JP2023537994A5 - - Google Patents
Info
- Publication number
- JP2023537994A5 JP2023537994A5 JP2023509840A JP2023509840A JP2023537994A5 JP 2023537994 A5 JP2023537994 A5 JP 2023537994A5 JP 2023509840 A JP2023509840 A JP 2023509840A JP 2023509840 A JP2023509840 A JP 2023509840A JP 2023537994 A5 JP2023537994 A5 JP 2023537994A5
- Authority
- JP
- Japan
- Prior art keywords
- aryl
- alkyl
- cycloalkyl
- heteroaryl
- acyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202063064262P | 2020-08-11 | 2020-08-11 | |
| US63/064,262 | 2020-08-11 | ||
| PCT/US2021/045446 WO2022035902A1 (en) | 2020-08-11 | 2021-08-10 | Proteasome enhancers and uses thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023537994A JP2023537994A (ja) | 2023-09-06 |
| JP2023537994A5 true JP2023537994A5 (enExample) | 2024-08-20 |
Family
ID=83103405
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023509840A Pending JP2023537994A (ja) | 2020-08-11 | 2021-08-10 | プロテアソームエンハンサーおよびその使用 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20230286982A1 (enExample) |
| EP (1) | EP4196121A4 (enExample) |
| JP (1) | JP2023537994A (enExample) |
| AU (1) | AU2021325024A1 (enExample) |
| CA (1) | CA3191436A1 (enExample) |
| MX (1) | MX2023001759A (enExample) |
| WO (1) | WO2022035902A1 (enExample) |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3238216A (en) * | 1963-06-20 | 1966-03-01 | Res Lab Dr C Janssen N V | Substituted 1, 3, 8-triaza-spiro (4, 5) decanes |
| US3956296A (en) * | 1974-12-11 | 1976-05-11 | A. H. Robins Company, Incorporated | 1-Substituted-4-benzylpiperidines |
| FR2373967A1 (fr) * | 1976-12-20 | 1978-07-13 | Wellcome Found | Derives de l'imidazoline et leur emploi comme agents pesticides |
| NZ249040A (en) * | 1992-02-06 | 1997-06-24 | Merrell Dow Pharma | Triphenyl azacycloalkane derivatives; treatment of drug resistance |
| GB9725541D0 (en) * | 1997-12-02 | 1998-02-04 | Pharmacia & Upjohn Spa | Amino-benzothiazole derivatives |
| US6011035A (en) * | 1998-06-30 | 2000-01-04 | Neuromed Technologies Inc. | Calcium channel blockers |
| US6686370B2 (en) * | 1999-12-06 | 2004-02-03 | Euro-Celtique S.A. | Triazospiro compounds having nociceptin receptor affinity |
| US6482829B2 (en) * | 2000-06-08 | 2002-11-19 | Hoffmann-La Roche Inc. | Substituted heterocyclic siprodecane compound active as an antagonist of neurokinin 1 receptor |
| GB0211759D0 (en) * | 2002-05-22 | 2002-07-03 | Glaxo Group Ltd | Novel compounds |
| CN101472924A (zh) * | 2006-06-20 | 2009-07-01 | 惠氏公司 | Kv1.5钾通道抑制剂 |
| CN101838269B (zh) * | 2009-03-18 | 2012-09-26 | 中国人民解放军军事医学科学院毒物药物研究所 | 1,3,8-三氮杂-螺[4.5]癸烷-4-酮类化合物及其医药用途 |
| WO2011143444A2 (en) * | 2010-05-14 | 2011-11-17 | President And Fellows Of Harvard College | Diphenylbutypiperidine autophagy inducers |
| IT201800007580A1 (it) * | 2018-07-27 | 2020-01-27 | Maria Cecilia Hospital Spa | Composti 1,3,8-triazaspiro e loro uso come medicamenti |
-
2021
- 2021-08-10 EP EP21856602.4A patent/EP4196121A4/en not_active Withdrawn
- 2021-08-10 CA CA3191436A patent/CA3191436A1/en active Pending
- 2021-08-10 WO PCT/US2021/045446 patent/WO2022035902A1/en not_active Ceased
- 2021-08-10 MX MX2023001759A patent/MX2023001759A/es unknown
- 2021-08-10 US US18/041,184 patent/US20230286982A1/en active Pending
- 2021-08-10 JP JP2023509840A patent/JP2023537994A/ja active Pending
- 2021-08-10 AU AU2021325024A patent/AU2021325024A1/en active Pending
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