JP2023544446A5 - - Google Patents

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Publication number
JP2023544446A5
JP2023544446A5 JP2023542830A JP2023542830A JP2023544446A5 JP 2023544446 A5 JP2023544446 A5 JP 2023544446A5 JP 2023542830 A JP2023542830 A JP 2023542830A JP 2023542830 A JP2023542830 A JP 2023542830A JP 2023544446 A5 JP2023544446 A5 JP 2023544446A5
Authority
JP
Japan
Prior art keywords
substituted
unsubstituted
group
polycyclic
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023542830A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023544446A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/051375 external-priority patent/WO2022061312A1/en
Publication of JP2023544446A publication Critical patent/JP2023544446A/ja
Publication of JP2023544446A5 publication Critical patent/JP2023544446A5/ja
Pending legal-status Critical Current

Links

JP2023542830A 2020-09-21 2021-09-21 Sik阻害剤およびその使用方法 Pending JP2023544446A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063081089P 2020-09-21 2020-09-21
US63/081,089 2020-09-21
PCT/US2021/051375 WO2022061312A1 (en) 2020-09-21 2021-09-21 Sik inhibitors and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2023544446A JP2023544446A (ja) 2023-10-23
JP2023544446A5 true JP2023544446A5 (https=) 2024-10-01

Family

ID=80775691

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023542830A Pending JP2023544446A (ja) 2020-09-21 2021-09-21 Sik阻害剤およびその使用方法

Country Status (7)

Country Link
US (1) US20230265099A1 (https=)
EP (1) EP4213851A4 (https=)
JP (1) JP2023544446A (https=)
CN (1) CN117136061A (https=)
AU (1) AU2021343539A1 (https=)
CA (1) CA3193194A1 (https=)
WO (1) WO2022061312A1 (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4526307A1 (en) * 2022-05-17 2025-03-26 Soltego, Inc. Pyrimidopyrimidone compounds and methods of use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN104418860B (zh) * 2013-08-20 2016-09-07 中国科学院广州生物医药与健康研究院 嘧啶并杂环类化合物及其药用组合物和应用
WO2018009544A1 (en) * 2016-07-05 2018-01-11 The Broad Institute, Inc. Bicyclic urea kinase inhibitors and uses thereof
US11241435B2 (en) * 2016-09-16 2022-02-08 The General Hospital Corporation Uses of salt-inducible kinase (SIK) inhibitors for treating osteoporosis
AU2018226771B2 (en) * 2017-02-28 2023-11-23 Dana-Farber Cancer Institute, Inc. Uses of pyrimidopyrimidinones as SIK inhibitors
CA3124574A1 (en) * 2018-12-28 2020-07-02 Spv Therapeutics Inc. Cyclin-dependent kinase inhibitors
AU2021262482A1 (en) * 2020-04-28 2023-01-05 Iomx Therapeutics Ag Bicyclic kinase inhibitors and uses thereof

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