JP2024510939A5 - - Google Patents

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Publication number
JP2024510939A5
JP2024510939A5 JP2023553301A JP2023553301A JP2024510939A5 JP 2024510939 A5 JP2024510939 A5 JP 2024510939A5 JP 2023553301 A JP2023553301 A JP 2023553301A JP 2023553301 A JP2023553301 A JP 2023553301A JP 2024510939 A5 JP2024510939 A5 JP 2024510939A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
alkyl
compound according
regulation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023553301A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024510939A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/018321 external-priority patent/WO2022187231A1/en
Publication of JP2024510939A publication Critical patent/JP2024510939A/ja
Publication of JP2024510939A5 publication Critical patent/JP2024510939A5/ja
Pending legal-status Critical Current

Links

JP2023553301A 2021-03-03 2022-03-01 オレキシン受容体アゴニストとしてのアリールスルホンアミド Pending JP2024510939A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163156164P 2021-03-03 2021-03-03
US63/156,164 2021-03-03
PCT/US2022/018321 WO2022187231A1 (en) 2021-03-03 2022-03-01 Arylsulfoxamides as orexin receptor agonists

Publications (2)

Publication Number Publication Date
JP2024510939A JP2024510939A (ja) 2024-03-12
JP2024510939A5 true JP2024510939A5 (https=) 2025-03-10

Family

ID=83154799

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023553301A Pending JP2024510939A (ja) 2021-03-03 2022-03-01 オレキシン受容体アゴニストとしてのアリールスルホンアミド

Country Status (8)

Country Link
US (1) US20240174605A1 (https=)
EP (1) EP4301728A4 (https=)
JP (1) JP2024510939A (https=)
CN (1) CN117015526B (https=)
AU (1) AU2022229350A1 (https=)
CA (1) CA3208567A1 (https=)
MX (1) MX2023009452A (https=)
WO (1) WO2022187231A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI4065585T3 (fi) 2019-11-25 2025-09-26 Alkermes Inc Substituoituja makrosyklisiä yhdisteitä ja niihin liittyviä hoitomenetelmiä
US11760747B2 (en) 2020-12-21 2023-09-19 Alkermes, Inc. Substituted piperidino compounds and related methods of treatment
US12006330B2 (en) 2020-12-21 2024-06-11 Alkermes, Inc. Substituted macrocyclic compounds and related methods of treatment
WO2025124698A1 (en) 2023-12-12 2025-06-19 Idorsia Pharmaceuticals Ltd Aryl sulfone and sulfanone derivatives as orexin receptor modulators
TW202542165A (zh) 2023-12-19 2025-11-01 瑞士商愛杜西亞製藥有限公司 大環食慾素激動劑

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8258163B2 (en) 2008-06-04 2012-09-04 Board Of Regents, The University Of Texas System Small-molecule agonists for type-2 orexin receptor
PE20161064A1 (es) * 2013-12-12 2016-10-28 Univ Tsukuba Derivado de sulfonamida o sales de adicion de acido farmaceuticamente aceptables del mismo
WO2016133160A1 (ja) * 2015-02-19 2016-08-25 国立大学法人筑波大学 スルホンアミド誘導体またはその薬学的に許容される酸付加塩
WO2016199906A1 (ja) * 2015-06-12 2016-12-15 国立大学法人筑波大学 スルホンアミド誘導体またはその薬学的に許容される酸付加塩
WO2019117148A1 (ja) * 2017-12-12 2019-06-20 国立大学法人 筑波大学 スルホンアミド誘導体またはその薬学的に許容される酸付加塩
MX2020010155A (es) * 2018-03-27 2021-03-25 Univ Texas Compuestos de ox2r.
US11098029B2 (en) 2019-02-13 2021-08-24 Merck Sharp & Dohme Corp. 5-alkyl pyrrolidine orexin receptor agonists

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