JP2022533433A5 - - Google Patents
Info
- Publication number
- JP2022533433A5 JP2022533433A5 JP2021569359A JP2021569359A JP2022533433A5 JP 2022533433 A5 JP2022533433 A5 JP 2022533433A5 JP 2021569359 A JP2021569359 A JP 2021569359A JP 2021569359 A JP2021569359 A JP 2021569359A JP 2022533433 A5 JP2022533433 A5 JP 2022533433A5
- Authority
- JP
- Japan
- Prior art keywords
- etoh
- methanesulfonylphenoxy
- fluoro
- propyl
- ethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP19176514 | 2019-05-24 | ||
| EP19176514.8 | 2019-05-24 | ||
| EP20166361 | 2020-03-27 | ||
| EP20166361.4 | 2020-03-27 | ||
| PCT/EP2020/064046 WO2020239568A1 (en) | 2019-05-24 | 2020-05-20 | Pharmaceutically acceptable salts of [2-(3-fluoro-5-methane-sulfonylphenoxy)ethyl](propyl)amine and uses thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2022533433A JP2022533433A (ja) | 2022-07-22 |
| JP2022533433A5 true JP2022533433A5 (https=) | 2023-05-29 |
| JP7623958B2 JP7623958B2 (ja) | 2025-01-29 |
Family
ID=70682855
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021569359A Active JP7623958B2 (ja) | 2019-05-24 | 2020-05-20 | [2-(3-フルオロ-5-メタンスルホニルフェノキシ)エチル](プロピル)アミンの薬学的に許容される塩、およびその使用 |
Country Status (21)
| Country | Link |
|---|---|
| US (2) | US12275694B2 (https=) |
| EP (2) | EP3976581B1 (https=) |
| JP (1) | JP7623958B2 (https=) |
| KR (1) | KR102892833B1 (https=) |
| CN (1) | CN113853369B (https=) |
| AU (1) | AU2020286003B2 (https=) |
| BR (1) | BR112021023563A2 (https=) |
| CA (1) | CA3140805A1 (https=) |
| CL (1) | CL2021003115A1 (https=) |
| CO (1) | CO2021016556A2 (https=) |
| DK (1) | DK3976581T3 (https=) |
| ES (1) | ES2970361T3 (https=) |
| FI (1) | FI3976581T3 (https=) |
| IL (1) | IL288271B2 (https=) |
| JO (1) | JOP20210312A1 (https=) |
| MX (1) | MX2021014271A (https=) |
| PH (1) | PH12021552844A1 (https=) |
| PL (1) | PL3976581T3 (https=) |
| PT (1) | PT3976581T (https=) |
| SG (1) | SG11202112165QA (https=) |
| WO (1) | WO2020239568A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR112021023563A2 (pt) | 2019-05-24 | 2022-01-04 | Integrative Res Laboratories Sweden Ab | Sais farmaceuticamente aceitáveis de [2-(3-fluoro-5-metano-sulfonilfenóxi)etil](propil) amina e usos dos mesmos |
| TW202233169A (zh) * | 2020-11-10 | 2022-09-01 | 瑞典商瑞典綜合研究實驗室公司 | 包含[2-(3-氟-5-甲磺醯苯氧基)乙基](丙基)胺之醫藥上可接受鹽類的醫藥組成物、及治療帕金森氏症的藥物及所述醫藥組成物的用途 |
| EP4577201A1 (en) * | 2022-08-24 | 2025-07-02 | Alkem Laboratories Limited | Mesdopetam compositions |
| EP4590657A1 (en) | 2022-09-21 | 2025-07-30 | Assia Chemical Industries Ltd. | Solid state forms of mesdopetam and salts therof |
| GB202312055D0 (en) | 2023-08-07 | 2023-09-20 | Ipsen Biopharm Ltd | Pharmaceutical compositions |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS51123821A (en) | 1975-04-18 | 1976-10-28 | Nippon Kayaku Co Ltd | An algicide and protective agent |
| US4128574A (en) * | 1976-10-04 | 1978-12-05 | General Electric Company | Method for making organic polycarboxylic acids |
| GB8823405D0 (en) | 1988-10-05 | 1988-11-09 | Erba Carlo Spa | Aryloxy-arythio-heteraryloxy-heteroarylthio-alkenylene derivatives of amines |
| ATE210657T1 (de) | 1994-10-14 | 2001-12-15 | Merck Patent Gmbh | Zns wirksames (r)-(-)-2-(5-(4-fluorophenyl)-3- pyridylmethylaminomethyl)chroman |
| SE9904723D0 (sv) * | 1999-12-22 | 1999-12-22 | Carlsson A Research Ab | New modulators of dopamine neurotransmission II |
| DOP2001000189A (es) | 2000-06-30 | 2002-03-30 | Pfizer Prod Inc | Benzofenonas y sulfonas como inhibidores de la captación de glicina |
| JP2006193494A (ja) | 2005-01-17 | 2006-07-27 | Dainippon Ink & Chem Inc | 4級アンモニウム系化合物を有効成分とする心臓疾患治療剤 |
| US20100069346A1 (en) | 2005-06-23 | 2010-03-18 | Sara Holmqvist | New Azetidine Derivatives as Neurokinin Receptor Antagonists for the Treatment of Gastrointestinal Diseases |
| JP5210637B2 (ja) | 2005-11-29 | 2013-06-12 | キッセイ薬品工業株式会社 | 新規なカテコール誘導体、それを含有する医薬組成物およびそれらの用途 |
| WO2007072041A1 (en) | 2005-12-23 | 2007-06-28 | Astex Therapeutics Limited | Therapeutic compounds |
| ATE534638T1 (de) * | 2006-02-15 | 2011-12-15 | Ms Science Corp | Piperazin-derivate |
| CA2687721A1 (en) * | 2007-06-08 | 2008-12-18 | Arena Pharmaceuticals, Inc. | Crystalline forms of (r)-1-{2-[4'-(3-methoxy-propane-1-sulfonyl)-biphenyl-4-yl]-ethyl}-2-methyl-pyrrolidine, and compositions, and methods related thereto |
| TW200932225A (en) * | 2007-12-14 | 2009-08-01 | Lundbeck & Co As H | 4-[2,3-difluoro-6-(2-fluoro-4-methyl-phenylsulfanyl)-phenyl]-piperidine |
| JP2011519839A (ja) | 2008-04-29 | 2011-07-14 | エヌエスエイビー、フィリアル アヴ ノイロサーチ スウェーデン エービー、スヴェーリエ | ドーパミン神経伝達のモジュレーター |
| MX2010011724A (es) | 2008-04-29 | 2010-11-30 | Nsab Af Neurosearch Sweden Ab | Moduladores de neurotransmision de dopamina. |
| EP2271638B1 (en) | 2008-04-29 | 2011-08-31 | NSAB, Filial af NeuroSearch Sweden AB, Sverige | Modulators of dopamine neurotransmission |
| EP2699543B1 (en) * | 2011-04-19 | 2016-03-02 | Integrative Research Laboratories Sweden AB | Novel modulators of cortical dopaminergic- and nmda-receptor-mediated glutamatergic neurotransmission |
| MX2017008136A (es) | 2014-12-22 | 2018-03-06 | Teva Pharmaceuticals Int Gmbh | Sal de l-tartrato de pridopidina. |
| CN117304079A (zh) | 2016-02-08 | 2023-12-29 | 默克专利股份有限公司 | N-(4,5-双甲磺酰基-2-甲基苯甲酰基)胍盐酸盐和n-(4,5-双甲磺酰基-2-甲基苯甲酰基)胍盐的结晶变体 |
| EP3625213B1 (en) | 2017-05-19 | 2023-03-08 | Integrative Research Laboratories Sweden AB | (+)-3-(2,3-difluorophenyl)-3-methoxypyrrolidine fumarate, a process for its preparation and uses thereof |
| ES2874628T3 (es) * | 2017-08-07 | 2021-11-05 | Suven Life Sciences Ltd | Compuestos de fluoropiperidina como antagonistas puros del receptor 5-HT6 |
| WO2020110128A1 (en) | 2018-11-29 | 2020-06-04 | Prilenia Neurotherapeutics Ltd. | Combination of pridopidine and an additional therapeutic agent for treating drug induced dyskinesia |
| BR112021023563A2 (pt) | 2019-05-24 | 2022-01-04 | Integrative Res Laboratories Sweden Ab | Sais farmaceuticamente aceitáveis de [2-(3-fluoro-5-metano-sulfonilfenóxi)etil](propil) amina e usos dos mesmos |
-
2020
- 2020-05-20 BR BR112021023563A patent/BR112021023563A2/pt unknown
- 2020-05-20 ES ES20725728T patent/ES2970361T3/es active Active
- 2020-05-20 SG SG11202112165QA patent/SG11202112165QA/en unknown
- 2020-05-20 DK DK20725728.8T patent/DK3976581T3/da active
- 2020-05-20 KR KR1020217037818A patent/KR102892833B1/ko active Active
- 2020-05-20 EP EP20725728.8A patent/EP3976581B1/en active Active
- 2020-05-20 US US17/612,902 patent/US12275694B2/en active Active
- 2020-05-20 CN CN202080036829.0A patent/CN113853369B/zh active Active
- 2020-05-20 EP EP23190702.3A patent/EP4292653B1/en active Active
- 2020-05-20 PT PT207257288T patent/PT3976581T/pt unknown
- 2020-05-20 PL PL20725728.8T patent/PL3976581T3/pl unknown
- 2020-05-20 AU AU2020286003A patent/AU2020286003B2/en active Active
- 2020-05-20 WO PCT/EP2020/064046 patent/WO2020239568A1/en not_active Ceased
- 2020-05-20 MX MX2021014271A patent/MX2021014271A/es unknown
- 2020-05-20 PH PH1/2021/552844A patent/PH12021552844A1/en unknown
- 2020-05-20 CA CA3140805A patent/CA3140805A1/en active Pending
- 2020-05-20 FI FIEP20725728.8T patent/FI3976581T3/fi active
- 2020-05-20 IL IL288271A patent/IL288271B2/en unknown
- 2020-05-20 JP JP2021569359A patent/JP7623958B2/ja active Active
-
2021
- 2021-11-24 CL CL2021003115A patent/CL2021003115A1/es unknown
- 2021-11-24 JO JOP/2021/0312A patent/JOP20210312A1/ar unknown
- 2021-12-06 CO CONC2021/0016556A patent/CO2021016556A2/es unknown
-
2025
- 2025-03-14 US US19/080,430 patent/US20250243155A1/en active Pending
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