JP2023538393A5 - - Google Patents

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Publication number
JP2023538393A5
JP2023538393A5 JP2023512226A JP2023512226A JP2023538393A5 JP 2023538393 A5 JP2023538393 A5 JP 2023538393A5 JP 2023512226 A JP2023512226 A JP 2023512226A JP 2023512226 A JP2023512226 A JP 2023512226A JP 2023538393 A5 JP2023538393 A5 JP 2023538393A5
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JP
Japan
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JP2023512226A
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Japanese (ja)
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JPWO2022040259A5 (https=
JP7813775B2 (ja
JP2023538393A (ja
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Priority claimed from PCT/US2021/046420 external-priority patent/WO2022040259A1/en
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Publication of JP2023538393A5 publication Critical patent/JP2023538393A5/ja
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JP2023512226A 2020-08-19 2021-08-18 線維症の処置のためのtlr9の阻害剤としてのイミダゾ[1,2-a]ピリジンおよび[1,2,4]トリアゾロ[1,5-a]ピリジン誘導体 Active JP7813775B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063067452P 2020-08-19 2020-08-19
US63/067,452 2020-08-19
PCT/US2021/046420 WO2022040259A1 (en) 2020-08-19 2021-08-18 Imidazo[1,2-a]pyridine and [1,2,4]triazolo[1,5-a]pyridine derivatives as tlr9 inhibitors for the treatment of fibrosis

Publications (4)

Publication Number Publication Date
JP2023538393A JP2023538393A (ja) 2023-09-07
JPWO2022040259A5 JPWO2022040259A5 (https=) 2024-08-26
JP2023538393A5 true JP2023538393A5 (https=) 2024-08-26
JP7813775B2 JP7813775B2 (ja) 2026-02-13

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ID=77693624

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Application Number Title Priority Date Filing Date
JP2023512226A Active JP7813775B2 (ja) 2020-08-19 2021-08-18 線維症の処置のためのtlr9の阻害剤としてのイミダゾ[1,2-a]ピリジンおよび[1,2,4]トリアゾロ[1,5-a]ピリジン誘導体

Country Status (13)

Country Link
US (1) US12486267B2 (https=)
EP (1) EP4200297A1 (https=)
JP (1) JP7813775B2 (https=)
KR (1) KR20230053644A (https=)
CN (1) CN116096717B (https=)
AR (1) AR123281A1 (https=)
AU (1) AU2021328575A1 (https=)
BR (1) BR112023002737A2 (https=)
CA (1) CA3190065A1 (https=)
IL (1) IL300727A (https=)
MX (1) MX2023001885A (https=)
TW (1) TW202227432A (https=)
WO (1) WO2022040259A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11807622B2 (en) 2019-01-30 2023-11-07 Insilico Medicine Ip Limited TLR 9 inhibitors
US20250163054A1 (en) * 2022-02-18 2025-05-22 Bristol-Myers Squibb Company Substituted bicyclic heteroaryl compounds useful as inhibitors of tlr9
CN120230100B (zh) * 2025-05-30 2025-09-05 中国药科大学 一种咪唑并[1,2-a]吡嗪或咪唑并[1,2-a]吡啶类化合物及其医药用途

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