JP2023100974A5 - - Google Patents
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- Publication number
- JP2023100974A5 JP2023100974A5 JP2023079468A JP2023079468A JP2023100974A5 JP 2023100974 A5 JP2023100974 A5 JP 2023100974A5 JP 2023079468 A JP2023079468 A JP 2023079468A JP 2023079468 A JP2023079468 A JP 2023079468A JP 2023100974 A5 JP2023100974 A5 JP 2023100974A5
- Authority
- JP
- Japan
- Prior art keywords
- degrees
- composition
- polymorph
- skin disorder
- further exhibiting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 239000000203 mixture Substances 0.000 claims 15
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical compound OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 claims 3
- 230000001747 exhibiting effect Effects 0.000 claims 3
- -1 pomade Substances 0.000 claims 3
- 208000017520 skin disease Diseases 0.000 claims 3
- 102000003702 retinoic acid receptors Human genes 0.000 claims 2
- 108090000064 retinoic acid receptors Proteins 0.000 claims 2
- MFBCDACCJCDGBA-UHFFFAOYSA-N 4-[3-(3-tert-butyl-4-pyrrolidin-1-ylphenyl)-4-(2-hydroxyethoxy)phenyl]benzoic acid Chemical compound CC(C)(C)C1=CC(C=2C(=CC=C(C=2)C=2C=CC(=CC=2)C(O)=O)OCCO)=CC=C1N1CCCC1 MFBCDACCJCDGBA-UHFFFAOYSA-N 0.000 claims 1
- 208000002874 Acne Vulgaris Diseases 0.000 claims 1
- 241000195940 Bryophyta Species 0.000 claims 1
- 206010000496 acne Diseases 0.000 claims 1
- 238000004140 cleaning Methods 0.000 claims 1
- 150000001875 compounds Chemical class 0.000 claims 1
- 239000006071 cream Substances 0.000 claims 1
- 239000000499 gel Substances 0.000 claims 1
- 230000001404 mediated effect Effects 0.000 claims 1
- 239000008267 milk Substances 0.000 claims 1
- 210000004080 milk Anatomy 0.000 claims 1
- 235000013336 milk Nutrition 0.000 claims 1
- 235000011929 mousse Nutrition 0.000 claims 1
- 239000002674 ointment Substances 0.000 claims 1
- 230000037361 pathway Effects 0.000 claims 1
- 239000000546 pharmaceutical excipient Substances 0.000 claims 1
- 239000000843 powder Substances 0.000 claims 1
- 238000000634 powder X-ray diffraction Methods 0.000 claims 1
- 239000002453 shampoo Substances 0.000 claims 1
- 239000000243 solution Substances 0.000 claims 1
- 239000007921 spray Substances 0.000 claims 1
- 239000000725 suspension Substances 0.000 claims 1
- 239000000271 synthetic detergent Substances 0.000 claims 1
- 230000000699 topical effect Effects 0.000 claims 1
- 229950008964 trifarotene Drugs 0.000 claims 1
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025188194A JP2026016786A (ja) | 2019-12-11 | 2025-11-07 | トリファロテンならびにその中間体および多形体の調製 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962946943P | 2019-12-11 | 2019-12-11 | |
| US62/946,943 | 2019-12-11 | ||
| JP2022534812A JP7281016B2 (ja) | 2019-12-11 | 2020-12-10 | トリファロテンならびにその中間体および多形体の調製 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022534812A Division JP7281016B2 (ja) | 2019-12-11 | 2020-12-10 | トリファロテンならびにその中間体および多形体の調製 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025188194A Division JP2026016786A (ja) | 2019-12-11 | 2025-11-07 | トリファロテンならびにその中間体および多形体の調製 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2023100974A JP2023100974A (ja) | 2023-07-19 |
| JP2023100974A5 true JP2023100974A5 (https=) | 2023-12-15 |
Family
ID=74141909
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022534812A Active JP7281016B2 (ja) | 2019-12-11 | 2020-12-10 | トリファロテンならびにその中間体および多形体の調製 |
| JP2023079468A Pending JP2023100974A (ja) | 2019-12-11 | 2023-05-12 | トリファロテンならびにその中間体および多形体の調製 |
| JP2025188194A Pending JP2026016786A (ja) | 2019-12-11 | 2025-11-07 | トリファロテンならびにその中間体および多形体の調製 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022534812A Active JP7281016B2 (ja) | 2019-12-11 | 2020-12-10 | トリファロテンならびにその中間体および多形体の調製 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025188194A Pending JP2026016786A (ja) | 2019-12-11 | 2025-11-07 | トリファロテンならびにその中間体および多形体の調製 |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US11691946B2 (https=) |
| EP (2) | EP4073035B1 (https=) |
| JP (3) | JP7281016B2 (https=) |
| CN (1) | CN114787129B (https=) |
| AU (2) | AU2020402049B2 (https=) |
| CA (1) | CA3161509A1 (https=) |
| ES (1) | ES3037292T3 (https=) |
| IL (2) | IL293800B2 (https=) |
| WO (1) | WO2021119351A1 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL293800B2 (en) * | 2019-12-11 | 2024-10-01 | Taro Pharma Ind | Preparation of trifarotene and intermediates and polymorphs thereof |
| CN117342993A (zh) * | 2022-07-05 | 2024-01-05 | 石家庄迪斯凯威医药科技有限公司 | 一种曲法罗汀盐及其药物组合物和用途 |
| CN115745913B (zh) * | 2022-09-16 | 2024-05-24 | 南京迈诺威医药科技有限公司 | 曲法罗汀多晶型及其制备方法 |
| JP2026507122A (ja) * | 2023-02-28 | 2026-02-27 | タロー・ファーマシューティカル・インダストリーズ・リミテッド | トリファロテンを調製する方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1248869A2 (en) * | 2000-01-07 | 2002-10-16 | Transform Pharmaceuticals, Inc. | High-throughput formation, identification, and analysis of diverse solid-forms |
| WO2004083335A2 (en) * | 2003-03-21 | 2004-09-30 | University Of Rochester | Glassy chiral-nematic liquid crystals and optical devices containing same |
| US8354427B2 (en) | 2004-06-24 | 2013-01-15 | Vertex Pharmaceutical Incorporated | Modulators of ATP-binding cassette transporters |
| DK1817301T3 (da) * | 2004-11-22 | 2012-02-27 | Lilly Co Eli | Forstærkere af glutamat-receptorer |
| PL1831149T3 (pl) * | 2004-12-23 | 2012-06-29 | Galderma Res & Dev | Nowe ligandy, które modulują receptory RAR, i ich zastosowanie w medycynie i kosmetyce |
| GB2426247A (en) | 2005-05-20 | 2006-11-22 | Arrow Int Ltd | Methods of preparing purine derivatives such as famciclovir |
| EP3475312B1 (en) * | 2016-06-23 | 2020-05-27 | Galderma S.A. | Cyclodextrin-grafted cross-linked hyaluronic acid complexed with active drug substances and uses thereof |
| IL293800B2 (en) * | 2019-12-11 | 2024-10-01 | Taro Pharma Ind | Preparation of trifarotene and intermediates and polymorphs thereof |
-
2020
- 2020-12-10 IL IL293800A patent/IL293800B2/en unknown
- 2020-12-10 JP JP2022534812A patent/JP7281016B2/ja active Active
- 2020-12-10 AU AU2020402049A patent/AU2020402049B2/en active Active
- 2020-12-10 EP EP20838774.6A patent/EP4073035B1/en active Active
- 2020-12-10 EP EP25166751.5A patent/EP4552691A3/en active Pending
- 2020-12-10 ES ES20838774T patent/ES3037292T3/es active Active
- 2020-12-10 IL IL312356A patent/IL312356A/en unknown
- 2020-12-10 CA CA3161509A patent/CA3161509A1/en active Pending
- 2020-12-10 CN CN202080085458.5A patent/CN114787129B/zh active Active
- 2020-12-10 WO PCT/US2020/064365 patent/WO2021119351A1/en not_active Ceased
- 2020-12-10 US US17/756,994 patent/US11691946B2/en active Active
-
2023
- 2023-05-12 JP JP2023079468A patent/JP2023100974A/ja active Pending
- 2023-05-12 US US18/316,742 patent/US20230278956A1/en active Pending
- 2023-09-01 AU AU2023222982A patent/AU2023222982B2/en active Active
-
2025
- 2025-11-07 JP JP2025188194A patent/JP2026016786A/ja active Pending
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