JP2024511832A5 - - Google Patents
Info
- Publication number
- JP2024511832A5 JP2024511832A5 JP2023560282A JP2023560282A JP2024511832A5 JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5 JP 2023560282 A JP2023560282 A JP 2023560282A JP 2023560282 A JP2023560282 A JP 2023560282A JP 2024511832 A5 JP2024511832 A5 JP 2024511832A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- membered
- deuterium
- independently selected
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2021/083783 | 2021-03-30 | ||
| CN2021083783 | 2021-03-30 | ||
| CN2021090945 | 2021-04-29 | ||
| CNPCT/CN2021/090945 | 2021-04-29 | ||
| CN2021111479 | 2021-08-09 | ||
| CNPCT/CN2021/111479 | 2021-08-09 | ||
| CNPCT/CN2021/128942 | 2021-11-05 | ||
| CN2021128942 | 2021-11-05 | ||
| CN2021130097 | 2021-11-11 | ||
| CNPCT/CN2021/130097 | 2021-11-11 | ||
| CNPCT/CN2021/138806 | 2021-12-16 | ||
| CN2021138806 | 2021-12-16 | ||
| CN2021143043 | 2021-12-30 | ||
| CNPCT/CN2021/143043 | 2021-12-30 | ||
| CN2022071548 | 2022-01-12 | ||
| CNPCT/CN2022/071548 | 2022-01-12 | ||
| PCT/CN2022/083557 WO2022206725A1 (en) | 2021-03-30 | 2022-03-29 | Novel compounds useful as sting agonists and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024511832A JP2024511832A (ja) | 2024-03-15 |
| JP2024511832A5 true JP2024511832A5 (cg-RX-API-DMAC10.html) | 2025-04-07 |
Family
ID=83457956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023560282A Pending JP2024511832A (ja) | 2021-03-30 | 2022-03-29 | Stingアゴニストとして有用な新規化合物およびその使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20240116909A1 (cg-RX-API-DMAC10.html) |
| EP (1) | EP4313962B1 (cg-RX-API-DMAC10.html) |
| JP (1) | JP2024511832A (cg-RX-API-DMAC10.html) |
| CN (1) | CN117203194A (cg-RX-API-DMAC10.html) |
| AR (1) | AR125608A1 (cg-RX-API-DMAC10.html) |
| TW (1) | TW202302579A (cg-RX-API-DMAC10.html) |
| UY (1) | UY39705A (cg-RX-API-DMAC10.html) |
| WO (1) | WO2022206725A1 (cg-RX-API-DMAC10.html) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20250108123A1 (en) * | 2021-12-17 | 2025-04-03 | Jacobio Pharmaceuticals Co., Ltd. | Compound-linker constructs comprising novel compounds useful as sting agonists and uses thereof |
| WO2024032782A1 (en) * | 2022-08-12 | 2024-02-15 | Jacobio Pharmaceuticals Co.Ltd. | Vaccine adjuvants and uses thereof |
| TW202615010A (zh) * | 2024-06-24 | 2026-04-16 | 大陸商北京加科思新藥研發有限公司 | 藥物連接子、其偶聯物及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10793557B2 (en) | 2018-04-03 | 2020-10-06 | Merck Sharp & Dohme Corp. | Sting agonist compounds |
| US11702430B2 (en) * | 2018-04-03 | 2023-07-18 | Merck Sharp & Dohme Llc | Aza-benzothiophene compounds as STING agonists |
| DK4004002T3 (da) * | 2019-07-22 | 2024-09-30 | Lupin Ltd | Makrocykliske forbindelser som sting-agonister samt fremgangsmåder og anvendelser dermed |
-
2022
- 2022-03-29 US US18/284,897 patent/US20240116909A1/en active Pending
- 2022-03-29 EP EP22778907.0A patent/EP4313962B1/en active Active
- 2022-03-29 UY UY0001039705A patent/UY39705A/es unknown
- 2022-03-29 CN CN202280023908.7A patent/CN117203194A/zh active Pending
- 2022-03-29 TW TW111112050A patent/TW202302579A/zh unknown
- 2022-03-29 WO PCT/CN2022/083557 patent/WO2022206725A1/en not_active Ceased
- 2022-03-29 JP JP2023560282A patent/JP2024511832A/ja active Pending
- 2022-03-29 AR ARP220100748A patent/AR125608A1/es not_active Application Discontinuation
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