JP2024516199A5 - - Google Patents
Info
- Publication number
- JP2024516199A5 JP2024516199A5 JP2023565369A JP2023565369A JP2024516199A5 JP 2024516199 A5 JP2024516199 A5 JP 2024516199A5 JP 2023565369 A JP2023565369 A JP 2023565369A JP 2023565369 A JP2023565369 A JP 2023565369A JP 2024516199 A5 JP2024516199 A5 JP 2024516199A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- reacting
- hcl
- item
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163180043P | 2021-04-26 | 2021-04-26 | |
| US63/180,043 | 2021-04-26 | ||
| US202163286764P | 2021-12-07 | 2021-12-07 | |
| US63/286,764 | 2021-12-07 | ||
| PCT/US2022/026208 WO2022232060A1 (en) | 2021-04-26 | 2022-04-25 | Processes for the synthesis of valbenazine |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024516199A JP2024516199A (ja) | 2024-04-12 |
| JP2024516199A5 true JP2024516199A5 (https=) | 2025-05-08 |
Family
ID=81654703
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023565369A Pending JP2024516199A (ja) | 2021-04-26 | 2022-04-25 | バルベナジンの合成方法 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20240239791A1 (https=) |
| EP (1) | EP4330255A1 (https=) |
| JP (1) | JP2024516199A (https=) |
| CA (1) | CA3215792A1 (https=) |
| IL (1) | IL307826A (https=) |
| WO (1) | WO2022232060A1 (https=) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2026050236A1 (en) | 2024-08-27 | 2026-03-05 | Neurocrine Biosciences, Inc. | Muscarinic receptor agonist in combination with a vesicular monoamine transporter 2 inhibitor, for use in the treatment of a neurological or psychiatric disorder |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2081929B1 (en) | 2006-11-08 | 2013-01-09 | Neurocrine Biosciences, Inc. | Substituted 3-isobutyl-9, 10-dimethoxy-1,3,4,6,7,11b-hexahydro-2h-pyrido[2,1-a]isoquinolin-2-ol compounds and methods relating thereto |
| RS61645B1 (sr) | 2015-10-30 | 2021-04-29 | Neurocrine Biosciences Inc | Valbenazin ditozilat i njihovi polimorfi |
| JP6869988B2 (ja) * | 2015-12-23 | 2021-05-12 | ニューロクライン バイオサイエンシーズ,インコーポレイテッド | (S)−(2R,3R,11bR)−3−イソブチル−9,10−ジメトキシ−2,3,4,6,7,11b−ヘキサヒドロ−1H−ピリド[2,1−a]イソキノリン−2−イル2−アミノ−3−メチルブタノエートジ(4−メチルベンゼンスルホネート)の調製のための合成方法 |
| CA3076000A1 (en) | 2017-09-21 | 2019-03-28 | Neurocrine Biosciences, Inc. | High dosage valbenazine formulation and compositions, methods, and kits related thereto |
| CA3150961A1 (en) * | 2019-09-13 | 2021-03-18 | John Tucker | Processes for the synthesis of valbenazine |
-
2022
- 2022-04-25 EP EP22723872.2A patent/EP4330255A1/en not_active Withdrawn
- 2022-04-25 WO PCT/US2022/026208 patent/WO2022232060A1/en not_active Ceased
- 2022-04-25 US US18/288,311 patent/US20240239791A1/en active Pending
- 2022-04-25 IL IL307826A patent/IL307826A/en unknown
- 2022-04-25 JP JP2023565369A patent/JP2024516199A/ja active Pending
- 2022-04-25 CA CA3215792A patent/CA3215792A1/en active Pending
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