JP2024540525A5 - - Google Patents

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Publication number
JP2024540525A5
JP2024540525A5 JP2024529529A JP2024529529A JP2024540525A5 JP 2024540525 A5 JP2024540525 A5 JP 2024540525A5 JP 2024529529 A JP2024529529 A JP 2024529529A JP 2024529529 A JP2024529529 A JP 2024529529A JP 2024540525 A5 JP2024540525 A5 JP 2024540525A5
Authority
JP
Japan
Prior art keywords
methyl
pyrrolo
hexahydro
pharmaceutically acceptable
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024529529A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024540525A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/082174 external-priority patent/WO2023088987A1/en
Publication of JP2024540525A publication Critical patent/JP2024540525A/ja
Publication of JP2024540525A5 publication Critical patent/JP2024540525A5/ja
Pending legal-status Critical Current

Links

JP2024529529A 2021-11-19 2022-11-17 Nlrp3の阻害剤としてのピリダジン誘導体 Pending JP2024540525A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP21209168.0 2021-11-19
EP21209168 2021-11-19
EP22188185 2022-08-02
EP22188185.7 2022-08-02
PCT/EP2022/082174 WO2023088987A1 (en) 2021-11-19 2022-11-17 Pyridazine derivatives as inhibitors of nlrp3

Publications (2)

Publication Number Publication Date
JP2024540525A JP2024540525A (ja) 2024-10-31
JP2024540525A5 true JP2024540525A5 (enExample) 2025-11-17

Family

ID=84421135

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024529529A Pending JP2024540525A (ja) 2021-11-19 2022-11-17 Nlrp3の阻害剤としてのピリダジン誘導体

Country Status (6)

Country Link
US (1) US20240308977A1 (enExample)
EP (1) EP4433459A1 (enExample)
JP (1) JP2024540525A (enExample)
AR (1) AR127704A1 (enExample)
TW (1) TW202327603A (enExample)
WO (1) WO2023088987A1 (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11618751B1 (en) 2022-03-25 2023-04-04 Ventus Therapeutics U.S., Inc. Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 derivatives
US11319319B1 (en) 2021-04-07 2022-05-03 Ventus Therapeutics U.S., Inc. Compounds for inhibiting NLRP3 and uses thereof
JP2025523930A (ja) * 2022-07-21 2025-07-25 エフ. ホフマン-ラ ロシュ アーゲー Nlrp3阻害剤
US12331048B2 (en) 2022-10-31 2025-06-17 Ventus Therapeutics U.S., Inc. Pyrido-[3,4-d]pyridazine amine derivatives useful as NLRP3 inhibitors
US20260167637A1 (en) * 2022-11-04 2026-06-18 Transthera Sciences (Nanjing), Inc. Nlrp3 inflammasome inhibitor and use thereof
TW202545527A (zh) 2024-01-16 2025-12-01 英商諾得瑟拉公司 Nlrp3及glp-1a組合療法
WO2025229146A1 (en) * 2024-05-02 2025-11-06 Sanofi Crystalline form of a pyridazine nlrp3 inhibitor
WO2025247338A1 (zh) * 2024-05-30 2025-12-04 纽欧申医药(上海)有限公司 哒嗪环类化合物、其药物组合物及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR119731A1 (es) 2019-05-17 2022-01-05 Novartis Ag Inhibidores del inflamasoma nlrp3
CN115279739B (zh) * 2020-03-27 2025-07-22 尼科治疗有限公司 取代哒嗪化合物
EP4289823A4 (en) * 2021-02-08 2025-02-26 Medshine Discovery Inc. SUBSTITUTED PYRIDAZINE PHENOL DERIVATIVES

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