JP2022544536A5 - - Google Patents

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Publication number
JP2022544536A5
JP2022544536A5 JP2022509051A JP2022509051A JP2022544536A5 JP 2022544536 A5 JP2022544536 A5 JP 2022544536A5 JP 2022509051 A JP2022509051 A JP 2022509051A JP 2022509051 A JP2022509051 A JP 2022509051A JP 2022544536 A5 JP2022544536 A5 JP 2022544536A5
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JP
Japan
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JP2022509051A
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Japanese (ja)
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JP7583027B2 (ja
JP2022544536A (ja
JPWO2021034627A5 (https=
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Priority claimed from PCT/US2020/046269 external-priority patent/WO2021034627A1/en
Publication of JP2022544536A publication Critical patent/JP2022544536A/ja
Publication of JP2022544536A5 publication Critical patent/JP2022544536A5/ja
Publication of JPWO2021034627A5 publication Critical patent/JPWO2021034627A5/ja
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Publication of JP7583027B2 publication Critical patent/JP7583027B2/ja
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JP2022509051A 2019-08-16 2020-08-14 プロテアソームのコア粒子の低分子刺激物質 Active JP7583027B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962887732P 2019-08-16 2019-08-16
US62/887,732 2019-08-16
PCT/US2020/046269 WO2021034627A1 (en) 2019-08-16 2020-08-14 Small molecule stimulators of the core particle of the proteasome

Publications (4)

Publication Number Publication Date
JP2022544536A JP2022544536A (ja) 2022-10-19
JP2022544536A5 true JP2022544536A5 (https=) 2023-06-15
JPWO2021034627A5 JPWO2021034627A5 (https=) 2023-06-15
JP7583027B2 JP7583027B2 (ja) 2024-11-13

Family

ID=74659522

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JP2022509051A Active JP7583027B2 (ja) 2019-08-16 2020-08-14 プロテアソームのコア粒子の低分子刺激物質

Country Status (5)

Country Link
US (1) US20220267280A1 (https=)
EP (1) EP4013405A4 (https=)
JP (1) JP7583027B2 (https=)
CN (1) CN114222573A (https=)
WO (1) WO2021034627A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113620881A (zh) * 2021-08-12 2021-11-09 浙江禾本科技股份有限公司 一种1-[2-(2,4-二氯苯基)-2羟基乙基]-1h咪唑的合成方法
WO2023036936A1 (en) 2021-09-09 2023-03-16 Booster Therapeutics Gmbh Bifunctional molecules as proteasome stimulators for improved targeted protein degradation, and their uses as targeted boosting degraders (tarbods)
EP4147723A1 (en) 2021-09-09 2023-03-15 Booster Therapeutics GmbH Bifunctional molecules as proteasome stimulators for improved targeted protein degradation, and their uses as targeted boosting degraders (tarbods)
WO2025219559A1 (en) 2024-04-18 2025-10-23 Booster Therapeutics Gmbh Pyrrolidine compounds as proteasome stimulators

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU557755A3 (ru) * 1968-08-19 1977-05-05 Янссен Фармасьютика Н.В. (Фирма) Способ получени производных имидазола
US3991202A (en) * 1974-01-31 1976-11-09 Janssen Pharmaceutica N.V. Imidazolium salts
US5633274A (en) * 1993-02-18 1997-05-27 President And Fellows Of Harvard College Cancer treatments
EP0829478A3 (en) * 1996-09-09 1998-03-25 F. Hoffmann-La Roche Ag N-Benzylimidazolium and N-benzyltriazolium derivatives, their preparation and their use as antifungal and antimycotic agents
NZ328607A (en) * 1996-09-09 1999-08-30 Hoffmann La Roche Heterocyclically substituted n-benzyl-azolium derivatives and fungicidal compositions
JPWO2004022546A1 (ja) * 2002-09-04 2006-03-02 敬銘 王 ジャスモン酸の生合成を阻害する物質
MX2007016186A (es) * 2005-06-14 2008-03-07 Schering Corp Preparacion y uso de inhibidores de proteasas.
BRPI0904249B1 (pt) * 2009-08-28 2018-03-06 Biolab Sanus Farmacêutica Ltda. Compostos éteres aralquil benzílicos, processo de preparação dos mesmos, uso dos referidos compostos, composição farmacêutica
US11197862B2 (en) * 2015-07-16 2021-12-14 Xomics Biopharma, Inc. Methods of preventing toxicity of platinum drugs

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