JP2025508896A5 - - Google Patents

Info

Publication number
JP2025508896A5
JP2025508896A5 JP2024550789A JP2024550789A JP2025508896A5 JP 2025508896 A5 JP2025508896 A5 JP 2025508896A5 JP 2024550789 A JP2024550789 A JP 2024550789A JP 2024550789 A JP2024550789 A JP 2024550789A JP 2025508896 A5 JP2025508896 A5 JP 2025508896A5
Authority
JP
Japan
Prior art keywords
inhibitor
ctps1
bcl2
pharmaceutically acceptable
composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024550789A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508896A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/055217 external-priority patent/WO2023166076A1/en
Publication of JP2025508896A publication Critical patent/JP2025508896A/ja
Publication of JP2025508896A5 publication Critical patent/JP2025508896A5/ja
Pending legal-status Critical Current

Links

JP2024550789A 2022-03-01 2023-03-01 癌のためのctps1阻害剤とbcl2阻害剤の組合せ Pending JP2025508896A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP22305225.9 2022-03-01
EP22305225 2022-03-01
EP22306429.6 2022-09-27
EP22306429 2022-09-27
PCT/EP2023/055217 WO2023166076A1 (en) 2022-03-01 2023-03-01 Combinations of ctps1 and bcl2 inhibitors for cancer

Publications (2)

Publication Number Publication Date
JP2025508896A JP2025508896A (ja) 2025-04-10
JP2025508896A5 true JP2025508896A5 (https=) 2026-03-09

Family

ID=85384465

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024550789A Pending JP2025508896A (ja) 2022-03-01 2023-03-01 癌のためのctps1阻害剤とbcl2阻害剤の組合せ

Country Status (6)

Country Link
US (1) US20250177394A1 (https=)
EP (1) EP4486347A1 (https=)
JP (1) JP2025508896A (https=)
AU (1) AU2023228045A1 (https=)
CA (1) CA3244038A1 (https=)
WO (1) WO2023166076A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019106156A1 (en) 2017-11-30 2019-06-06 Step Pharma S.A.S. Compounds
IL288508B2 (en) 2019-06-04 2026-02-01 Step Pharma S A S History of n-(5-(6-ethoxypyrazin-2-yl)pyridin-2-yl)-4-(2-(methylsulfonamido)pyrimidin-4-yl)tetrahydro-h2-pyran-4-carboxamide and related compounds as human CTPS1 inhibitors for the treatment of proliferative diseases
WO2024133730A1 (en) * 2022-12-21 2024-06-27 Step Pharma S.A.S. Ctps1 inhibitors for use in the treatment of ctps2 deficient cancer

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3717465B1 (en) 2017-11-30 2026-01-21 Step Pharma S.A.S. Compounds
WO2019106156A1 (en) 2017-11-30 2019-06-06 Step Pharma S.A.S. Compounds
MX2020009887A (es) 2018-03-23 2020-10-12 Step Pharma S A S Derivados de aminopiridina como inhibidores de ctps1.
BR112021005986A2 (pt) 2018-10-23 2021-06-29 Step Pharma S.A.S. derivados de aminopirimidina como inibidores de ctps1
IL288508B2 (en) 2019-06-04 2026-02-01 Step Pharma S A S History of n-(5-(6-ethoxypyrazin-2-yl)pyridin-2-yl)-4-(2-(methylsulfonamido)pyrimidin-4-yl)tetrahydro-h2-pyran-4-carboxamide and related compounds as human CTPS1 inhibitors for the treatment of proliferative diseases
EP3980410B1 (en) 2019-06-04 2025-02-19 Step Pharma S.A.S. N-(4-(5-chloropyridin-3-yl)phenyl)-2-(2-(cyclopropanesulfonamido)pyrimidin-4-yl)butanamide derivatives and related compounds as human ctps1 inhibitors for the treatment of proliferative diseases
EP4041715A1 (en) 2019-09-20 2022-08-17 Step Pharma S.A.S. Sulfonamide inhibitors as ctps 1 inhibitors
WO2021053402A2 (en) 2019-09-20 2021-03-25 Step Pharma S.A.S. Compounds
US12331046B2 (en) 2020-10-23 2025-06-17 Nimbus Clotho, Inc. CTPS1 inhibitors and uses thereof

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