JP2022545005A5 - - Google Patents

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Publication number
JP2022545005A5
JP2022545005A5 JP2022511096A JP2022511096A JP2022545005A5 JP 2022545005 A5 JP2022545005 A5 JP 2022545005A5 JP 2022511096 A JP2022511096 A JP 2022511096A JP 2022511096 A JP2022511096 A JP 2022511096A JP 2022545005 A5 JP2022545005 A5 JP 2022545005A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
composition according
cancer
egfr
kras
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2022511096A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022545005A (ja
JP7602272B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/047090 external-priority patent/WO2021034992A1/en
Publication of JP2022545005A publication Critical patent/JP2022545005A/ja
Publication of JP2022545005A5 publication Critical patent/JP2022545005A5/ja
Application granted granted Critical
Publication of JP7602272B2 publication Critical patent/JP7602272B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022511096A 2019-08-22 2020-08-20 Kras関連がんを治療する方法 Active JP7602272B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962890119P 2019-08-22 2019-08-22
US62/890,119 2019-08-22
PCT/US2020/047090 WO2021034992A1 (en) 2019-08-22 2020-08-20 Method of treating kras-associated cancers

Publications (3)

Publication Number Publication Date
JP2022545005A JP2022545005A (ja) 2022-10-24
JP2022545005A5 true JP2022545005A5 (https=) 2023-08-28
JP7602272B2 JP7602272B2 (ja) 2024-12-18

Family

ID=74660044

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022511096A Active JP7602272B2 (ja) 2019-08-22 2020-08-20 Kras関連がんを治療する方法

Country Status (11)

Country Link
US (1) US20220273643A1 (https=)
EP (1) EP4017489B1 (https=)
JP (1) JP7602272B2 (https=)
KR (1) KR20220050143A (https=)
CN (2) CN119454706A (https=)
AU (1) AU2020334069B2 (https=)
BR (1) BR112022003165A2 (https=)
CA (1) CA3150759A1 (https=)
IL (1) IL290454B2 (https=)
MX (1) MX2022002108A (https=)
WO (1) WO2021034992A1 (https=)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2019217307A1 (en) 2018-05-07 2019-11-14 Mirati Therapeutics, Inc. Kras g12c inhibitors
EP3849537B1 (en) 2018-09-10 2024-10-23 Mirati Therapeutics, Inc. Combination therapies
EA202190749A1 (ru) 2018-09-10 2021-07-09 Мирати Терапьютикс, Инк. Способы комбинированной терапии
EP3849535A4 (en) 2018-09-10 2022-06-29 Mirati Therapeutics, Inc. Combination therapies
JP2022500385A (ja) 2018-09-10 2022-01-04 ミラティ セラピューティクス, インコーポレイテッド 組み合わせ療法
MX2021002804A (es) 2018-12-05 2021-07-15 Mirati Therapeutics Inc Terapias de combinacion.
EP3908283A4 (en) 2019-01-10 2022-10-12 Mirati Therapeutics, Inc. KRAS G12C INHIBITORS
MX2022002465A (es) 2019-08-29 2022-05-19 Mirati Therapeutics Inc Inhibidores de kras g12d.
WO2021061749A1 (en) 2019-09-24 2021-04-01 Mirati Therapeutics, Inc. Combination therapies
PH12022551513A1 (en) 2019-12-20 2023-04-24 Mirati Therapeutics Inc Sos1 inhibitors
EP4210833A4 (en) 2020-09-11 2024-09-11 Mirati Therapeutics, Inc. CRYSTALLINE FORMS OF A KRAS G12C INHIBITOR
JP2023553492A (ja) 2020-12-15 2023-12-21 ミラティ セラピューティクス, インコーポレイテッド アザキナゾリン汎KRas阻害剤
EP4262803A4 (en) 2020-12-16 2025-03-12 Mirati Therapeutics, Inc. Tetrahydropyridopyrimidine pan-kras inhibitors
CA3214172A1 (en) * 2021-04-02 2022-10-06 Mukesh K. Nyati Combination therapy for cancer treatment
WO2023003417A1 (ko) * 2021-07-22 2023-01-26 국립암센터 Kras 돌연변이 특이적 저해제 및 이를 포함하는 암 예방 또는 치료용 조성물

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5466468A (en) 1990-04-03 1995-11-14 Ciba-Geigy Corporation Parenterally administrable liposome formulation comprising synthetic lipids
CA2612183C (en) * 2005-06-28 2015-08-11 Genentech, Inc. Egfr and kras mutations
WO2010114922A1 (en) * 2009-03-31 2010-10-07 Agios Pharmaceuticals, Inc. Methods of treating cancer having an aberrant egfr or kras genotype
WO2012064642A1 (en) * 2010-11-08 2012-05-18 Glaxosmithkline Llc Fatty acid synthase inhibitors
US20140256767A1 (en) 2011-10-31 2014-09-11 The Broad Institute, Inc. Direct inhibitors of keap1-nrf2 interaction as antioxidant inflammation modulators
WO2014176475A2 (en) 2013-04-26 2014-10-30 The Regents Of The University Of Michigan Egfr inhibitors and uses thereof
EP3755323A4 (en) * 2018-02-23 2021-11-24 The Regents Of The University Of Michigan EGFR DIMER DISRUPTORS AND THEIR USES

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