JP2024502231A5 - - Google Patents

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Publication number
JP2024502231A5
JP2024502231A5 JP2023536951A JP2023536951A JP2024502231A5 JP 2024502231 A5 JP2024502231 A5 JP 2024502231A5 JP 2023536951 A JP2023536951 A JP 2023536951A JP 2023536951 A JP2023536951 A JP 2023536951A JP 2024502231 A5 JP2024502231 A5 JP 2024502231A5
Authority
JP
Japan
Prior art keywords
pain
compound according
pharmaceutical composition
hydrogen atom
alkyl group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP2023536951A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024502231A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2021/086101 external-priority patent/WO2022129283A1/en
Publication of JP2024502231A publication Critical patent/JP2024502231A/ja
Publication of JP2024502231A5 publication Critical patent/JP2024502231A5/ja
Ceased legal-status Critical Current

Links

JP2023536951A 2020-12-18 2021-12-16 Nav1.8電位依存性ナトリウムチャネルを阻害するためおよびNav1.8介在疾患を治療するために有用な化学化合物 Ceased JP2024502231A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063127341P 2020-12-18 2020-12-18
US63/127,341 2020-12-18
PCT/EP2021/086101 WO2022129283A1 (en) 2020-12-18 2021-12-16 Chemical compounds useful for inhibiting nav1.8 voltage-gated sodium channels and treating nav1.8 mediated diseases

Publications (2)

Publication Number Publication Date
JP2024502231A JP2024502231A (ja) 2024-01-18
JP2024502231A5 true JP2024502231A5 (https=) 2024-12-20

Family

ID=79025144

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023536951A Ceased JP2024502231A (ja) 2020-12-18 2021-12-16 Nav1.8電位依存性ナトリウムチャネルを阻害するためおよびNav1.8介在疾患を治療するために有用な化学化合物

Country Status (13)

Country Link
EP (1) EP4262978A1 (https=)
JP (1) JP2024502231A (https=)
KR (1) KR20230121827A (https=)
CN (1) CN116710463A (https=)
AU (1) AU2021403606B2 (https=)
CA (1) CA3202328A1 (https=)
CL (1) CL2023001750A1 (https=)
CO (1) CO2023008049A2 (https=)
IL (1) IL303795A (https=)
MX (1) MX2023007244A (https=)
PH (1) PH12023551406A1 (https=)
SA (1) SA523441263B1 (https=)
WO (1) WO2022129283A1 (https=)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2931550C (en) * 2013-12-13 2023-09-26 Vertex Pharmaceuticals Incorporated Prodrugs of pyridone amides useful as modulators of sodium channels
GB201322602D0 (en) * 2013-12-19 2014-02-05 Almac Discovery Ltd Pharmaceutical compounds
EP3625214B1 (en) * 2017-05-16 2022-07-06 Vertex Pharmaceuticals Incorporated Deuterated pyridone amides and prodrugs thereof as modulators of sodium channels
MX2021015605A (es) * 2019-06-27 2022-02-16 Glaxosmithkline Ip Dev Ltd Compuestos 2,3-dihidroquinazolin como inhibidores nav1.8.

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