JP2023521032A5 - - Google Patents

Info

Publication number
JP2023521032A5
JP2023521032A5 JP2022560236A JP2022560236A JP2023521032A5 JP 2023521032 A5 JP2023521032 A5 JP 2023521032A5 JP 2022560236 A JP2022560236 A JP 2022560236A JP 2022560236 A JP2022560236 A JP 2022560236A JP 2023521032 A5 JP2023521032 A5 JP 2023521032A5
Authority
JP
Japan
Prior art keywords
methyl
pyridine
oxy
dichlorophenyl
piperidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022560236A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023521032A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/025382 external-priority patent/WO2021202874A1/en
Publication of JP2023521032A publication Critical patent/JP2023521032A/ja
Publication of JP2023521032A5 publication Critical patent/JP2023521032A5/ja
Pending legal-status Critical Current

Links

JP2022560236A 2020-04-02 2021-04-01 コロナウイルス感染症を処置するためのフーリンインヒビター Pending JP2023521032A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US202063004365P 2020-04-02 2020-04-02
US63/004,365 2020-04-02
US202063013382P 2020-04-21 2020-04-21
US63/013,382 2020-04-21
US202163156058P 2021-03-03 2021-03-03
US63/156,058 2021-03-03
PCT/US2021/025382 WO2021202874A1 (en) 2020-04-02 2021-04-01 Furin inhibitors for treating coronavirus infections

Publications (2)

Publication Number Publication Date
JP2023521032A JP2023521032A (ja) 2023-05-23
JP2023521032A5 true JP2023521032A5 (https=) 2024-04-11

Family

ID=75660352

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022560236A Pending JP2023521032A (ja) 2020-04-02 2021-04-01 コロナウイルス感染症を処置するためのフーリンインヒビター

Country Status (9)

Country Link
US (1) US20230149401A1 (https=)
EP (1) EP4125897A1 (https=)
JP (1) JP2023521032A (https=)
KR (1) KR20220167296A (https=)
CN (1) CN115666567A (https=)
AU (1) AU2021249149A1 (https=)
CA (1) CA3173921A1 (https=)
IL (1) IL296885A (https=)
WO (1) WO2021202874A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN115583984A (zh) * 2022-01-11 2023-01-10 嘉兴安谛康生物科技有限公司 氮杂螺类化合物及其制备方法、药物组合物和用途
DE102023126563A1 (de) * 2023-09-28 2025-04-03 Philipps-Universität Marburg, Körperschaft des öffentlichen Rechts Hemmstoffe der Proproteinkonvertase Furin, Verfahren zu deren Herstellung und Verwendung

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070116716A1 (en) * 2003-12-10 2007-05-24 Shuo Shen Sars coronavirus s proteins and uses thereof
EP2478766A3 (en) 2007-05-09 2012-08-15 Burnham Institute for Medical Research Targeting host proteinases as a therapeutic strategy against viral and bacterial pathogens
BR112020022961A2 (pt) * 2018-05-11 2021-02-17 Glaxosmithkline Intellectual Property Development Limited inibidores de furina

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