JP2024521774A5 - - Google Patents

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Publication number
JP2024521774A5
JP2024521774A5 JP2023572737A JP2023572737A JP2024521774A5 JP 2024521774 A5 JP2024521774 A5 JP 2024521774A5 JP 2023572737 A JP2023572737 A JP 2023572737A JP 2023572737 A JP2023572737 A JP 2023572737A JP 2024521774 A5 JP2024521774 A5 JP 2024521774A5
Authority
JP
Japan
Application number
JP2023572737A
Other languages
Japanese (ja)
Other versions
JP2024521774A (ja
JPWO2022251292A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/030823 external-priority patent/WO2022251292A1/en
Publication of JP2024521774A publication Critical patent/JP2024521774A/ja
Publication of JP2024521774A5 publication Critical patent/JP2024521774A5/ja
Publication of JPWO2022251292A5 publication Critical patent/JPWO2022251292A5/ja
Pending legal-status Critical Current

Links

JP2023572737A 2021-05-25 2022-05-25 Rasの阻害方法 Pending JP2024521774A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163192837P 2021-05-25 2021-05-25
US63/192,837 2021-05-25
PCT/US2022/030823 WO2022251292A1 (en) 2021-05-25 2022-05-25 Methods for inhibiting ras

Publications (3)

Publication Number Publication Date
JP2024521774A JP2024521774A (ja) 2024-06-04
JP2024521774A5 true JP2024521774A5 (https=) 2025-06-02
JPWO2022251292A5 JPWO2022251292A5 (https=) 2025-06-02

Family

ID=82115695

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023572737A Pending JP2024521774A (ja) 2021-05-25 2022-05-25 Rasの阻害方法

Country Status (11)

Country Link
US (1) US20240277796A1 (https=)
EP (1) EP4346898A1 (https=)
JP (1) JP2024521774A (https=)
KR (1) KR20240026526A (https=)
CN (2) CN118557730A (https=)
AU (1) AU2022281343A1 (https=)
CA (1) CA3219533A1 (https=)
IL (1) IL308771A (https=)
MX (1) MX2023013912A (https=)
TW (1) TW202313631A (https=)
WO (1) WO2022251292A1 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2022005359A (es) 2019-11-04 2022-06-02 Revolution Medicines Inc Inhibidores de ras.
MX2023003060A (es) 2020-09-15 2023-04-05 Revolution Medicines Inc Derivados indolicos como inhibidores de ras en el tratamiento del cancer.
AU2022268962A1 (en) 2021-05-05 2023-12-14 Revolution Medicines, Inc. Ras inhibitors for the treatment of cancer
AR127308A1 (es) * 2021-10-08 2024-01-10 Revolution Medicines Inc Inhibidores ras
CN118922423A (zh) * 2022-01-10 2024-11-08 锐新医药公司 Ras抑制剂
CN119301132A (zh) * 2022-06-01 2025-01-10 豪夫迈·罗氏有限公司 用于治疗癌症的卤代吲哚大环化合物
CN119522225A (zh) 2022-09-29 2025-02-25 广州嘉越医药科技有限公司 大环衍生物及其应用
CR20250329A (es) 2023-02-14 2025-09-12 Hoffmann La Roche Compuestos tricíclicos para el tratamiento del cáncer
EP4687905A1 (en) * 2023-03-30 2026-02-11 Revolution Medicines, Inc. Compositions for inducing ras gtp hydrolysis and uses thereof
TW202446387A (zh) * 2023-04-06 2024-12-01 瑞士商赫孚孟拉羅股份公司 用於治療癌症之三環化合物
AU2024265078A1 (en) 2023-05-04 2025-12-11 Revolution Medicines, Inc. Combination therapy for a ras related disease or disorder
WO2025019318A2 (en) * 2023-07-14 2025-01-23 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2025162395A1 (zh) * 2024-02-01 2025-08-07 山东先声生物制药有限公司 吲哚衍生物作为ras抑制剂及其应用
CN119431325A (zh) * 2024-10-31 2025-02-14 诚达药业股份有限公司 一种3-(1h-吡唑-1-基)氮杂环丁烷类化合物及其合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20210116479A (ko) 2018-12-21 2021-09-27 레볼루션 메디슨즈, 인크. 공동 결합에 참여하는 화합물 및 그의 용도
DE102019122206B4 (de) 2019-08-19 2021-07-08 Webasto SE Dachmodul zur Bildung eines Fahrzeugdachs mit Umfeldsensor
MX2022005359A (es) 2019-11-04 2022-06-02 Revolution Medicines Inc Inhibidores de ras.
CN120699039A (zh) 2019-11-04 2025-09-26 锐新医药公司 Ras抑制剂
WO2021091956A1 (en) 2019-11-04 2021-05-14 Revolution Medicines, Inc. Ras inhibitors
MX2023003060A (es) 2020-09-15 2023-04-05 Revolution Medicines Inc Derivados indolicos como inhibidores de ras en el tratamiento del cancer.

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