JP2022552881A5 - - Google Patents

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Publication number
JP2022552881A5
JP2022552881A5 JP2022523519A JP2022523519A JP2022552881A5 JP 2022552881 A5 JP2022552881 A5 JP 2022552881A5 JP 2022523519 A JP2022523519 A JP 2022523519A JP 2022523519 A JP2022523519 A JP 2022523519A JP 2022552881 A5 JP2022552881 A5 JP 2022552881A5
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JP
Japan
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day
pharmaceutical composition
cycle
approximately
administered
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JP2022523519A
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English (en)
Japanese (ja)
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JP2022552881A (ja
JP7581345B2 (ja
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Priority claimed from PCT/US2020/056409 external-priority patent/WO2021080936A1/en
Publication of JP2022552881A publication Critical patent/JP2022552881A/ja
Publication of JP2022552881A5 publication Critical patent/JP2022552881A5/ja
Application granted granted Critical
Publication of JP7581345B2 publication Critical patent/JP7581345B2/ja
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JP2022523519A 2019-10-21 2020-10-20 2-(2,6-ジオキソピペリジン-3-イル)-4-((2-フルオロ-4-((3-モルホリノアゼチジン-1-イル)メチル)ベンジル)アミノ)イソインドリン-1,3-ジオンを用いて慢性リンパ性白血病を治療する方法 Active JP7581345B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962923955P 2019-10-21 2019-10-21
US62/923,955 2019-10-21
US202063011147P 2020-04-16 2020-04-16
US63/011,147 2020-04-16
PCT/US2020/056409 WO2021080936A1 (en) 2019-10-21 2020-10-20 Methods of treating chronic lymphocytic leukemia using 2-(2,6-dioxopiperidin-3yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isoindoline-1. 3-dione

Publications (3)

Publication Number Publication Date
JP2022552881A JP2022552881A (ja) 2022-12-20
JP2022552881A5 true JP2022552881A5 (enExample) 2023-10-20
JP7581345B2 JP7581345B2 (ja) 2024-11-12

Family

ID=73452273

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022523519A Active JP7581345B2 (ja) 2019-10-21 2020-10-20 2-(2,6-ジオキソピペリジン-3-イル)-4-((2-フルオロ-4-((3-モルホリノアゼチジン-1-イル)メチル)ベンジル)アミノ)イソインドリン-1,3-ジオンを用いて慢性リンパ性白血病を治療する方法

Country Status (13)

Country Link
US (2) US11628172B2 (enExample)
EP (1) EP4048279B1 (enExample)
JP (1) JP7581345B2 (enExample)
KR (1) KR20220103953A (enExample)
CN (2) CN115919870B (enExample)
AU (1) AU2020369497C1 (enExample)
CA (1) CA3154510A1 (enExample)
CL (1) CL2022000991A1 (enExample)
ES (1) ES3066029T3 (enExample)
IL (1) IL292265B2 (enExample)
MX (1) MX2022004727A (enExample)
WO (1) WO2021080936A1 (enExample)
ZA (1) ZA202204446B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SMT202600194T1 (it) 2019-10-21 2026-05-12 Celgene Corp Combinazione di composti di 4-amminoisoindolin-1,3-dione sostituiti e di secondi agenti attivi per l'uso nel trattamento di una condizione maligna ematologica
CA3154504A1 (en) 2019-10-21 2021-04-29 Maria Soraya Carrancio ANTON Methods of treating hematological malignancies using 2-(2,6-dioxopiperidin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino )isoindoline-1,3-dione
US11628172B2 (en) * 2019-10-21 2023-04-18 Celgene Corporation Methods of treating chronic lymphocytic leukemia using 2-(2,6-dioxopiperidin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isoindoline-1,3-dione
BR112022007580A2 (pt) 2019-10-21 2022-07-05 Celgene Corp Formas sólidas que compreendem (s)-2-(2,6-dioxopiperidin-3-il)-4-((2-fluoro-4-((3-morfolinoazetidin-1-il)metil)benzil)amino)isoindolino-1,3-diona e seus sais e composições que compreendem as mesmas e seus usos
KR20220103952A (ko) * 2019-10-21 2022-07-25 셀진 코포레이션 (s)-2-(2,6-디옥소피페리딘-3-일)-4-((2-플루오로-4-((3-모르폴리노아제티딘-1-일)메틸)벤질)아미노)이소인돌린-1,3-디온을 포함하는 제약 조성물 및 그의 사용 방법
IL292305A (en) * 2019-10-21 2022-06-01 Celgene Corp Methods for the treatment of hematological cancer and the use of associated biomarkers for 2-(2,6-deoxypyridin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isodonyl 1,3-discussion

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008033567A1 (en) 2006-09-15 2008-03-20 Celgene Corporation N-methylaminomethyl isoindole compounds and compositions comprising and methods of using the same
NZ772688A (en) * 2010-06-03 2022-09-30 Pharmacyclics Llc The use of inhibitors of bruton’s tyrosine kinase (btk)
CA2907908A1 (en) 2013-04-02 2014-10-09 Celgene Corporation Methods and compositions using 4-amino-2-(2,6-dioxo-piperidine-3-yl)-isoindoline-1,3-dione for treatment and management of central nervous system cancers
CA2954652A1 (en) 2014-07-11 2016-01-14 Celgene Corporation Combination therapy for cancer
FI3784663T3 (fi) * 2018-04-23 2023-10-06 Celgene Corp Substituoituja 4-aminoisoindoliini-1,3-dioniyhdisteitä ja niiden käyttö lymfooman hoitamiseksi
AR119715A1 (es) * 2019-04-12 2022-01-05 Celgene Corp Métodos para tratar linfoma no hodgkin con el uso de 2-(2,6-dioxopiperidin-3-il)-4-((2-fluoro-4-((3-morfolinoazetidin-1-il)metil)bencil)amino)isoindolin-1,3-diona
SMT202600194T1 (it) * 2019-10-21 2026-05-12 Celgene Corp Combinazione di composti di 4-amminoisoindolin-1,3-dione sostituiti e di secondi agenti attivi per l'uso nel trattamento di una condizione maligna ematologica
CA3154504A1 (en) * 2019-10-21 2021-04-29 Maria Soraya Carrancio ANTON Methods of treating hematological malignancies using 2-(2,6-dioxopiperidin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino )isoindoline-1,3-dione
US11628172B2 (en) * 2019-10-21 2023-04-18 Celgene Corporation Methods of treating chronic lymphocytic leukemia using 2-(2,6-dioxopiperidin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isoindoline-1,3-dione
KR20220103952A (ko) * 2019-10-21 2022-07-25 셀진 코포레이션 (s)-2-(2,6-디옥소피페리딘-3-일)-4-((2-플루오로-4-((3-모르폴리노아제티딘-1-일)메틸)벤질)아미노)이소인돌린-1,3-디온을 포함하는 제약 조성물 및 그의 사용 방법
IL292305A (en) * 2019-10-21 2022-06-01 Celgene Corp Methods for the treatment of hematological cancer and the use of associated biomarkers for 2-(2,6-deoxypyridin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isodonyl 1,3-discussion

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