JP2023539336A5 - - Google Patents

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Publication number
JP2023539336A5
JP2023539336A5 JP2023514050A JP2023514050A JP2023539336A5 JP 2023539336 A5 JP2023539336 A5 JP 2023539336A5 JP 2023514050 A JP2023514050 A JP 2023514050A JP 2023514050 A JP2023514050 A JP 2023514050A JP 2023539336 A5 JP2023539336 A5 JP 2023539336A5
Authority
JP
Japan
Prior art keywords
disorder
disorders
tetrahydro
pyridine
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023514050A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023539336A (ja
JP7761635B2 (ja
JP7761635B6 (ja
Filing date
Publication date
Priority claimed from GBGB2013558.8A external-priority patent/GB202013558D0/en
Application filed filed Critical
Publication of JP2023539336A publication Critical patent/JP2023539336A/ja
Publication of JP2023539336A5 publication Critical patent/JP2023539336A5/ja
Publication of JP7761635B2 publication Critical patent/JP7761635B2/ja
Application granted granted Critical
Publication of JP7761635B6 publication Critical patent/JP7761635B6/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023514050A 2020-08-28 2021-08-31 Gpr52モジュレーター化合物 Active JP7761635B6 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2013558.8 2020-08-28
GBGB2013558.8A GB202013558D0 (en) 2020-08-28 2020-08-28 GRP52 Modularor compounds
PCT/GB2021/052247 WO2022043714A1 (en) 2020-08-28 2021-08-31 Gpr52 modulator compounds

Publications (4)

Publication Number Publication Date
JP2023539336A JP2023539336A (ja) 2023-09-13
JP2023539336A5 true JP2023539336A5 (enExample) 2024-09-06
JP7761635B2 JP7761635B2 (ja) 2025-10-28
JP7761635B6 JP7761635B6 (ja) 2025-11-27

Family

ID=72749711

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023514050A Active JP7761635B6 (ja) 2020-08-28 2021-08-31 Gpr52モジュレーター化合物

Country Status (12)

Country Link
US (1) US20230348416A1 (enExample)
EP (1) EP4204408A1 (enExample)
JP (1) JP7761635B6 (enExample)
KR (1) KR20230058132A (enExample)
CN (1) CN116507622B (enExample)
AU (1) AU2021330379A1 (enExample)
BR (1) BR112023003696A2 (enExample)
CA (1) CA3193487A1 (enExample)
GB (1) GB202013558D0 (enExample)
IL (1) IL301007B2 (enExample)
MX (1) MX2023002389A (enExample)
WO (1) WO2022043714A1 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB202003668D0 (en) 2020-03-13 2020-04-29 Heptares Therapeutics Ltd GPR52 Modulator compounds
EP4139284A1 (en) 2020-04-22 2023-03-01 Neurocrine Biosciences, Inc. Gpr52 modulators and methods of use
CN122555695A (zh) * 2023-11-29 2026-08-11 爱克堤欧生物科学股份有限公司 可用作kcnt1抑制剂的杂环化合物
CN121313618B (zh) * 2025-12-09 2026-07-21 杭州师范大学附属医院(杭州市第二人民医院) 丙酸在制备治疗肝豆状核变性肠肝轴紊乱的药物中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX373876B (es) * 2015-04-29 2020-03-26 Arena Pharm Inc 1-heteroaril-indolin-4-carboxamidas como moduladores de gpr52 útiles para el tratamiento o prevención de trastornos relacionados a las mismas.
WO2017077280A1 (en) * 2015-11-02 2017-05-11 Sonia Lain Tetrahydroindazoles and medical uses thereof
WO2021009003A1 (en) * 2019-07-16 2021-01-21 Universität Hamburg Computer-based identification of types in the empirical sciences by tangle theory
CN114650992A (zh) * 2019-11-08 2022-06-21 赫普泰雅治疗有限公司 Gpr52调节剂化合物

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