JP2024500377A5 - - Google Patents

Info

Publication number
JP2024500377A5
JP2024500377A5 JP2023535990A JP2023535990A JP2024500377A5 JP 2024500377 A5 JP2024500377 A5 JP 2024500377A5 JP 2023535990 A JP2023535990 A JP 2023535990A JP 2023535990 A JP2023535990 A JP 2023535990A JP 2024500377 A5 JP2024500377 A5 JP 2024500377A5
Authority
JP
Japan
Prior art keywords
mixture
ethoxy
compound according
tautomers
methoxyphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023535990A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024500377A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/062995 external-priority patent/WO2022132603A1/en
Publication of JP2024500377A publication Critical patent/JP2024500377A/ja
Publication of JP2024500377A5 publication Critical patent/JP2024500377A5/ja
Pending legal-status Critical Current

Links

JP2023535990A 2020-12-14 2021-12-13 Pde4分解剤、医薬組成物、及び治療的応用 Pending JP2024500377A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063124877P 2020-12-14 2020-12-14
US63/124,877 2020-12-14
PCT/US2021/062995 WO2022132603A1 (en) 2020-12-14 2021-12-13 Pde4 degraders, pharmaceutical compositions, and therapeutic applications

Publications (2)

Publication Number Publication Date
JP2024500377A JP2024500377A (ja) 2024-01-09
JP2024500377A5 true JP2024500377A5 (https=) 2024-12-20

Family

ID=79288082

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023535990A Pending JP2024500377A (ja) 2020-12-14 2021-12-13 Pde4分解剤、医薬組成物、及び治療的応用

Country Status (10)

Country Link
US (1) US20240124418A1 (https=)
EP (1) EP4259621A1 (https=)
JP (1) JP2024500377A (https=)
KR (1) KR20230157936A (https=)
CN (1) CN117203196A (https=)
AU (1) AU2021402911A1 (https=)
CA (1) CA3201965A1 (https=)
IL (1) IL303611A (https=)
TW (1) TW202237580A (https=)
WO (1) WO2022132603A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021119571A1 (en) * 2019-12-12 2021-06-17 Biotheryx, Inc. Pde4 inhibitors, pharmaceutical compositions, and therapeutic applications
WO2024168096A2 (en) * 2023-02-07 2024-08-15 Biotheryx, Inc. Pde4 degraders, pharmaceutical compositions, and therapeutic applications
US20240327381A1 (en) * 2023-02-08 2024-10-03 Celgene Corporation Compounds and Compositions for Selective Degradation of Engineered Proteins
AU2024323358A1 (en) * 2023-08-17 2026-02-26 Katalytic Therapeutics, Inc. Pde4 protein degraders, pharmaceutical compositions, and therapeutic applications

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JP2022533260A (ja) 2019-05-24 2022-07-21 バイオセリックス, インコーポレイテッド タンパク質を標的とする化合物及びその医薬組成物並びにそれらの治療的応用
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