JP2022535743A5 - - Google Patents

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Publication number
JP2022535743A5
JP2022535743A5 JP2021570361A JP2021570361A JP2022535743A5 JP 2022535743 A5 JP2022535743 A5 JP 2022535743A5 JP 2021570361 A JP2021570361 A JP 2021570361A JP 2021570361 A JP2021570361 A JP 2021570361A JP 2022535743 A5 JP2022535743 A5 JP 2022535743A5
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JP
Japan
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ring
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Pending
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JP2021570361A
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English (en)
Japanese (ja)
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JP2022535743A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/035249 external-priority patent/WO2020243519A1/en
Publication of JP2022535743A publication Critical patent/JP2022535743A/ja
Publication of JP2022535743A5 publication Critical patent/JP2022535743A5/ja
Pending legal-status Critical Current

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JP2021570361A 2019-05-29 2020-05-29 Sting活性に関連する状態を治療するための化合物および組成物 Pending JP2022535743A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962854288P 2019-05-29 2019-05-29
US62/854,288 2019-05-29
PCT/US2020/035249 WO2020243519A1 (en) 2019-05-29 2020-05-29 Compounds and compositions for treating conditions associated with sting activity

Publications (2)

Publication Number Publication Date
JP2022535743A JP2022535743A (ja) 2022-08-10
JP2022535743A5 true JP2022535743A5 (enExample) 2023-06-01

Family

ID=71787083

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021570361A Pending JP2022535743A (ja) 2019-05-29 2020-05-29 Sting活性に関連する状態を治療するための化合物および組成物

Country Status (5)

Country Link
US (1) US20220227760A1 (enExample)
EP (1) EP3976584A1 (enExample)
JP (1) JP2022535743A (enExample)
MA (1) MA56047A (enExample)
WO (1) WO2020243519A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN120004785A (zh) 2018-07-03 2025-05-16 诺华制药股份有限公司 用于治疗与sting活性有关的疾病的化合物和组合物
TW202200136A (zh) 2020-04-10 2022-01-01 日商小野藥品工業股份有限公司 癌治療方法
JP2023554393A (ja) * 2020-12-16 2023-12-27 アイエフエム デュー インコーポレイテッド Sting活性に関連する状態を治療するための化合物および組成物
US20240051970A1 (en) * 2020-12-16 2024-02-15 Ifm Due, Inc. Compounds and compositions for treating conditions associated with sting activity
EP4267129A1 (en) 2020-12-22 2023-11-01 IFM Due, Inc. Methods of treating cancer
EP4267128A1 (en) 2020-12-22 2023-11-01 IFM Due, Inc. Methods of treating cancer
JP2024500874A (ja) 2020-12-22 2024-01-10 アイエフエム デュー インコーポレイテッド がんを処置する方法
US20240060982A1 (en) * 2020-12-22 2024-02-22 Ifm Due, Inc. Methods of treating cancer
EP4274824A1 (en) 2021-01-08 2023-11-15 IFM Due, Inc. Heterobicyclic compounds having an urea or analogue and their compositions for treating conditions associated with sting activity
IL310724A (en) 2021-08-10 2024-04-01 Ifm Due Inc COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF CONDITIONS ASSOCIATED WITH STING ACTIVITY
WO2024064358A1 (en) 2022-09-23 2024-03-28 Ifm Due, Inc. Compounds and compositions for treating conditions associated with sting activity

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002022605A1 (en) * 2000-09-15 2002-03-21 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
UA95244C2 (ru) * 2005-06-22 2011-07-25 Плексикон, Инк. Соединения и способ модулирования активности киназ, и показания для их применения
CN102812023A (zh) * 2010-01-13 2012-12-05 韩国巴斯德研究所 抗感染吡啶并(1,2-a)嘧啶类
US8497285B2 (en) 2010-12-03 2013-07-30 The Trustees Of The University Of Pennsylvania Therapy of autoimmune colitis using a TIP60 inhibitor
JP6121658B2 (ja) * 2011-06-29 2017-04-26 大塚製薬株式会社 治療用化合物、及び関連する使用の方法
US9260426B2 (en) * 2012-12-14 2016-02-16 Arrien Pharmaceuticals Llc Substituted 1H-pyrrolo [2, 3-b] pyridine and 1H-pyrazolo [3, 4-b] pyridine derivatives as salt inducible kinase 2 (SIK2) inhibitors
PE20160080A1 (es) 2013-05-18 2016-02-21 Aduro Biotech Inc Composiciones y metodos para activar la senalizacion que depende del estimulador del gen de interferon
CA2927009C (en) 2013-10-21 2019-04-23 Drexel University Use of sting agonists to treat chronic hepatitis b virus infection
WO2015131005A1 (en) * 2014-02-28 2015-09-03 The Regents Of The University Of Michigan 9h-pyrimido[4,5-b]indoles and related analogs as bet bromodomain inhibitors
EP3632915A1 (en) * 2014-11-27 2020-04-08 Genentech, Inc. 4,5,6,7-tetrahydro-1 h-pyrazolo[4,3-c]pyridin-3-amine compounds as cbp and/or ep300 inhibitors
JP7636322B2 (ja) * 2018-11-15 2025-02-26 アンスティテュ・ギュスターヴ・ルシー 癌を処置するためのマドラシン誘導体化合物、組成物およびこれらの使用
JP2022507697A (ja) * 2018-11-19 2022-01-18 アイエフエム デュー インコーポレイテッド Sting活性に関連する状態を治療するための化合物および組成物

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