JP2023551110A5 - - Google Patents
Info
- Publication number
- JP2023551110A5 JP2023551110A5 JP2023527430A JP2023527430A JP2023551110A5 JP 2023551110 A5 JP2023551110 A5 JP 2023551110A5 JP 2023527430 A JP2023527430 A JP 2023527430A JP 2023527430 A JP2023527430 A JP 2023527430A JP 2023551110 A5 JP2023551110 A5 JP 2023551110A5
- Authority
- JP
- Japan
- Prior art keywords
- ethyl
- fluorobicyclo
- dicyclopropyl
- pentan
- imidazo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB2017642.6A GB202017642D0 (en) | 2020-11-09 | 2020-11-09 | Therapeputic agents |
| GB2017642.6 | 2020-11-09 | ||
| GB2108945.3 | 2021-06-22 | ||
| GBGB2108945.3A GB202108945D0 (en) | 2021-06-22 | 2021-06-22 | Therapeutic agents |
| PCT/EP2021/080251 WO2022096412A1 (en) | 2020-11-09 | 2021-11-01 | Dicyclopropylmethyl derivatives as il-17 modulators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023551110A JP2023551110A (ja) | 2023-12-07 |
| JP2023551110A5 true JP2023551110A5 (https=) | 2024-10-15 |
Family
ID=78536191
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023527430A Pending JP2023551110A (ja) | 2020-11-09 | 2021-11-01 | Il‐17モジュレーターとしてのジシクロプロピルメチル誘導体 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20230399328A1 (https=) |
| EP (1) | EP4240742A1 (https=) |
| JP (1) | JP2023551110A (https=) |
| CN (1) | CN116406267A (https=) |
| CA (1) | CA3199816A1 (https=) |
| WO (1) | WO2022096412A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR126255A1 (es) | 2021-07-01 | 2023-10-04 | UCB Biopharma SRL | Derivados de imidazotriazina como moduladores de il-17 |
| WO2023025783A1 (en) | 2021-08-23 | 2023-03-02 | Leo Pharma A/S | Small molecule modulators of il-17 |
| WO2023111181A1 (en) | 2021-12-16 | 2023-06-22 | Leo Pharma A/S | Small molecule modulators of il-17 |
| WO2023166172A1 (en) | 2022-03-04 | 2023-09-07 | Leo Pharma A/S | Small molecule modulators of il-17 |
| GB202210731D0 (en) | 2022-07-22 | 2022-09-07 | UCB Biopharma SRL | Therapeutic agents |
| TW202430165A (zh) | 2022-12-02 | 2024-08-01 | 丹麥商理奧藥品公司 | Il-17之小分子調節劑 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2242504B1 (en) | 2008-01-09 | 2021-07-14 | The Schepens Eye Research Institute, Inc. | Therapeutic compositions for treatment of ocular inflammatory disorders |
| EP2809660B1 (en) | 2012-02-02 | 2016-01-20 | Ensemble Therapeutics Corporation | Macrocyclic compounds for modulating il-17 |
| WO2014066726A2 (en) | 2012-10-26 | 2014-05-01 | Ensemble Therapeutics Corporation | Compounds for modulating il-17 |
| GB201709456D0 (en) | 2017-06-14 | 2017-07-26 | Ucb Biopharma Sprl | Therapeutic agents |
| US11472794B2 (en) * | 2018-01-15 | 2022-10-18 | UCB Biopharma SRL | Fused imidazole derivatives as IL-17 modulators |
| CN110511213B (zh) | 2018-05-22 | 2021-10-19 | 成都先导药物开发股份有限公司 | 一种免疫调节剂 |
| EP3820567A1 (en) | 2018-07-12 | 2021-05-19 | UCB Biopharma SRL | Spirocyclic indane analogues as il-17 modulators |
| GB201820165D0 (en) | 2018-12-11 | 2019-01-23 | Ucb Biopharma Sprl | Therapeutic agents |
| GB201820166D0 (en) | 2018-12-11 | 2019-01-23 | Ucb Biopharma Sprl | Therapeutic agents |
| SG11202106444WA (en) * | 2018-12-19 | 2021-07-29 | Leo Pharma As | Amino-acid anilides as small molecule modulators of il-17 |
| TWI752400B (zh) | 2019-01-07 | 2022-01-11 | 美商美國禮來大藥廠 | Il-17a抑制劑 |
| US20220162191A1 (en) | 2019-03-08 | 2022-05-26 | Leo Pharma A/S | Small molecule modulators of il-17 |
| GB201909191D0 (en) | 2019-06-26 | 2019-08-07 | Ucb Biopharma Sprl | Therapeutic agents |
| GB201909190D0 (en) | 2019-06-26 | 2019-08-07 | Ucb Biopharma Sprl | Therapeutic agents |
| GB201909194D0 (en) | 2019-06-26 | 2019-08-07 | Ucb Biopharma Sprl | Therapeutic agents |
-
2021
- 2021-11-01 US US18/035,332 patent/US20230399328A1/en active Pending
- 2021-11-01 JP JP2023527430A patent/JP2023551110A/ja active Pending
- 2021-11-01 EP EP21805444.3A patent/EP4240742A1/en active Pending
- 2021-11-01 CN CN202180075513.7A patent/CN116406267A/zh active Pending
- 2021-11-01 CA CA3199816A patent/CA3199816A1/en active Pending
- 2021-11-01 WO PCT/EP2021/080251 patent/WO2022096412A1/en not_active Ceased
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