JP2024522304A5 - - Google Patents

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Publication number
JP2024522304A5
JP2024522304A5 JP2024518956A JP2024518956A JP2024522304A5 JP 2024522304 A5 JP2024522304 A5 JP 2024522304A5 JP 2024518956 A JP2024518956 A JP 2024518956A JP 2024518956 A JP2024518956 A JP 2024518956A JP 2024522304 A5 JP2024522304 A5 JP 2024522304A5
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JP
Japan
Prior art keywords
cancer
alkyl
compound according
cancers
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024518956A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024522304A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/032203 external-priority patent/WO2022256680A1/en
Publication of JP2024522304A publication Critical patent/JP2024522304A/ja
Publication of JP2024522304A5 publication Critical patent/JP2024522304A5/ja
Pending legal-status Critical Current

Links

JP2024518956A 2021-06-04 2022-06-03 Wee1キナーゼ阻害剤として有用なピリドピリミジン誘導体 Pending JP2024522304A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163196744P 2021-06-04 2021-06-04
US63/196,744 2021-06-04
PCT/US2022/032203 WO2022256680A1 (en) 2021-06-04 2022-06-03 Pyridopyrimidine derivatives useful as wee1 kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2024522304A JP2024522304A (ja) 2024-06-13
JP2024522304A5 true JP2024522304A5 (enExample) 2025-06-10

Family

ID=82321319

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024518956A Pending JP2024522304A (ja) 2021-06-04 2022-06-03 Wee1キナーゼ阻害剤として有用なピリドピリミジン誘導体

Country Status (10)

Country Link
US (1) US20240254123A1 (enExample)
EP (1) EP4347592A1 (enExample)
JP (1) JP2024522304A (enExample)
KR (1) KR20240044409A (enExample)
CN (1) CN117794932A (enExample)
AU (2) AU2022287033B2 (enExample)
CA (1) CA3225152A1 (enExample)
IL (1) IL309037A (enExample)
MX (1) MX2023014466A (enExample)
WO (1) WO2022256680A1 (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3253688A1 (en) 2022-03-07 2023-09-14 Debiopharm International S.A. TREATMENT METHODS FOR SMALL CELL LUNG CANCER
WO2025056747A1 (en) 2023-09-14 2025-03-20 Debiopharm International S.A. Combination of a wee1 inhibitor and a pkmyt1 inhibitor
CN120189510A (zh) * 2023-12-21 2025-06-24 北京哲源科技有限责任公司 一种并环化合物的应用
TW202541810A (zh) 2023-12-22 2025-11-01 瑞士商德彪製藥國際公司 治療實體腫瘤之方法
WO2025186213A1 (en) 2024-03-04 2025-09-12 Debiopharm International S.A. Combination of a wee1 inhibitor and a topoisomerase 1 inhibitor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002250236A1 (en) 2001-03-02 2002-09-19 Medimmune, Inc. Cd2 antagonists for treatment of autoimmune or inflammatory disease
PE20080695A1 (es) * 2006-04-27 2008-06-28 Banyu Pharma Co Ltd Derivados de dihidropirazolopirimidinona como inhibidores de quinasa weel
MX2014010176A (es) * 2012-02-23 2014-11-10 Abbvie Inc Inhibidores de cinasas de piridopirimidinona.
GB201306610D0 (en) * 2013-04-11 2013-05-29 Almac Discovery Ltd Pharmaceutical compounds
GB201612095D0 (en) * 2016-07-12 2016-08-24 Almac Discovery Ltd Pharmaceutical compounds
MX2020001235A (es) * 2017-08-01 2020-07-20 Recurium Ip Holdings Llc Análogos de 1,2-dihidro-3h-pirazolo[3,4-d]pirimidin-3-ona.
GB201800378D0 (en) * 2018-01-10 2018-02-21 Almac Discovery Ltd Pharmaceutical compounds

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