JP2025503592A5 - - Google Patents

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Publication number
JP2025503592A5
JP2025503592A5 JP2024540747A JP2024540747A JP2025503592A5 JP 2025503592 A5 JP2025503592 A5 JP 2025503592A5 JP 2024540747 A JP2024540747 A JP 2024540747A JP 2024540747 A JP2024540747 A JP 2024540747A JP 2025503592 A5 JP2025503592 A5 JP 2025503592A5
Authority
JP
Japan
Prior art keywords
alkyl
pharmaceutically acceptable
compound according
independently
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024540747A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025503592A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/060039 external-priority patent/WO2023133375A1/en
Publication of JP2025503592A publication Critical patent/JP2025503592A/ja
Publication of JP2025503592A5 publication Critical patent/JP2025503592A5/ja
Pending legal-status Critical Current

Links

JP2024540747A 2022-01-05 2023-01-03 大環状化合物およびキナーゼ阻害剤としての使用 Pending JP2025503592A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202263296705P 2022-01-05 2022-01-05
US63/296,705 2022-01-05
US202263435654P 2022-12-28 2022-12-28
US63/435,654 2022-12-28
PCT/US2023/060039 WO2023133375A1 (en) 2022-01-05 2023-01-03 Macrocyclic compounds and use as kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2025503592A JP2025503592A (ja) 2025-02-04
JP2025503592A5 true JP2025503592A5 (https=) 2026-01-14

Family

ID=87074235

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024540747A Pending JP2025503592A (ja) 2022-01-05 2023-01-03 大環状化合物およびキナーゼ阻害剤としての使用

Country Status (10)

Country Link
US (1) US20250074920A1 (https=)
EP (1) EP4460498A4 (https=)
JP (1) JP2025503592A (https=)
KR (1) KR20240131416A (https=)
AU (1) AU2023204770A1 (https=)
CA (1) CA3246487A1 (https=)
IL (1) IL314070A (https=)
MX (1) MX2024008413A (https=)
TW (1) TW202334168A (https=)
WO (1) WO2023133375A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2024266587A1 (en) * 2023-05-02 2025-09-11 Blossomhill Therapeutics, Inc. Egfr inhibitors for treating disease
WO2025212729A1 (en) * 2024-04-03 2025-10-09 Blossomhill Therapeutics, Inc. Macrocyclic compounds and their use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ME03376B (me) * 2010-05-20 2020-01-20 Array Biopharma Inc Makrociklička jedinjenja kао inhibiтori trk kinaze
US20160031888A1 (en) * 2013-03-13 2016-02-04 Boston Biomedical, Inc. 3-(aryl or heteroaryl) methyleneindolin-2-one derivatives as inhibitors of cancer stem cell pathway kinases for the treatment of cancer
ES2933350T3 (es) * 2014-01-24 2023-02-06 Turning Point Therapeutics Inc Macrociclos de diarilo como moduladores de proteína quinasas
TWI707852B (zh) * 2015-09-02 2020-10-21 美商林伯士拉克許米公司 Tyk2 抑制劑及其用途
EP4178958A4 (en) * 2020-07-10 2024-12-11 Blossomhill Therapeutics, Inc. MACROCYCLES AND THEIR USE

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