JP2024516795A5 - - Google Patents

Info

Publication number
JP2024516795A5
JP2024516795A5 JP2023562510A JP2023562510A JP2024516795A5 JP 2024516795 A5 JP2024516795 A5 JP 2024516795A5 JP 2023562510 A JP2023562510 A JP 2023562510A JP 2023562510 A JP2023562510 A JP 2023562510A JP 2024516795 A5 JP2024516795 A5 JP 2024516795A5
Authority
JP
Japan
Prior art keywords
cancer
pharmaceutically acceptable
everolimus
amsenestrant
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023562510A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024516795A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2022/059704 external-priority patent/WO2022218958A1/en
Publication of JP2024516795A publication Critical patent/JP2024516795A/ja
Publication of JP2024516795A5 publication Critical patent/JP2024516795A5/ja
Pending legal-status Critical Current

Links

JP2023562510A 2021-04-12 2022-04-12 エベロリムスおよびアムセネストラントを含む組合せ物 Pending JP2024516795A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP21315063.4 2021-04-12
EP21315063 2021-04-12
PCT/EP2022/059704 WO2022218958A1 (en) 2021-04-12 2022-04-12 Combination comprising everolimus and amcenestrant

Publications (2)

Publication Number Publication Date
JP2024516795A JP2024516795A (ja) 2024-04-17
JP2024516795A5 true JP2024516795A5 (https=) 2025-04-16

Family

ID=75825773

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023562510A Pending JP2024516795A (ja) 2021-04-12 2022-04-12 エベロリムスおよびアムセネストラントを含む組合せ物

Country Status (8)

Country Link
US (1) US20240197692A1 (https=)
EP (1) EP4322942B1 (https=)
JP (1) JP2024516795A (https=)
CN (1) CN117177743A (https=)
AR (1) AR125330A1 (https=)
ES (1) ES3036485T3 (https=)
TW (1) TW202304424A (https=)
WO (1) WO2022218958A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112021003440A2 (pt) 2018-09-07 2021-05-18 Sanofi sais de 6-(2,4-diclorofenil)-5-[4-[(3s)-1-(3-fluoropropil) pirrolidin-3-il]oxifenil]-8,9-di-hidro-7h-benzo[7]anuleno-2-carboxilato de metila e seu processo de preparação
EP4037768B1 (en) 2019-10-01 2023-10-11 Sanofi Novel substituted 6,7-dihydro-5h-benzo[7]annulene compounds, processes for their preparation and therapeutic uses thereof
AU2020399168A1 (en) 2019-12-09 2022-07-28 Sanofi Crystalline form of a 7H-benzo[7]annulene-2-carboxylic acid derivative
TW202146007A (zh) 2020-02-27 2021-12-16 法商賽諾菲公司 包含阿培利司(alpelisib)與6-(2,4-二氯苯基)-5-[4-[(3s)-1-(3-氟丙基)吡咯啶-3-基]氧苯基]-8,9-二氫-7h-苯并[7]輪烯-2-羧酸之組合
TW202233572A (zh) 2020-10-19 2022-09-01 法商賽諾菲公司 新穎之經取代的6,7-二氫-5h-苯並[7]輪烯衍生物,其製備方法及其治療用途
WO2022084280A1 (en) 2020-10-19 2022-04-28 Sanofi Substituted 6,7-dihydro-5h-benzo[7]annulene compounds and their derivatives, processes for their preparation and therapeutic uses thereof
TW202543650A (zh) 2024-03-08 2025-11-16 美商海爾達醫療運營公司 異雙官能化合物及其在治療疾病中之用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105828822B (zh) * 2013-08-14 2019-10-18 诺华股份有限公司 用于治疗癌症的组合疗法
EA034994B1 (ru) 2016-02-15 2020-04-15 Санофи 6,7-дигидро-5h-бензо[7]аннуленовые производные в качестве модуляторов эстрогеновых рецепторов
CA3169679A1 (en) * 2020-03-06 2021-09-10 Olema Pharmaceuticals, Inc. Methods of treating estrogen receptor-associated diseases

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