JP2023507402A5 - - Google Patents

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Publication number
JP2023507402A5
JP2023507402A5 JP2022537305A JP2022537305A JP2023507402A5 JP 2023507402 A5 JP2023507402 A5 JP 2023507402A5 JP 2022537305 A JP2022537305 A JP 2022537305A JP 2022537305 A JP2022537305 A JP 2022537305A JP 2023507402 A5 JP2023507402 A5 JP 2023507402A5
Authority
JP
Japan
Prior art keywords
alkyl
substituted
hydrogen
heterocycloalkyl
compound according
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022537305A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023507402A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/066073 external-priority patent/WO2021127480A1/en
Publication of JP2023507402A publication Critical patent/JP2023507402A/ja
Publication of JP2023507402A5 publication Critical patent/JP2023507402A5/ja
Pending legal-status Critical Current

Links

JP2022537305A 2019-12-19 2020-12-18 Ｃ１７位に窒素ベースの置換基を有する合成トリテルペノイドおよびその使用方法 Pending JP2023507402A (ja)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201962950927P 2019-12-19 2019-12-19
US201962950919P 2019-12-19 2019-12-19
US62/950,919 2019-12-19
US62/950,927 2019-12-19
US202063198310P 2020-10-09 2020-10-09
US63/198,310 2020-10-09
PCT/US2020/066073 WO2021127480A1 (en) 2019-12-19 2020-12-18 Synthetic triterpenoids with nitrogen-based substituents at c-17 and methods of use thereof

Publications (2)

Publication Number Publication Date
JP2023507402A JP2023507402A (ja) 2023-02-22
JP2023507402A5 true JP2023507402A5 (https=) 2023-12-25

Family

ID=74554207

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022537305A Pending JP2023507402A (ja) 2019-12-19 2020-12-18 Ｃ１７位に窒素ベースの置換基を有する合成トリテルペノイドおよびその使用方法

Country Status (20)

Country Link
US (1) US20230111914A1 (https=)
EP (1) EP4077347A1 (https=)
JP (1) JP2023507402A (https=)
KR (1) KR20220116209A (https=)
CN (1) CN115087660A (https=)
AU (1) AU2020405181A1 (https=)
BR (1) BR112022011919A2 (https=)
CA (1) CA3159778A1 (https=)
CL (1) CL2022001661A1 (https=)
CO (1) CO2022010070A2 (https=)
CR (1) CR20220345A (https=)
DO (1) DOP2022000127A (https=)
EC (1) ECSP22055210A (https=)
IL (1) IL293876B2 (https=)
MX (1) MX2022007595A (https=)
PE (1) PE20221662A1 (https=)
PH (1) PH12022551493A1 (https=)
SA (1) SA522432999B1 (https=)
TW (1) TWI889738B (https=)
WO (1) WO2021127480A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5529851B2 (ja) 2008-04-18 2014-06-25 リアタ ファーマシューティカルズ インコーポレイテッド 抗酸化炎症モジュレーター：ｃ−１７においてアミノ改変およびその他の改変を加えたオレアノール酸誘導体
JP7074674B2 (ja) 2015-09-23 2022-05-24 リアタ ファーマシューティカルズ インコーポレイテッド Ｉｌ－１７の阻害及び他の使用のためのｃ４修飾オレアノール酸誘導体
AU2021397631A1 (en) * 2020-12-11 2023-07-20 Reata Pharmaceuticals Holdings, LLC Synthetic triterpenoids for use in therapy
CN117964678A (zh) * 2024-01-29 2024-05-03 烟台大学 C17位杂芳族羰基修饰的齐墩果烷三萜衍生物及其制备方法和用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5529851B2 (ja) * 2008-04-18 2014-06-25 リアタ ファーマシューティカルズ インコーポレイテッド 抗酸化炎症モジュレーター：ｃ−１７においてアミノ改変およびその他の改変を加えたオレアノール酸誘導体
MX2010011439A (es) * 2008-04-18 2011-01-25 Reata Pharmaceuticals Inc Moduladores de inflamacion antioxidantes: derivados del acido oleanolico homologacion c-17.
KR101713140B1 (ko) * 2008-04-18 2017-03-08 리타 파마슈티컬스 잉크. Ｃ-환에서 포화된 산화방지성 염증 조절제 올레아놀산 유도체
AR096046A1 (es) * 2013-04-24 2015-12-02 Abbvie Inc Derivados de 2,2-difluoropropanamida de metil bardoxolona, formas polimórficas y métodos de uso
MX2021003643A (es) * 2018-09-28 2021-08-19 Sichuan Haisco Pharmaceutical Co Ltd Derivados de terpenoides y usos de los mismos.

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