JP2024543452A5 - - Google Patents
Info
- Publication number
- JP2024543452A5 JP2024543452A5 JP2024527750A JP2024527750A JP2024543452A5 JP 2024543452 A5 JP2024543452 A5 JP 2024543452A5 JP 2024527750 A JP2024527750 A JP 2024527750A JP 2024527750 A JP2024527750 A JP 2024527750A JP 2024543452 A5 JP2024543452 A5 JP 2024543452A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- hydroxy
- thiadiazolidine
- dihydro
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163278339P | 2021-11-11 | 2021-11-11 | |
| US63/278,339 | 2021-11-11 | ||
| PCT/US2022/049584 WO2023086498A1 (en) | 2021-11-11 | 2022-11-10 | Protein tyrosine phosphatase inhibitors and methods of use thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024543452A JP2024543452A (ja) | 2024-11-21 |
| JP2024543452A5 true JP2024543452A5 (https=) | 2025-11-17 |
Family
ID=84689141
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024527750A Pending JP2024543452A (ja) | 2021-11-11 | 2022-11-10 | プロテインチロシンホスファターゼ阻害剤及びその使用方法 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20250019374A1 (https=) |
| EP (1) | EP4430038A1 (https=) |
| JP (1) | JP2024543452A (https=) |
| CN (1) | CN118525016A (https=) |
| AU (1) | AU2022387106A1 (https=) |
| CA (1) | CA3236854A1 (https=) |
| MX (1) | MX2024005658A (https=) |
| WO (1) | WO2023086498A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20252789A1 (es) | 2023-05-24 | 2025-12-22 | Kumquat Biosciences Inc | Compuestos heterociclicos y usos de estos |
| WO2025026158A1 (zh) * | 2023-07-28 | 2025-02-06 | 杭州中美华东制药有限公司 | 具有ptpn2抑制作用的化合物及其用途 |
| WO2025242216A1 (zh) * | 2024-05-24 | 2025-11-27 | 杭州百新生物医药科技有限公司 | 吲哚啉类化合物及其用途 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA94921C2 (en) * | 2005-12-08 | 2011-06-25 | Новартис Аг | 1-orthofluorophenyl substituted 1, 2, 5-thiazolidinedione derivatives as ptp-as inhibitors |
| UA94724C2 (en) * | 2005-12-08 | 2011-06-10 | Новартис Аг | Thiadiazolidinone derivatives as antidiabetic agents |
| BR112020026086A2 (pt) * | 2018-06-21 | 2021-03-23 | Calico Life Sciences Llc | inibidores da proteína tirosina fosfatase e métodos de uso destes |
| IL286373B2 (en) * | 2019-03-14 | 2026-03-01 | Calico Life Sciences Llc | Protein tyrosine phosphate inhibitor compounds and uses thereof |
| CA3162069A1 (en) * | 2019-12-18 | 2021-06-24 | Elliot P. Farney | Protein tyrosine phosphatase inhibitors and methods of use thereof |
-
2022
- 2022-11-10 WO PCT/US2022/049584 patent/WO2023086498A1/en not_active Ceased
- 2022-11-10 JP JP2024527750A patent/JP2024543452A/ja active Pending
- 2022-11-10 MX MX2024005658A patent/MX2024005658A/es unknown
- 2022-11-10 CA CA3236854A patent/CA3236854A1/en active Pending
- 2022-11-10 AU AU2022387106A patent/AU2022387106A1/en active Pending
- 2022-11-10 US US18/709,214 patent/US20250019374A1/en active Pending
- 2022-11-10 CN CN202280088273.9A patent/CN118525016A/zh active Pending
- 2022-11-10 EP EP22834767.0A patent/EP4430038A1/en active Pending
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