JP2023503465A5 - - Google Patents

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Publication number
JP2023503465A5
JP2023503465A5 JP2022530662A JP2022530662A JP2023503465A5 JP 2023503465 A5 JP2023503465 A5 JP 2023503465A5 JP 2022530662 A JP2022530662 A JP 2022530662A JP 2022530662 A JP2022530662 A JP 2022530662A JP 2023503465 A5 JP2023503465 A5 JP 2023503465A5
Authority
JP
Japan
Prior art keywords
alkyl
membered
cycloalkyl
group
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022530662A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023503465A (ja
JP7691753B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/IB2020/061158 external-priority patent/WO2021105908A1/en
Publication of JP2023503465A publication Critical patent/JP2023503465A/ja
Publication of JP2023503465A5 publication Critical patent/JP2023503465A5/ja
Application granted granted Critical
Publication of JP7691753B2 publication Critical patent/JP7691753B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022530662A 2019-11-25 2020-11-25 ベータ-グルコセレブロシダーゼの活性の変質に関連する状態におけるヘテロアリール化合物およびその治療的使用 Active JP7691753B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP19383037.9 2019-11-25
EP19383037 2019-11-25
PCT/IB2020/061158 WO2021105908A1 (en) 2019-11-25 2020-11-25 Heteroaryl compounds and therapeutic uses thereof in conditions associated with the alteration of the activity of beta-glucocerebrosidase

Publications (3)

Publication Number Publication Date
JP2023503465A JP2023503465A (ja) 2023-01-30
JP2023503465A5 true JP2023503465A5 (https=) 2023-11-17
JP7691753B2 JP7691753B2 (ja) 2025-06-12

Family

ID=68808239

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022530662A Active JP7691753B2 (ja) 2019-11-25 2020-11-25 ベータ-グルコセレブロシダーゼの活性の変質に関連する状態におけるヘテロアリール化合物およびその治療的使用

Country Status (10)

Country Link
US (1) US20230107499A1 (https=)
EP (1) EP4065563A1 (https=)
JP (1) JP7691753B2 (https=)
KR (1) KR20220150878A (https=)
CN (1) CN115348959B (https=)
AU (1) AU2020394602A1 (https=)
BR (1) BR112022010126A2 (https=)
IL (1) IL293309A (https=)
MX (1) MX2022006065A (https=)
WO (1) WO2021105908A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4642455A1 (en) 2022-12-30 2025-11-05 GT Gain Therapeutics SA Method of treating tauopathies
WO2025221055A1 (ko) * 2024-04-18 2025-10-23 에스케이바이오팜 주식회사 유레아 화합물 및 이의 용도

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1052988A (https=) * 1962-07-03
ES2273047T3 (es) * 2002-10-28 2007-05-01 Bayer Healthcare Ag Fenilaminopirimidinas sustituidas con heteroariloxi como inhibidores de rho-cinasa.
SI2995306T1 (sl) 2009-10-19 2019-04-30 Amicus Therapeutics, Inc. Novi sestavki za preprečevanje in/ali zdravljenje motenj lizosomskega shranjevanja
KR101987736B1 (ko) 2011-03-18 2019-06-11 젠자임 코포레이션 글루코실세라마이드 합성효소 억제제
MA42189A (fr) * 2015-04-15 2018-04-18 Biomarin Pharm Inc Mã‰thodes de traitement des troubles du stockage lysosomal
CN110325516A (zh) * 2016-12-29 2019-10-11 米尼奥尔克斯治疗有限公司 杂芳基化合物和它们的用途

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