JP2023553094A5 - - Google Patents

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Publication number
JP2023553094A5
JP2023553094A5 JP2023534880A JP2023534880A JP2023553094A5 JP 2023553094 A5 JP2023553094 A5 JP 2023553094A5 JP 2023534880 A JP2023534880 A JP 2023534880A JP 2023534880 A JP2023534880 A JP 2023534880A JP 2023553094 A5 JP2023553094 A5 JP 2023553094A5
Authority
JP
Japan
Prior art keywords
optionally
substituted
atoms
alkyl
hydrogen atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023534880A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023553094A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CA2021/051755 external-priority patent/WO2022120475A1/en
Publication of JP2023553094A publication Critical patent/JP2023553094A/ja
Publication of JP2023553094A5 publication Critical patent/JP2023553094A5/ja
Pending legal-status Critical Current

Links

JP2023534880A 2020-12-07 2021-12-07 中枢神経系障害の治療のためのセロトニン作動性薬としての3位環-アミンインドール誘導体 Pending JP2023553094A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063122181P 2020-12-07 2020-12-07
US63/122,181 2020-12-07
PCT/CA2021/051755 WO2022120475A1 (en) 2020-12-07 2021-12-07 3-cyclic amine-indole derivatives as serotonergic agents for the treatment of cns disorders

Publications (2)

Publication Number Publication Date
JP2023553094A JP2023553094A (ja) 2023-12-20
JP2023553094A5 true JP2023553094A5 (cg-RX-API-DMAC10.html) 2024-12-06

Family

ID=81973031

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023534880A Pending JP2023553094A (ja) 2020-12-07 2021-12-07 中枢神経系障害の治療のためのセロトニン作動性薬としての3位環-アミンインドール誘導体

Country Status (10)

Country Link
US (1) US20240051978A1 (cg-RX-API-DMAC10.html)
EP (1) EP4255913A4 (cg-RX-API-DMAC10.html)
JP (1) JP2023553094A (cg-RX-API-DMAC10.html)
KR (1) KR20230117597A (cg-RX-API-DMAC10.html)
CN (1) CN116917305A (cg-RX-API-DMAC10.html)
AU (1) AU2021394129A1 (cg-RX-API-DMAC10.html)
CA (1) CA3201080A1 (cg-RX-API-DMAC10.html)
IL (1) IL303467A (cg-RX-API-DMAC10.html)
MX (1) MX2023006652A (cg-RX-API-DMAC10.html)
WO (1) WO2022120475A1 (cg-RX-API-DMAC10.html)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3519816A4 (en) 2016-09-29 2020-05-06 The Regents of the University of California CONNECTIONS FOR INCREASING NEURONAL PLASTICITY
KR102946120B1 (ko) 2019-02-27 2026-03-30 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 뇌 장애를 치료하기 위한 아제피노-인돌 및 다른 헤테로사이클
WO2022221415A2 (en) 2021-04-13 2022-10-20 The Regents Of The University Of California Tetracyclic compounds for treating brain disorders
KR20240017363A (ko) * 2021-06-02 2024-02-07 세인트 조셉스 유니버시티 플루오린화 트립타민 화합물, 이의 유사체 및 이를 사용하는 방법
JP2025502615A (ja) 2021-12-15 2025-01-28 デリックス セラピューティクス,インク. フェノキシおよびベンジルオキシ置換サイコプラストゲンならびにその使用
EP4447954A4 (en) * 2021-12-16 2025-12-03 Icahn School Med Mount Sinai HETEROCYCLIC COMPOUNDS AS POLARIZED 5HT2A AGONISTS
WO2023168023A1 (en) 2022-03-04 2023-09-07 Reset Pharmaceuticals, Inc. Co-crystals or salts comprising psilocin
EP4551211A1 (en) * 2022-07-08 2025-05-14 Institut Curie Serotonin analogues for use in treating metalloptosis-associated disorders
US12396981B2 (en) 2023-03-09 2025-08-26 William Shulman Methods of using DMT

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5789402A (en) * 1995-01-17 1998-08-04 Eli Lilly Company Compounds having effects on serotonin-related systems
US5846982A (en) * 1996-06-14 1998-12-08 Eli Lilly And Company Inhibition of serotonin reuptake
US6133287A (en) * 1998-03-24 2000-10-17 Allelix Biopharmaceuticals Inc. Piperidine-indole compounds having 5-HT6 affinity
GB9810886D0 (en) * 1998-05-13 1998-07-22 Lilly Industries Ltd Pharmaceutical compounds
EP1173432B9 (en) * 1999-04-21 2008-10-15 NPS Allelix Corp. Piperidine-indole compounds having 5-ht6 affinity
EA200300717A1 (ru) * 2000-12-22 2003-12-25 Уайт Гетероциклилиндазольные и -азаиндазольные соединения в качестве 5-гидрокситриптамин-6-лигандов
WO2004069828A1 (ja) * 2003-02-04 2004-08-19 Mitsubishi Pharma Corporation ピペリジン化合物およびその医薬用途
WO2005066157A1 (en) * 2004-01-02 2005-07-21 Suven Life Sciences 3-(pyrolidin-3-l) indoles as 5-ht6 receptor modulators
EP1984351A1 (en) * 2006-02-17 2008-10-29 Memory Pharmaceuticals Corporation Compounds having 5-ht6 receptor affinity
US8912220B2 (en) * 2009-08-10 2014-12-16 Galenea Pharmaceuticals Compounds and methods of use thereof
US20230405026A1 (en) * 2020-11-06 2023-12-21 Mynd Life Sciences Inc. A Method of Treating Depression by Immune Modulation

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