JP2024521774A5 - - Google Patents

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Publication number
JP2024521774A5
JP2024521774A5 JP2023572737A JP2023572737A JP2024521774A5 JP 2024521774 A5 JP2024521774 A5 JP 2024521774A5 JP 2023572737 A JP2023572737 A JP 2023572737A JP 2023572737 A JP2023572737 A JP 2023572737A JP 2024521774 A5 JP2024521774 A5 JP 2024521774A5
Authority
JP
Japan
Prior art keywords
optionally substituted
membered
alkyl
hydrogen
bonded
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023572737A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024521774A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/030823 external-priority patent/WO2022251292A1/en
Publication of JP2024521774A publication Critical patent/JP2024521774A/ja
Publication of JP2024521774A5 publication Critical patent/JP2024521774A5/ja
Pending legal-status Critical Current

Links

JP2023572737A 2021-05-25 2022-05-25 Rasの阻害方法 Pending JP2024521774A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163192837P 2021-05-25 2021-05-25
US63/192,837 2021-05-25
PCT/US2022/030823 WO2022251292A1 (en) 2021-05-25 2022-05-25 Methods for inhibiting ras

Publications (2)

Publication Number Publication Date
JP2024521774A JP2024521774A (ja) 2024-06-04
JP2024521774A5 true JP2024521774A5 (https=) 2025-06-02

Family

ID=82115695

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023572737A Pending JP2024521774A (ja) 2021-05-25 2022-05-25 Rasの阻害方法

Country Status (11)

Country Link
US (1) US20240277796A1 (https=)
EP (1) EP4346898A1 (https=)
JP (1) JP2024521774A (https=)
KR (1) KR20240026526A (https=)
CN (2) CN118557730A (https=)
AU (1) AU2022281343A1 (https=)
CA (1) CA3219533A1 (https=)
IL (1) IL308771A (https=)
MX (1) MX2023013912A (https=)
TW (1) TW202313631A (https=)
WO (1) WO2022251292A1 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202132316A (zh) 2019-11-04 2021-09-01 美商銳新醫藥公司 Ras抑制劑
CA3194067A1 (en) 2020-09-15 2022-03-24 Revolution Medicines, Inc. Ras inhibitors
KR20240017811A (ko) 2021-05-05 2024-02-08 레볼루션 메디슨즈, 인크. 암의 치료를 위한 ras 억제제
AR127308A1 (es) 2021-10-08 2024-01-10 Revolution Medicines Inc Inhibidores ras
CN118922423A (zh) * 2022-01-10 2024-11-08 锐新医药公司 Ras抑制剂
JP2025519199A (ja) * 2022-06-01 2025-06-24 エフ・ホフマン-ラ・ロシュ・アクチェンゲゼルシャフト がんの治療のためのハロインドール大環状化合物
KR20250085767A (ko) 2022-09-29 2025-06-12 광조우 조요 파마테크 컴퍼니 리미티드 거대고리 유도체 및 이의 적용
CN120813588A (zh) 2023-02-14 2025-10-17 豪夫迈·罗氏有限公司 用于治疗癌症的三环化合物
AU2024241633A1 (en) * 2023-03-30 2025-11-06 Revolution Medicines, Inc. Compositions for inducing ras gtp hydrolysis and uses thereof
TW202446387A (zh) * 2023-04-06 2024-12-01 瑞士商赫孚孟拉羅股份公司 用於治療癌症之三環化合物
TW202508595A (zh) 2023-05-04 2025-03-01 美商銳新醫藥公司 用於ras相關疾病或病症之組合療法
US20250041295A1 (en) * 2023-07-14 2025-02-06 Revolution Medicines, Inc. Methods of treating a ras related disease or disorder
WO2025162395A1 (zh) * 2024-02-01 2025-08-07 山东先声生物制药有限公司 吲哚衍生物作为ras抑制剂及其应用
CN119431325A (zh) * 2024-10-31 2025-02-14 诚达药业股份有限公司 一种3-(1h-吡唑-1-基)氮杂环丁烷类化合物及其合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021012057A2 (pt) 2018-12-21 2021-10-19 Revolution Medicines, Inc. Compostos que participam de ligação cooperativa e usos dos mesmos
DE102019122206B4 (de) 2019-08-19 2021-07-08 Webasto SE Dachmodul zur Bildung eines Fahrzeugdachs mit Umfeldsensor
TW202132316A (zh) 2019-11-04 2021-09-01 美商銳新醫藥公司 Ras抑制劑
IL322454A (en) 2019-11-04 2025-09-01 Revolution Medicines Inc ras inhibitors
AU2020377925A1 (en) 2019-11-04 2022-05-05 Revolution Medicines, Inc. Ras inhibitors
CA3194067A1 (en) 2020-09-15 2022-03-24 Revolution Medicines, Inc. Ras inhibitors

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