JP2024537619A5 - - Google Patents
Info
- Publication number
- JP2024537619A5 JP2024537619A5 JP2024514096A JP2024514096A JP2024537619A5 JP 2024537619 A5 JP2024537619 A5 JP 2024537619A5 JP 2024514096 A JP2024514096 A JP 2024514096A JP 2024514096 A JP2024514096 A JP 2024514096A JP 2024537619 A5 JP2024537619 A5 JP 2024537619A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- amino
- acid
- dimethyl
- dimethylhexanoic acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP21194937.5A EP4144352A1 (en) | 2021-09-03 | 2021-09-03 | 2-amino-5,5-dimethylhexanoic acid derivatives as sortilin modulators for use in the treatment of disease of the central nervous system |
| EP21194937.5 | 2021-09-03 | ||
| PCT/EP2022/074536 WO2023031440A1 (en) | 2021-09-03 | 2022-09-02 | 2-amino-5,5-dimethylhexanoic acid derivatives as sortilin modulators for use in the treatment of disease of the central nervous system |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024537619A JP2024537619A (ja) | 2024-10-16 |
| JP2024537619A5 true JP2024537619A5 (https=) | 2025-09-09 |
Family
ID=77640524
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024514096A Pending JP2024537619A (ja) | 2021-09-03 | 2022-09-02 | 中枢神経系の疾患の処置における使用のためのソルチリンモジュレーターとしての２－アミノ－５，５－ジメチルヘキサン酸誘導体 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20250268854A1 (https=) |
| EP (2) | EP4144352A1 (https=) |
| JP (1) | JP2024537619A (https=) |
| KR (1) | KR20240056551A (https=) |
| CN (1) | CN118019533A (https=) |
| AU (1) | AU2022339056A1 (https=) |
| CA (1) | CA3229686A1 (https=) |
| IL (1) | IL311208A (https=) |
| MX (1) | MX2024002696A (https=) |
| WO (1) | WO2023031440A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20250028349A (ko) | 2022-06-23 | 2025-02-28 | 드라우프니르 바이오 에이피에스 | 리소좀 내 세포외 표적의 분해를 선택적으로 유도하는 이작용성 분자 |
| EP4342530A1 (en) * | 2022-09-02 | 2024-03-27 | Insusense ApS | Sortilin modulators |
| EP4428122A1 (en) * | 2023-03-07 | 2024-09-11 | Vesper Bio Aps | Sortiline modulators |
| EP4719366A1 (en) | 2023-05-26 | 2026-04-08 | Bertram Wiedenmann | Sortilin inhibitors for treatment of patients with functional neuroendocrine tumors |
| WO2025178062A1 (en) * | 2024-02-20 | 2025-08-28 | Otsuka Pharmaceutical Co., Ltd. | Piperidine- and morpholine-carboxylate compounds as sort1 inhibitors |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2948147B1 (en) * | 2013-01-28 | 2019-03-13 | H. Lundbeck A/S | N-substituted-5-substituted phthalamic acids as sortilin inhibitors |
| US20160331746A1 (en) | 2015-05-12 | 2016-11-17 | University Of South Florida | Sortilin-Binding Small Molecules for Increasing Glucose Uptake |
| US20230044608A1 (en) | 2019-12-10 | 2023-02-09 | Aarhus Universitet | Compounds for treatment of eye diseases |
-
2021
- 2021-09-03 EP EP21194937.5A patent/EP4144352A1/en not_active Withdrawn
-
2022
- 2022-09-02 AU AU2022339056A patent/AU2022339056A1/en active Pending
- 2022-09-02 IL IL311208A patent/IL311208A/en unknown
- 2022-09-02 US US18/688,974 patent/US20250268854A1/en active Pending
- 2022-09-02 WO PCT/EP2022/074536 patent/WO2023031440A1/en not_active Ceased
- 2022-09-02 EP EP22773450.6A patent/EP4395776A1/en active Pending
- 2022-09-02 MX MX2024002696A patent/MX2024002696A/es unknown
- 2022-09-02 CA CA3229686A patent/CA3229686A1/en active Pending
- 2022-09-02 CN CN202280059105.7A patent/CN118019533A/zh active Pending
- 2022-09-02 KR KR1020247010428A patent/KR20240056551A/ko active Pending
- 2022-09-02 JP JP2024514096A patent/JP2024537619A/ja active Pending
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