JP2024506116A5 - - Google Patents

Info

Publication number
JP2024506116A5
JP2024506116A5 JP2023531615A JP2023531615A JP2024506116A5 JP 2024506116 A5 JP2024506116 A5 JP 2024506116A5 JP 2023531615 A JP2023531615 A JP 2023531615A JP 2023531615 A JP2023531615 A JP 2023531615A JP 2024506116 A5 JP2024506116 A5 JP 2024506116A5
Authority
JP
Japan
Prior art keywords
optionally substituted
pharmaceutically acceptable
acceptable salt
cancer
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023531615A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024506116A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2021/133429 external-priority patent/WO2022111621A1/en
Publication of JP2024506116A publication Critical patent/JP2024506116A/ja
Publication of JP2024506116A5 publication Critical patent/JP2024506116A5/ja
Pending legal-status Critical Current

Links

JP2023531615A 2020-11-27 2021-11-26 アミノヘテロアリールキナーゼ阻害剤 Pending JP2024506116A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CN2020132454 2020-11-27
CNPCT/CN2020/132454 2020-11-27
CNPCT/CN2021/081236 2021-03-17
CN2021081236 2021-03-17
PCT/CN2021/133429 WO2022111621A1 (en) 2020-11-27 2021-11-26 Aminoheteroaryl kinase inhibitors

Publications (2)

Publication Number Publication Date
JP2024506116A JP2024506116A (ja) 2024-02-09
JP2024506116A5 true JP2024506116A5 (https=) 2024-12-04

Family

ID=81753779

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2023531615A Pending JP2024506116A (ja) 2020-11-27 2021-11-26 アミノヘテロアリールキナーゼ阻害剤
JP2024531423A Pending JP2024541533A (ja) 2020-11-27 2022-11-23 アミノヘテロアリールキナーゼ阻害薬

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2024531423A Pending JP2024541533A (ja) 2020-11-27 2022-11-23 アミノヘテロアリールキナーゼ阻害薬

Country Status (10)

Country Link
US (2) US20240166635A1 (https=)
EP (2) EP4251613A4 (https=)
JP (2) JP2024506116A (https=)
KR (1) KR20230127228A (https=)
CN (2) CN116528869B (https=)
AU (3) AU2021385745C1 (https=)
CA (2) CA3202990A1 (https=)
IL (1) IL303237A (https=)
MX (1) MX2024006300A (https=)
WO (2) WO2022111621A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4251613A4 (en) * 2020-11-27 2024-11-20 Allorion Therapeutics Inc. AMINOHETEROARYL KINASE INHIBITORS
CA3207392A1 (en) * 2021-02-05 2022-08-11 Xiaoxia Yan Cdk inhibitor
EP4532473A1 (en) * 2022-05-27 2025-04-09 Allorion Therapeutics Inc. Aminoheteroaryl kinase inhibitors
WO2025006400A1 (en) * 2023-06-25 2025-01-02 Allorion Therapeutics Inc Isotopologues of aminoheteroaryl kinase inhibitors and uses thereof
WO2026024674A1 (en) 2024-07-22 2026-01-29 Genesis Therapeutics, Inc. Methods of treating skp2-associated cancers
EP4725942A1 (en) * 2024-10-09 2026-04-15 Sibylla Biotech S.p.A. Compounds active on cyclin d1 pathway and their use

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GB0016877D0 (en) * 2000-07-11 2000-08-30 Astrazeneca Ab Chemical compounds
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BR0116452A (pt) * 2000-12-21 2003-09-30 Glaxo Group Ltd Composto, composição farmacêutica, uso de um composto
BR0209774A (pt) * 2001-05-29 2004-06-01 Schering Ag Pirimidinas inibidoras de cdk, sua preparação e aplicação como medicamento
GB0113041D0 (en) * 2001-05-30 2001-07-18 Astrazeneca Ab Chemical compounds
IL161663A0 (en) * 2001-11-01 2004-09-27 Janssen Pharmaceutica Nv AMINOBENZAMIDE DERIVATIVES AS GLYCOGEN SYNTHASE KINASE 3beta INHIBITORS
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EP1483260A1 (de) * 2002-03-11 2004-12-08 Schering Aktiengesellschaft Cdk inhibitorische 2-heteroaryl-pyrimidine, deren herstellung und verwendung als arzneimittel
JP2006508997A (ja) * 2002-11-28 2006-03-16 シエーリング アクチエンゲゼルシャフト Chk−、Pdk−およびAkt−阻害性ピリミジン、それらの製造および薬剤としての使用
US7504396B2 (en) * 2003-06-24 2009-03-17 Amgen Inc. Substituted heterocyclic compounds and methods of use
DE102005008310A1 (de) * 2005-02-17 2006-08-24 Schering Ag Verwendung von CDKII Inhibitoren zur Fertilitätskontrolle
AU2006244195B2 (en) * 2005-05-05 2012-03-15 Ardea Biosciences, Inc. Diaryl-purine, azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitors for treatment of HIV
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CA3207392A1 (en) * 2021-02-05 2022-08-11 Xiaoxia Yan Cdk inhibitor

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