JP2023538521A5 - - Google Patents

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Publication number
JP2023538521A5
JP2023538521A5 JP2023507887A JP2023507887A JP2023538521A5 JP 2023538521 A5 JP2023538521 A5 JP 2023538521A5 JP 2023507887 A JP2023507887 A JP 2023507887A JP 2023507887 A JP2023507887 A JP 2023507887A JP 2023538521 A5 JP2023538521 A5 JP 2023538521A5
Authority
JP
Japan
Prior art keywords
optionally substituted
substituted
group
pharmaceutically acceptable
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023507887A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023538521A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/044907 external-priority patent/WO2022032071A1/en
Publication of JP2023538521A publication Critical patent/JP2023538521A/ja
Publication of JP2023538521A5 publication Critical patent/JP2023538521A5/ja
Pending legal-status Critical Current

Links

JP2023507887A 2020-08-07 2021-08-06 キナーゼ阻害剤およびその使用 Pending JP2023538521A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063063113P 2020-08-07 2020-08-07
US63/063,113 2020-08-07
PCT/US2021/044907 WO2022032071A1 (en) 2020-08-07 2021-08-06 Kinase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2023538521A JP2023538521A (ja) 2023-09-08
JP2023538521A5 true JP2023538521A5 (https=) 2024-08-15

Family

ID=77711412

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023507887A Pending JP2023538521A (ja) 2020-08-07 2021-08-06 キナーゼ阻害剤およびその使用

Country Status (10)

Country Link
US (1) US20230303570A1 (https=)
EP (1) EP4192582A1 (https=)
JP (1) JP2023538521A (https=)
KR (1) KR20230112605A (https=)
CN (1) CN116710453A (https=)
AU (1) AU2021321536A1 (https=)
BR (1) BR112023002248A2 (https=)
CA (1) CA3179671A1 (https=)
MX (1) MX2023001312A (https=)
WO (1) WO2022032071A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4577546A1 (en) * 2022-08-25 2025-07-02 Enliven Inc. Naphthyridine compounds for inhibition of raf kinases
WO2024199388A1 (zh) * 2023-03-29 2024-10-03 微境生物医药科技(上海)有限公司 作为myt1抑制剂的化合物
WO2025064567A1 (en) * 2023-09-19 2025-03-27 Enliven Inc. Tricyclic phenols for inhibition of raf kinases
WO2025152919A1 (en) * 2024-01-15 2025-07-24 Impact Therapeutics (Shanghai) , Inc. Crystal forms of a weel inhibitor and preparation method thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2006503802A (ja) * 2002-04-03 2006-02-02 エフ.ホフマン−ラ ロシュ アーゲー イミダゾ縮合化合物
EP2348020A1 (en) 2009-12-23 2011-07-27 Esteve Química, S.A. Preparation process of erlotinib
FR2974088A1 (fr) * 2011-04-12 2012-10-19 Pf Medicament Composes pyrazolo[3,4-b]pyridines tri- et tetracycliques comme agent anticancereux
RU2019102647A (ru) * 2016-07-01 2020-08-03 Г1 Терапьютикс, Инк. Антипролиферационные средства на основе пиримидина
EP3684772B1 (en) * 2017-09-20 2023-12-06 ABM Therapeutics Corporation Cyclic iminopyrimidine derivatives as kinase inhibitors
CN110950867A (zh) * 2018-09-27 2020-04-03 首药控股(北京)有限公司 一种fgfr4激酶抑制剂及其制备方法和用途

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