JP2024511832A5 - - Google Patents

Info

Publication number
JP2024511832A5
JP2024511832A5 JP2023560282A JP2023560282A JP2024511832A5 JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5 JP 2023560282 A JP2023560282 A JP 2023560282A JP 2023560282 A JP2023560282 A JP 2023560282A JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5
Authority
JP
Japan
Prior art keywords
alkyl
membered
deuterium
independently selected
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023560282A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024511832A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2022/083557 external-priority patent/WO2022206725A1/en
Publication of JP2024511832A publication Critical patent/JP2024511832A/ja
Publication of JP2024511832A5 publication Critical patent/JP2024511832A5/ja
Pending legal-status Critical Current

Links

JP2023560282A 2021-03-30 2022-03-29 Stingアゴニストとして有用な新規化合物およびその使用 Pending JP2024511832A (ja)

Applications Claiming Priority (17)

Application Number Priority Date Filing Date Title
CNPCT/CN2021/083783 2021-03-30
CN2021083783 2021-03-30
CN2021090945 2021-04-29
CNPCT/CN2021/090945 2021-04-29
CN2021111479 2021-08-09
CNPCT/CN2021/111479 2021-08-09
CNPCT/CN2021/128942 2021-11-05
CN2021128942 2021-11-05
CN2021130097 2021-11-11
CNPCT/CN2021/130097 2021-11-11
CNPCT/CN2021/138806 2021-12-16
CN2021138806 2021-12-16
CN2021143043 2021-12-30
CNPCT/CN2021/143043 2021-12-30
CN2022071548 2022-01-12
CNPCT/CN2022/071548 2022-01-12
PCT/CN2022/083557 WO2022206725A1 (en) 2021-03-30 2022-03-29 Novel compounds useful as sting agonists and uses thereof

Publications (2)

Publication Number Publication Date
JP2024511832A JP2024511832A (ja) 2024-03-15
JP2024511832A5 true JP2024511832A5 (cg-RX-API-DMAC10.html) 2025-04-07

Family

ID=83457956

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023560282A Pending JP2024511832A (ja) 2021-03-30 2022-03-29 Stingアゴニストとして有用な新規化合物およびその使用

Country Status (8)

Country Link
US (1) US20240116909A1 (cg-RX-API-DMAC10.html)
EP (1) EP4313962B1 (cg-RX-API-DMAC10.html)
JP (1) JP2024511832A (cg-RX-API-DMAC10.html)
CN (1) CN117203194A (cg-RX-API-DMAC10.html)
AR (1) AR125608A1 (cg-RX-API-DMAC10.html)
TW (1) TW202302579A (cg-RX-API-DMAC10.html)
UY (1) UY39705A (cg-RX-API-DMAC10.html)
WO (1) WO2022206725A1 (cg-RX-API-DMAC10.html)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20250108123A1 (en) * 2021-12-17 2025-04-03 Jacobio Pharmaceuticals Co., Ltd. Compound-linker constructs comprising novel compounds useful as sting agonists and uses thereof
WO2024032782A1 (en) * 2022-08-12 2024-02-15 Jacobio Pharmaceuticals Co.Ltd. Vaccine adjuvants and uses thereof
TW202615010A (zh) * 2024-06-24 2026-04-16 大陸商北京加科思新藥研發有限公司 藥物連接子、其偶聯物及其用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10793557B2 (en) 2018-04-03 2020-10-06 Merck Sharp & Dohme Corp. Sting agonist compounds
US11702430B2 (en) * 2018-04-03 2023-07-18 Merck Sharp & Dohme Llc Aza-benzothiophene compounds as STING agonists
DK4004002T3 (da) * 2019-07-22 2024-09-30 Lupin Ltd Makrocykliske forbindelser som sting-agonister samt fremgangsmåder og anvendelser dermed

Similar Documents

Publication Publication Date Title
CN114174303B (zh) 作为sting激动剂的大环化合物及其方法和用途
JP2024522990A5 (cg-RX-API-DMAC10.html)
JP2024512154A5 (cg-RX-API-DMAC10.html)
EA031030B1 (ru) Ингибиторы фактора в комплемента на основе производных пиперидинилиндола и их применение
JP2006528700A5 (cg-RX-API-DMAC10.html)
JP2013510883A5 (cg-RX-API-DMAC10.html)
JP2019500387A5 (cg-RX-API-DMAC10.html)
RU2014122340A (ru) Ингибиторы вируса гепатита с, имеющие жесткую вытянутую цепь и содержащие фрагмент {2-[4-(бифенил-4-ил)-1н-имидазо-2-ил]пирролидин-1-карбонилметил}амина
RU2014153800A (ru) Соединения 5-азаиндазола и способы их применения
JP2014528467A5 (cg-RX-API-DMAC10.html)
JP2013544812A5 (cg-RX-API-DMAC10.html)
RU2012117398A (ru) Бензоксазепиновые ингибиторы pi3 и способы применения
RU2009148320A (ru) Производные пиперидина/пиперазина
JP2015501833A5 (cg-RX-API-DMAC10.html)
JP2013520473A5 (cg-RX-API-DMAC10.html)
RU2018134780A (ru) Новые соединения и их фармацевтические композиции для лечения фиброза
JP2014532716A5 (cg-RX-API-DMAC10.html)
JP2008526999A5 (cg-RX-API-DMAC10.html)
RU2010101611A (ru) Полициклические производные гуанина и способы их применения
JP2024517861A5 (cg-RX-API-DMAC10.html)
RU2009135389A (ru) Четвертичные аммониевые дифенилметилсоединения, применимые в качестве антагонистов мускариновых рецепторов
RU2009103041A (ru) Селективные антагонисты аденозиновых а2а рецепторов
CA2626032A1 (en) Camptothecin derivatives as chemoradiosensitizing agents
JP2024535913A5 (cg-RX-API-DMAC10.html)
JP2024543016A5 (cg-RX-API-DMAC10.html)