 | 2025-01-24 | 中国药科大学 | 一类protac分子及其应用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR035721A1 (es) * | 2000-12-20 | 2004-07-07 | Sugen Inc | Indolinonas 4-aril sustituidas; sus composiciones farmaceuticas y metodo para modular la actividad catalitica de una proteina quinasa |
| CN102276584A (zh) * | 2010-06-08 | 2011-12-14 | 齐鲁制药有限公司 | 吡咯取代的2-二氢吲哚酮衍生物、其制备方法及用途 |
| CN103012428A (zh) * | 2013-01-08 | 2013-04-03 | 中国药科大学 | 4-(五元杂环并嘧啶/吡啶取代)氨基-1H-3-吡唑甲酰胺类CDK/Aurora双重抑制剂及其用途 |
| EP2837626A1 (en) * | 2013-08-16 | 2015-02-18 | Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. | Indolinone derivatives as GRK5 modulators |
| WO2021243040A2 (en) * | 2020-05-29 | 2021-12-02 | The Regents Of The University Of Michigan | Small molecule inhibitors of grk5 and grk5 subfamily members and uses thereof |
-
2023
- 2023-03-01 US US18/843,111 patent/US20250388567A1/en active Pending
- 2023-03-01 EP EP23764065.1A patent/EP4486335A4/en active Pending
- 2023-03-01 IL IL315279A patent/IL315279A/en unknown
- 2023-03-01 CN CN202380024914.9A patent/CN118891039A/zh active Pending
- 2023-03-01 WO PCT/US2023/063451 patent/WO2023168246A2/en not_active Ceased
- 2023-03-01 JP JP2024551922A patent/JP2025508932A/ja active Pending
- 2023-03-01 AU AU2023228660A patent/AU2023228660A1/en active Pending
- 2023-03-01 CA CA3244988A patent/CA3244988A1/en active Pending
- 2023-03-01 KR KR1020247032184A patent/KR20240169624A/ko active Pending
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