JP2024103495A5 - - Google Patents

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Publication number
JP2024103495A5
JP2024103495A5 JP2024074818A JP2024074818A JP2024103495A5 JP 2024103495 A5 JP2024103495 A5 JP 2024103495A5 JP 2024074818 A JP2024074818 A JP 2024074818A JP 2024074818 A JP2024074818 A JP 2024074818A JP 2024103495 A5 JP2024103495 A5 JP 2024103495A5
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Japan
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crystal
measured
ray powder
powder diffraction
composition
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JP2024074818A
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English (en)
Japanese (ja)
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JP2024103495A (ja
JP7842805B2 (ja
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Priority claimed from PCT/US2016/065799 external-priority patent/WO2017100553A1/en
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JP2024074818A 2015-12-10 2024-05-02 フマギロール誘導体およびその多形体 Active JP7842805B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201562265675P 2015-12-10 2015-12-10
US62/265,675 2015-12-10
PCT/US2016/065799 WO2017100553A1 (en) 2015-12-10 2016-12-09 Fumagillol derivatives and polymorphs thereof
JP2018529646A JP7553224B2 (ja) 2015-12-10 2016-12-09 フマギロール誘導体およびその多形体

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2018529646A Division JP7553224B2 (ja) 2015-12-10 2016-12-09 フマギロール誘導体およびその多形体

Publications (3)

Publication Number Publication Date
JP2024103495A JP2024103495A (ja) 2024-08-01
JP2024103495A5 true JP2024103495A5 (https=) 2024-11-25
JP7842805B2 JP7842805B2 (ja) 2026-04-08

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ID=57589276

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JP2018529646A Active JP7553224B2 (ja) 2015-12-10 2016-12-09 フマギロール誘導体およびその多形体
JP2024074818A Active JP7842805B2 (ja) 2015-12-10 2024-05-02 フマギロール誘導体およびその多形体

Family Applications Before (1)

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JP2018529646A Active JP7553224B2 (ja) 2015-12-10 2016-12-09 フマギロール誘導体およびその多形体

Country Status (11)

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US (2) US9969722B2 (https=)
EP (1) EP3386956B1 (https=)
JP (2) JP7553224B2 (https=)
KR (2) KR102849342B1 (https=)
CN (1) CN108290853B (https=)
AU (1) AU2016366306B2 (https=)
CA (1) CA3005450A1 (https=)
DK (1) DK3386956T3 (https=)
ES (1) ES2893749T3 (https=)
MX (2) MX2018006904A (https=)
WO (1) WO2017100553A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2576638T3 (da) 2010-05-25 2021-03-15 Syndevrx Inc Polymerkonjugerede metap2-inhibitorer og terapeutiske fremgangsmåder til anvendelse deraf
CN105431426A (zh) 2013-04-10 2016-03-23 新德发制药有限公司 Metap2抑制剂和治疗肥胖症的方法
US9969722B2 (en) * 2015-12-10 2018-05-15 Syndevrx, Inc. Fumagillol derivatives and polymorphs thereof
CN108697807B (zh) 2016-01-11 2021-11-26 辛德弗雷克斯公司 代谢功能障碍引起的肿瘤的治疗
CN113453721B (zh) 2018-10-26 2025-09-16 辛德弗雷克斯公司 Metap2抑制剂的生物标志物及其应用
WO2024040009A2 (en) * 2022-08-17 2024-02-22 Primetime Life Sciences, Llc Inhibitors of methionine aminopeptidase-2 and methods of preparation and uses thereof

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