JP2022527270A5 - - Google Patents

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Publication number
JP2022527270A5
JP2022527270A5 JP2021557231A JP2021557231A JP2022527270A5 JP 2022527270 A5 JP2022527270 A5 JP 2022527270A5 JP 2021557231 A JP2021557231 A JP 2021557231A JP 2021557231 A JP2021557231 A JP 2021557231A JP 2022527270 A5 JP2022527270 A5 JP 2022527270A5
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JP
Japan
Prior art keywords
pharmaceutical composition
disease
pharmaceutical
combination
disorder
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JP2021557231A
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English (en)
Japanese (ja)
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JP7461369B2 (ja
JP2022527270A (ja
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Priority claimed from PCT/IB2020/052825 external-priority patent/WO2020194209A1/en
Publication of JP2022527270A publication Critical patent/JP2022527270A/ja
Publication of JP2022527270A5 publication Critical patent/JP2022527270A5/ja
Application granted granted Critical
Publication of JP7461369B2 publication Critical patent/JP7461369B2/ja
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JP2021557231A 2019-03-26 2020-03-25 イソチアゾリジン1,1-ジオキシド及び1,4-ブタンスルトン含有ラパマイシン誘導体並びにその使用 Active JP7461369B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962824190P 2019-03-26 2019-03-26
US62/824,190 2019-03-26
PCT/IB2020/052825 WO2020194209A1 (en) 2019-03-26 2020-03-25 Isothiazolidine 1,1-dioxide and 1,4-butan sultone containing rapamycin derivatives and uses thereof

Publications (3)

Publication Number Publication Date
JP2022527270A JP2022527270A (ja) 2022-06-01
JP2022527270A5 true JP2022527270A5 (https=) 2023-04-03
JP7461369B2 JP7461369B2 (ja) 2024-04-03

Family

ID=70190042

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021557231A Active JP7461369B2 (ja) 2019-03-26 2020-03-25 イソチアゾリジン1,1-ジオキシド及び1,4-ブタンスルトン含有ラパマイシン誘導体並びにその使用

Country Status (20)

Country Link
US (1) US20220202787A1 (https=)
EP (1) EP3947392B1 (https=)
JP (1) JP7461369B2 (https=)
KR (1) KR20210142689A (https=)
CN (1) CN113614090B (https=)
AU (1) AU2020250026B2 (https=)
BR (1) BR112021018692A2 (https=)
CA (1) CA3134653A1 (https=)
DK (1) DK3947392T3 (https=)
ES (1) ES2987625T3 (https=)
FI (1) FI3947392T3 (https=)
HR (1) HRP20240633T1 (https=)
HU (1) HUE067396T2 (https=)
LT (1) LT3947392T (https=)
MX (1) MX2021011376A (https=)
PL (1) PL3947392T3 (https=)
PT (1) PT3947392T (https=)
RS (1) RS65531B1 (https=)
SI (1) SI3947392T1 (https=)
WO (1) WO2020194209A1 (https=)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR112834A1 (es) 2017-09-26 2019-12-18 Novartis Ag Derivados de rapamicina
WO2019241789A1 (en) 2018-06-15 2019-12-19 Navitor Pharmaceuticals, Inc. Rapamycin analogs and uses thereof
HRP20250197T1 (hr) 2018-12-18 2025-04-11 Novartis Ag Derivati rapamicina
AU2020397938A1 (en) 2019-12-05 2022-06-23 Janssen Pharmaceutica Nv Rapamycin analogs and uses thereof
JP2023028473A (ja) * 2021-08-19 2023-03-03 日本マイクロバイオファーマ株式会社 エベロリムスの製造方法
GB202415232D0 (en) 2024-10-16 2024-11-27 Nacamed As Composition

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA737247B (en) 1972-09-29 1975-04-30 Ayerst Mckenna & Harrison Rapamycin and process of preparation
ZA935112B (en) * 1992-07-17 1994-02-08 Smithkline Beecham Corp Rapamycin derivatives
CA2257803C (en) * 1996-07-12 2008-12-02 Ariad Pharmaceuticals, Inc. Non immunosuppressive antifungal rapalogs
ATE264863T1 (de) * 1999-08-24 2004-05-15 Ariad Gene Therapeutics Inc 28-epirapaloge
US20090023768A1 (en) * 2006-02-24 2009-01-22 Novartis Ag Rapamycin derivatives for treating neuroblastoma
JP6130391B2 (ja) 2011-11-23 2017-05-17 インテリカイン, エルエルシー Mtor阻害剤を使用する強化された治療レジメン
US10683308B2 (en) * 2015-09-11 2020-06-16 Navitor Pharmaceuticals, Inc. Rapamycin analogs and uses thereof
AR112834A1 (es) * 2017-09-26 2019-12-18 Novartis Ag Derivados de rapamicina

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