JP2023531411A5 - - Google Patents

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Publication number
JP2023531411A5
JP2023531411A5 JP2022577145A JP2022577145A JP2023531411A5 JP 2023531411 A5 JP2023531411 A5 JP 2023531411A5 JP 2022577145 A JP2022577145 A JP 2022577145A JP 2022577145 A JP2022577145 A JP 2022577145A JP 2023531411 A5 JP2023531411 A5 JP 2023531411A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutically acceptable
hydrogen
acceptable salt
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022577145A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023531411A (ja
JP7776453B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/036706 external-priority patent/WO2021257353A1/en
Publication of JP2023531411A publication Critical patent/JP2023531411A/ja
Publication of JP2023531411A5 publication Critical patent/JP2023531411A5/ja
Application granted granted Critical
Publication of JP7776453B2 publication Critical patent/JP7776453B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022577145A 2020-06-16 2021-06-10 血漿カリクレイン阻害剤 Active JP7776453B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063039873P 2020-06-16 2020-06-16
US63/039,873 2020-06-16
PCT/US2021/036706 WO2021257353A1 (en) 2020-06-16 2021-06-10 Plasma kallikrein inhibitors

Publications (3)

Publication Number Publication Date
JP2023531411A JP2023531411A (ja) 2023-07-24
JP2023531411A5 true JP2023531411A5 (https=) 2024-05-08
JP7776453B2 JP7776453B2 (ja) 2025-11-26

Family

ID=79268261

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022577145A Active JP7776453B2 (ja) 2020-06-16 2021-06-10 血漿カリクレイン阻害剤

Country Status (10)

Country Link
US (1) US12459927B2 (https=)
EP (1) EP4164634A4 (https=)
JP (1) JP7776453B2 (https=)
KR (1) KR102931248B1 (https=)
CN (1) CN115989224B (https=)
AU (1) AU2021292449A1 (https=)
BR (1) BR112022025528A2 (https=)
CA (1) CA3182626A1 (https=)
MX (1) MX2022016321A (https=)
WO (1) WO2021257353A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20230038526A (ko) 2020-07-10 2023-03-20 머크 샤프 앤드 돔 엘엘씨 혈장 칼리크레인 억제제
US20230416227A1 (en) * 2020-09-10 2023-12-28 Merck Sharp & Dohme Llc Plasma kallikrein inhibitors
CN116120272A (zh) * 2022-12-31 2023-05-16 淮北师范大学 一种合成咯菌腈中间体2,2-二氟-1,3-苯并二噁茂-4-甲醛的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20140378474A1 (en) * 2012-01-27 2014-12-25 Novartis Ag 5-membered heteroarylcarboxamide derivatives as plasma kallikrein inhibitors
KR102736869B1 (ko) 2014-03-07 2024-12-02 바이오크리스트파마슈티컬즈,인코포레이티드 인간 혈장 칼리크레인 저해제
GB201421083D0 (en) 2014-11-27 2015-01-14 Kalvista Pharmaceuticals Ltd Enzyme inhibitors
EP3368524B1 (en) 2015-10-27 2021-08-18 Boehringer Ingelheim International GmbH Heteroarylcarboxamide derivatives as plasma kallikrein inhibitors
DK3464271T3 (da) 2016-05-31 2020-06-15 Kalvista Pharmaceuticals Ltd Pyrazolderivater som plasma-kallikreininhibitorer
BR112020000463A2 (pt) 2017-07-13 2020-07-21 Syngenta Participations Ag derivados oxadiazol microbiocidas

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