JP2023526791A5 - - Google Patents
Info
- Publication number
- JP2023526791A5 JP2023526791A5 JP2022569555A JP2022569555A JP2023526791A5 JP 2023526791 A5 JP2023526791 A5 JP 2023526791A5 JP 2022569555 A JP2022569555 A JP 2022569555A JP 2022569555 A JP2022569555 A JP 2022569555A JP 2023526791 A5 JP2023526791 A5 JP 2023526791A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- independently selected
- halogenated
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202010433988 | 2020-05-21 | ||
| CN202010433988.6 | 2020-05-21 | ||
| CN202110529033 | 2021-05-14 | ||
| CN202110529033.5 | 2021-05-14 | ||
| PCT/CN2021/095191 WO2021233427A1 (zh) | 2020-05-21 | 2021-05-21 | 并环化合物及其制备方法、药物组合物和应用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2023526791A JP2023526791A (ja) | 2023-06-23 |
| JP2023526791A5 true JP2023526791A5 (https=) | 2024-05-23 |
| JP7774312B2 JP7774312B2 (ja) | 2025-11-21 |
Family
ID=78672734
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022569555A Active JP7774312B2 (ja) | 2020-05-21 | 2021-05-21 | 縮合環化合物、それらの製造方法、医薬組成物、およびそれらの使用 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20230192683A1 (https=) |
| EP (1) | EP4155305A4 (https=) |
| JP (1) | JP7774312B2 (https=) |
| KR (1) | KR20230015333A (https=) |
| CN (2) | CN115991703A (https=) |
| AU (1) | AU2021276301A1 (https=) |
| TW (1) | TWI910166B (https=) |
| WO (1) | WO2021233427A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI860849B (zh) | 2021-09-14 | 2024-11-01 | 美商美國禮來大藥廠 | Sstr4促效劑鹽 |
| KR20240122964A (ko) | 2023-02-06 | 2024-08-13 | 에이치엘만도 주식회사 | 피스톤 밸브 조립체 및 이를 구비한 쇼크 업소버 |
| JP2026509366A (ja) | 2023-03-10 | 2026-03-18 | イーライ リリー アンド カンパニー | Ｓｓｔｒ４アゴニスト及びその塩の調製のための方法 |
| AU2024236692A1 (en) | 2023-03-10 | 2025-10-16 | Eli Lilly And Company | Methods for the preparation and dose regimens for use of sstr4 agonists and salts thereof |
| WO2024245077A1 (zh) * | 2023-05-29 | 2024-12-05 | 武汉熙瑞医药科技有限公司 | 3-氮杂-双环[3.1.0]己烷衍生物、其制备方法及其应用 |
| WO2025096300A1 (en) | 2023-10-30 | 2025-05-08 | Eli Lilly And Company | Novel methods for the preparation of 3-azabicylco[3.1,0]hexane-6-carboxamide derivatives |
| CN120965687A (zh) * | 2024-05-17 | 2025-11-18 | 广州费米子科技有限责任公司 | Sstr4激动剂类化合物的晶体形式及其制备方法和用途 |
| WO2025247982A1 (en) | 2024-05-29 | 2025-12-04 | Grünenthal GmbH | Piperazines which act as sstr4 modulators |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2685828A4 (en) * | 2011-03-17 | 2014-08-13 | Merck Sharp & Dohme | SUBSTITUTED 3-AZABICYCLO [3,1,0-] HEXAN DERIVATIVES AS CCR2 ANTAGONISTS |
| KR101556318B1 (ko) * | 2013-05-15 | 2015-10-01 | 한국과학기술연구원 | 칼슘이온 채널 조절제로서 유효한 6-피라졸일아미도-3-치환된 아자바이사이클로[3.1.0]헥산 유도체 |
| US9371282B2 (en) * | 2013-05-17 | 2016-06-21 | Centrexion Therapeutics Corporation | Somatostatin receptor subtype 4 (SSTR4) agonists |
| EP3045448A4 (en) | 2013-09-12 | 2017-01-25 | Sumitomo Chemical Company Limited | Nitrogen-containing saturated heterocyclic compound |
| CN105315293A (zh) * | 2014-07-29 | 2016-02-10 | 上海科州药物研发有限公司 | 作为蛋白激酶抑制剂的杂环化合物及其制备方法和用途 |
-
2021
- 2021-05-21 JP JP2022569555A patent/JP7774312B2/ja active Active
- 2021-05-21 AU AU2021276301A patent/AU2021276301A1/en active Pending
- 2021-05-21 CN CN202211412069.6A patent/CN115991703A/zh active Pending
- 2021-05-21 TW TW110118416A patent/TWI910166B/zh active
- 2021-05-21 EP EP21808555.3A patent/EP4155305A4/en active Pending
- 2021-05-21 CN CN202110556640.0A patent/CN113717167B/zh active Active
- 2021-05-21 WO PCT/CN2021/095191 patent/WO2021233427A1/zh not_active Ceased
- 2021-05-21 US US17/926,523 patent/US20230192683A1/en active Pending
- 2021-05-21 KR KR1020227039715A patent/KR20230015333A/ko active Pending
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2023526791A5 (https=) | ||
| US6673799B1 (en) | Cyanophenyl derivative | |
| JP7502337B2 (ja) | Ｋｒａｓ ｇ１２ｃインヒビター及びその使用 | |
| KR102309986B1 (ko) | 사이클린 의존성 키나아제 cdk9의 신규 인히비터 | |
| EP1256576B1 (en) | Fused imidazolium derivatives | |
| IL268030B2 (en) | Bicyclics as allosteric shp2 inhibitors | |
| JP2023528394A (ja) | 大環状ｊａｋ阻害剤およびその適用 | |
| US20250066342A1 (en) | Cycloalkylurea derivative | |
| ES3062921T3 (en) | Preparation method for novel rho-related protein kinase inhibitor and intermediate in preparation method | |
| JP2008528467A5 (https=) | ||
| CN107922418A (zh) | 抗微生物化合物及制备和使用所述化合物的方法 | |
| WO2019200202A1 (en) | Antagonists of human integrin (alpha4)(beta7) | |
| AU2019344107B2 (en) | N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors | |
| WO2019079485A1 (en) | AMINO-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS AND DERIVATIVES THEREOF | |
| JP2018525363A (ja) | 疼痛に対する多様な活性を有する置換アミド誘導体 | |
| KR102926129B1 (ko) | 사이클린 의존성 키나아제 9 억제제로서의 화합물 및 그의 용도 | |
| FR2943669A1 (fr) | Derives de nicotinamide,leur preparation et leur application en therapeutique | |
| JP2014520108A5 (https=) | ||
| BR112017010402B1 (pt) | Carboxamida substituída à base de tiazol e oxazol e derivados de ureia como ligantes de receptor vanilóide ii | |
| JP2023528073A (ja) | Ｇｐｒ６５モジュレーターとしてのｎ－フェニルアミノカルボニル、ピリジノ－、ピリミジノ及びベンゾトロパン | |
| JP2024511389A5 (https=) | ||
| RU2444515C2 (ru) | Производное амида индазолакриловой кислоты | |
| KR20260006627A (ko) | 헤테로방향족 인돌설폰아미드 | |
| JP2022510700A5 (https=) | ||
| ES3013859T3 (en) | Mdm2 inhibitor, preparation method therefor, pharmaceutical composition thereof, and use thereof |