JP2023156372A5 - - Google Patents

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Publication number
JP2023156372A5
JP2023156372A5 JP2023123302A JP2023123302A JP2023156372A5 JP 2023156372 A5 JP2023156372 A5 JP 2023156372A5 JP 2023123302 A JP2023123302 A JP 2023123302A JP 2023123302 A JP2023123302 A JP 2023123302A JP 2023156372 A5 JP2023156372 A5 JP 2023156372A5
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JP
Japan
Prior art keywords
cancer
compound
medicament
manufacture
effective amount
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Application number
JP2023123302A
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English (en)
Japanese (ja)
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JP2023156372A (ja
JP7778750B2 (ja
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Priority claimed from JP2020530441A external-priority patent/JP7424639B2/ja
Application filed filed Critical
Publication of JP2023156372A publication Critical patent/JP2023156372A/ja
Publication of JP2023156372A5 publication Critical patent/JP2023156372A5/ja
Priority to JP2025168516A priority Critical patent/JP2026012715A/ja
Application granted granted Critical
Publication of JP7778750B2 publication Critical patent/JP7778750B2/ja
Active legal-status Critical Current
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JP2023123302A 2017-08-11 2023-07-28 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態 Active JP7778750B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025168516A JP2026012715A (ja) 2017-08-11 2025-10-06 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201762544277P 2017-08-11 2017-08-11
US62/544,277 2017-08-11
JP2020530441A JP7424639B2 (ja) 2017-08-11 2018-08-10 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態
PCT/US2018/046203 WO2019032958A1 (en) 2017-08-11 2018-08-10 SOLID FORMS OF 3- (5-FLUOROBENZOFURAN-3-YL) -4- (5-METHYL-5H [1,3] DIOXOLO [4,5-F] INDOL-7-YL) PYRROLE-2,5-DIONE

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2020530441A Division JP7424639B2 (ja) 2017-08-11 2018-08-10 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025168516A Division JP2026012715A (ja) 2017-08-11 2025-10-06 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Publications (3)

Publication Number Publication Date
JP2023156372A JP2023156372A (ja) 2023-10-24
JP2023156372A5 true JP2023156372A5 (https=) 2024-04-12
JP7778750B2 JP7778750B2 (ja) 2025-12-02

Family

ID=63405430

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2020530441A Active JP7424639B2 (ja) 2017-08-11 2018-08-10 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態
JP2023123302A Active JP7778750B2 (ja) 2017-08-11 2023-07-28 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態
JP2025168516A Pending JP2026012715A (ja) 2017-08-11 2025-10-06 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2020530441A Active JP7424639B2 (ja) 2017-08-11 2018-08-10 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025168516A Pending JP2026012715A (ja) 2017-08-11 2025-10-06 3-(5-フルオロベンゾフラン-3-イル)-4-(5-メチル-5H-[1,3]ジオキソロ[4,5-f]インドール-7-イル)ピロール-2,5-ジオンの固体形態

Country Status (16)

Country Link
US (3) US11136334B2 (https=)
EP (1) EP3665176B1 (https=)
JP (3) JP7424639B2 (https=)
KR (3) KR20250070131A (https=)
CN (2) CN111247153B (https=)
AU (3) AU2018313259B2 (https=)
BR (1) BR112020002892A2 (https=)
CA (1) CA3072240A1 (https=)
DK (1) DK3665176T3 (https=)
ES (1) ES2974328T3 (https=)
FI (1) FI3665176T3 (https=)
IL (2) IL313800A (https=)
MX (3) MX2020001547A (https=)
PL (1) PL3665176T3 (https=)
PT (1) PT3665176T (https=)
WO (1) WO2019032958A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3697794T (pt) * 2017-10-16 2026-03-04 Actuate Therapeutics Inc Formas sólidas de 3-(5-fluorobenzofuran-3-il)-4-(5-metil-5h-[1,3]dioxolo[4,5-f]indol-7-il)pirrol-2,5-diona
EP3793545A4 (en) * 2018-05-17 2022-04-06 Actuate Therapeutics Inc. TREATMENT OF IDIOPATHIC PULMONARY FIBROSIS WITH BETA INHIBITORS IN THE FORM OF GLYCOGEN SYNTHASE KINASE 3
JP2025525407A (ja) 2022-06-27 2025-08-05 アクチュエイト セラピューティクス インク. エルラグルシブの経口剤形

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2446269T3 (es) 2006-12-19 2014-03-06 The Board Of Trustees Of The University Of Illinois 3-Benzofuranil-4-indolil-maleimidas como potentes inhibidores de GSK-3 para trastornos neurodegenerativos
MY156701A (en) 2009-12-23 2016-03-15 Arqule Inc Purified pyrroloquinolinyl-pyrrolidine-2,5-dione compositions and methods for preparing and using same

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